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DK1223933T3 - 5-leddet derivater af heterocyklusser og deres anvendelse som monoaminoxidaseinhibitorer - Google Patents

5-leddet derivater af heterocyklusser og deres anvendelse som monoaminoxidaseinhibitorer

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Publication number
DK1223933T3
DK1223933T3 DK00967988T DK00967988T DK1223933T3 DK 1223933 T3 DK1223933 T3 DK 1223933T3 DK 00967988 T DK00967988 T DK 00967988T DK 00967988 T DK00967988 T DK 00967988T DK 1223933 T3 DK1223933 T3 DK 1223933T3
Authority
DK
Denmark
Prior art keywords
heterocycles
monoamine oxidase
oxidase inhibitors
membered derivatives
membered
Prior art date
Application number
DK00967988T
Other languages
English (en)
Inventor
De Lassauniere Pierre Chabrier
Jeremiah Harnett
Dennis Bigg
Jacques Pommier
Anne-Marie Liberatore
Christophe Thurieau
Jacques Lannoy
Original Assignee
Sod Conseils Rech Applic
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9912643A external-priority patent/FR2799461B1/fr
Priority claimed from FR0010151A external-priority patent/FR2812546B1/fr
Application filed by Sod Conseils Rech Applic filed Critical Sod Conseils Rech Applic
Application granted granted Critical
Publication of DK1223933T3 publication Critical patent/DK1223933T3/da

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    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D277/28—Radicals substituted by nitrogen atoms
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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DK00967988T 1999-10-11 2000-10-10 5-leddet derivater af heterocyklusser og deres anvendelse som monoaminoxidaseinhibitorer DK1223933T3 (da)

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FR9912643A FR2799461B1 (fr) 1999-10-11 1999-10-11 Derives d'heterocycles a 5 chainons, leur preparation et leur application a titre de medicaments
FR0010151A FR2812546B1 (fr) 2000-08-01 2000-08-01 Derives d'heterocycles a 5 chainons, leur preparation et leur application a titre de medicaments
FR0011169 2000-09-01

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DK00967988T DK1223933T3 (da) 1999-10-11 2000-10-10 5-leddet derivater af heterocyklusser og deres anvendelse som monoaminoxidaseinhibitorer

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BR0014649A (pt) 2002-06-18
NZ533429A (en) 2004-09-24
NO20021689D0 (no) 2002-04-10
IL148896A (en) 2009-02-11
MY145388A (en) 2012-01-31
CN1391474A (zh) 2003-01-15
JP2003511416A (ja) 2003-03-25
ES2270873T3 (es) 2007-04-16
EP1223933B1 (fr) 2006-09-06
EP1589007A2 (fr) 2005-10-26
US20070179153A1 (en) 2007-08-02
CY1106237T1 (el) 2011-06-08
NZ518304A (en) 2004-07-30
ES2544856T3 (es) 2015-09-04
HK1049957A1 (zh) 2003-06-06
RU2002112227A (ru) 2004-01-27
US20080146627A1 (en) 2008-06-19
WO2001026656A3 (fr) 2002-04-18
IL185118A0 (en) 2007-12-03
DE60030574T2 (de) 2007-09-20
EP1228760A2 (fr) 2002-08-07
EP1589007B1 (fr) 2015-06-03
KR20070068491A (ko) 2007-06-29
US8288560B2 (en) 2012-10-16
EP1228760A3 (fr) 2004-01-28
ATE522213T1 (de) 2011-09-15
KR20020060195A (ko) 2002-07-16
HK1049957B (zh) 2009-08-28
JP4972263B2 (ja) 2012-07-11
CZ304331B6 (cs) 2014-03-05
EP1223933A2 (fr) 2002-07-24
AU783129B2 (en) 2005-09-29
TWI283577B (en) 2007-07-11
RU2271355C2 (ru) 2006-03-10
DK1589007T3 (da) 2015-08-10
PL355147A1 (en) 2004-04-05
MXPA02003665A (es) 2003-10-14
DE60030574D1 (de) 2006-10-19
HUP0203841A2 (en) 2003-05-28
NO20021689L (no) 2002-05-30
AR029006A1 (es) 2003-06-04
US20110172434A1 (en) 2011-07-14
CA2388505A1 (fr) 2001-04-19
AU7796500A (en) 2001-04-23
ATE338547T1 (de) 2006-09-15
US20070021390A1 (en) 2007-01-25
HU228254B1 (en) 2013-02-28
NO331874B1 (no) 2012-04-23
IL148896A0 (en) 2002-09-12
PT1223933E (pt) 2006-12-29
EP1589007A3 (fr) 2009-04-29
CN100488506C (zh) 2009-05-20
US7956075B2 (en) 2011-06-07
CA2388505C (fr) 2013-03-12
PL215580B1 (pl) 2013-12-31
HUP0203841A3 (en) 2003-07-28
WO2001026656A2 (fr) 2001-04-19
PT1589007E (pt) 2015-10-12
TWI292316B (en) 2008-01-11
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KR100731698B1 (ko) 2007-06-25
TW200509916A (en) 2005-03-16

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