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DK1296970T3 - Fremgangsmåde til fremstilling af citalopram - Google Patents

Fremgangsmåde til fremstilling af citalopram

Info

Publication number
DK1296970T3
DK1296970T3 DK01931469T DK01931469T DK1296970T3 DK 1296970 T3 DK1296970 T3 DK 1296970T3 DK 01931469 T DK01931469 T DK 01931469T DK 01931469 T DK01931469 T DK 01931469T DK 1296970 T3 DK1296970 T3 DK 1296970T3
Authority
DK
Denmark
Prior art keywords
citalopram
preparation
Prior art date
Application number
DK01931469T
Other languages
English (en)
Inventor
Hans Petersen
Robert Dancer
Original Assignee
Lundbeck & Co As H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Application granted granted Critical
Publication of DK1296970T3 publication Critical patent/DK1296970T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • C07D307/88—Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Furan Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK01931469T 2000-05-12 2001-05-10 Fremgangsmåde til fremstilling af citalopram DK1296970T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DKPA200000783 2000-05-12
PCT/DK2001/000333 WO2001085712A1 (en) 2000-05-12 2001-05-10 Method for the preparation of citalopram

Publications (1)

Publication Number Publication Date
DK1296970T3 true DK1296970T3 (da) 2008-07-14

Family

ID=8159493

Family Applications (1)

Application Number Title Priority Date Filing Date
DK01931469T DK1296970T3 (da) 2000-05-12 2001-05-10 Fremgangsmåde til fremstilling af citalopram

Country Status (29)

Country Link
US (1) US6660873B2 (da)
EP (1) EP1296970B1 (da)
JP (1) JP2003532721A (da)
CN (1) CN100422166C (da)
AR (1) AR032455A1 (da)
AT (1) ATE389645T1 (da)
AU (2) AU5823901A (da)
BG (1) BG65820B1 (da)
BR (1) BR0110996A (da)
CA (1) CA2408292C (da)
CZ (1) CZ20024065A3 (da)
DE (1) DE60133280T2 (da)
DK (1) DK1296970T3 (da)
EA (1) EA005674B1 (da)
ES (1) ES2301541T3 (da)
HR (1) HRP20020881A2 (da)
HU (1) HUP0301942A2 (da)
IL (2) IL152645A0 (da)
IS (1) IS2586B (da)
MX (1) MXPA02011125A (da)
NO (1) NO327963B1 (da)
NZ (1) NZ522475A (da)
PL (1) PL358144A1 (da)
PT (1) PT1296970E (da)
SI (1) SI1296970T1 (da)
SK (1) SK287035B6 (da)
UA (1) UA72039C2 (da)
WO (1) WO2001085712A1 (da)
ZA (1) ZA200208973B (da)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL198024B1 (pl) 1999-04-14 2008-05-30 Lundbeck & Co As H Sposób wytwarzania citalopramu, związki pośrednie i ich zastosowanie do wytwarzania citalopramu
US6310222B1 (en) * 1999-11-01 2001-10-30 Sumika Fine Chemicals Co., Ltd. Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
US6433196B1 (en) * 2000-02-17 2002-08-13 Sumika Fine Chemicals Co., Ltd. Production method of citalopram, intermediate therefor and production method of the intermediate
IES20010157A2 (en) 2000-03-03 2002-03-06 Lundbeck & Co As H Method for the preparation of citalopram
IES20010206A2 (en) 2000-03-13 2002-03-06 Lundbeck & Co As H Method for the preparation of citalopram
CN1427835A (zh) 2000-03-13 2003-07-02 H·隆德贝克有限公司 5－取代的1－(4－氟苯基)－1,3－二氢异苯并呋喃的分步烷基化
AR032455A1 (es) 2000-05-12 2003-11-12 Lundbeck & Co As H Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
IN192057B (da) * 2001-07-19 2004-02-14 Ranbaxy Lab Ltd
TR200504022T1 (tr) * 2003-03-24 2006-08-21 Hetero Drugs Limited (S)-sitalopram oksalatın yeni sıvı kristal formları.
BR0318581A (pt) * 2003-10-28 2006-10-10 Wockhardt Ltd processo melhorando para fabriacação de bromidrato de citalopram
US20050143350A1 (en) * 2003-11-19 2005-06-30 Seed John C. Combination drug therapy to treat obesity
EP1797060A2 (en) 2004-08-23 2007-06-20 Sun Pharmaceutical Industries Limited "process for preparation of citalopram and enantiomers"

Family Cites Families (40)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1143702A (da) 1965-03-18
GB1526331A (en) * 1976-01-14 1978-09-27 Kefalas As Phthalanes
GB8419963D0 (en) 1984-08-06 1984-09-12 Lundbeck & Co As H Intermediate compound and method
GB8814057D0 (en) 1988-06-14 1988-07-20 Lundbeck & Co As H New enantiomers & their isolation
US5296507A (en) 1990-09-06 1994-03-22 H.Lundbeck A/S Treatment of cerbrovascular disorders
DE19626659A1 (de) 1996-07-03 1998-01-08 Basf Ag Verfahren zur Herstellung von Phthaliden
DE19627697A1 (de) 1996-07-10 1998-01-15 Basf Ag Verfahren zur Herstellung von Phthaliden
DK1015416T3 (da) 1997-07-08 2001-11-05 Lundbeck & Co As H Fremgangsmåde til fremstilling af citalopram
UA62985C2 (en) 1997-11-10 2004-01-15 Lunnbeck As H A method for the preparation of citalopram
JP3813820B2 (ja) 1997-11-11 2006-08-23 ハー・ルンドベック・アクチエゼルスカベット シタロプラムの製造方法
ATE230738T1 (de) 1998-10-20 2003-01-15 Lundbeck & Co As H Verfahren zur herstellung von citalopram
TR200101796T2 (tr) 1998-12-23 2001-11-21 H. Lundbeck A/S 5-Siyanofitalitin preparasyonuna yönelik metot
AR022329A1 (es) 1999-01-29 2002-09-04 Lundbeck & Co As H Metodo para la preparacion de 5-cianoftalida
PL198024B1 (pl) 1999-04-14 2008-05-30 Lundbeck & Co As H Sposób wytwarzania citalopramu, związki pośrednie i ich zastosowanie do wytwarzania citalopramu
ITMI991579A1 (it) 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
ITMI991581A1 (it) 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
ITMI991486A1 (it) 1999-07-06 2001-01-06 Vis Farmaceutici S P A Processo per la sintesi di citalopram
ES2169709A1 (es) 1999-10-25 2002-07-01 Lundbeck & Co As H Metodo para la preparacion de citalopram
US6310222B1 (en) 1999-11-01 2001-10-30 Sumika Fine Chemicals Co., Ltd. Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
AR026063A1 (es) 1999-11-01 2002-12-26 Lundbeck & Co As H Metodo para la preparacion de 5-carboxiftalida.
CN1398263A (zh) 1999-12-28 2003-02-19 H·隆德贝克有限公司 制备西酞普兰的方法
PL198803B1 (pl) 1999-12-30 2008-07-31 Lundbeck & Co As H Sposób wytwarzania 5-cyjano-3H-izobenzofuran-1-onu
EP1254129B1 (en) 2000-01-14 2003-10-22 H. Lundbeck A/S Method for the preparation of 5-cyanophthalide
IT1317729B1 (it) 2000-01-18 2003-07-15 Norpharma S P A Procedimento per la preparazione della 5-carbossiftalide.
US6433196B1 (en) 2000-02-17 2002-08-13 Sumika Fine Chemicals Co., Ltd. Production method of citalopram, intermediate therefor and production method of the intermediate
IES20010143A2 (en) 2000-02-24 2001-07-25 Lundbeck & Co As H Method for the preparation of citalopram
NL1017415C1 (nl) 2000-02-24 2001-05-18 Lundbeck & Co As H Werkwijze voor de bereiding van Citalopram.
IES20010157A2 (en) 2000-03-03 2002-03-06 Lundbeck & Co As H Method for the preparation of citalopram
GB0005477D0 (en) 2000-03-07 2000-04-26 Resolution Chemicals Limited Process for the preparation of citalopram
IES20010206A2 (en) 2000-03-13 2002-03-06 Lundbeck & Co As H Method for the preparation of citalopram
CN1427835A (zh) 2000-03-13 2003-07-02 H·隆德贝克有限公司 5－取代的1－(4－氟苯基)－1,3－二氢异苯并呋喃的分步烷基化
JP2003527387A (ja) 2000-03-13 2003-09-16 ハー・ルンドベック・アクチエゼルスカベット シタロプラムの製造方法
GB2357762B (en) 2000-03-13 2002-01-30 Lundbeck & Co As H Crystalline base of citalopram
DK1265882T3 (da) 2000-03-14 2004-06-01 Lundbeck & Co As H Fremgangsmåde til fremstilling af citalopram
KR20020080483A (ko) 2000-03-16 2002-10-23 하. 룬트벡 아크티에 셀스카브 5-시아노-1-(4-플루오로페닐)-1,3-디히드로이소벤조푸란의제조 방법
AR032455A1 (es) 2000-05-12 2003-11-12 Lundbeck & Co As H Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
AU2001272368A1 (en) 2000-07-06 2002-01-21 H. Lundbeck, A/S Method for the preparation of citalopram
IL144817A0 (en) 2000-08-18 2002-06-30 Lundbeck & Co As H Method for the preparation of citalopram
SG167655A1 (en) 2000-12-22 2011-01-28 Lundbeck & Co As H Method for the preparation of pure citalopram
HRP20020005A2 (en) 2000-12-28 2003-04-30 Lundbeck & Co As H Process for the preparation of pure citalopram

Also Published As

Publication number Publication date
WO2001085712A1 (en) 2001-11-15
MXPA02011125A (es) 2003-03-10
ZA200208973B (en) 2003-11-05
IS2586B (is) 2010-02-15
CN1441795A (zh) 2003-09-10
EA005674B1 (ru) 2005-04-28
NO20025423D0 (no) 2002-11-12
NO20025423L (no) 2002-11-12
CN100422166C (zh) 2008-10-01
ATE389645T1 (de) 2008-04-15
JP2003532721A (ja) 2003-11-05
HRP20020881A2 (en) 2004-12-31
US20030134895A1 (en) 2003-07-17
DE60133280T2 (de) 2009-04-16
HUP0301942A2 (hu) 2003-09-29
IL152645A (en) 2009-12-24
SK17542002A3 (sk) 2003-04-01
DE60133280D1 (de) 2008-04-30
CA2408292A1 (en) 2001-11-15
US6660873B2 (en) 2003-12-09
HK1056171A1 (zh) 2004-02-06
BG65820B1 (bg) 2010-01-29
IS6605A (is) 2002-10-31
BG107349A (bg) 2003-09-30
AU2001258239B2 (en) 2005-12-08
AR032455A1 (es) 2003-11-12
EP1296970A1 (en) 2003-04-02
NZ522475A (en) 2004-09-24
CZ20024065A3 (cs) 2003-03-12
EP1296970B1 (en) 2008-03-19
IL152645A0 (en) 2003-06-24
UA72039C2 (en) 2005-01-17
SK287035B6 (sk) 2009-10-07
BR0110996A (pt) 2003-03-18
PT1296970E (pt) 2008-06-11
AU5823901A (en) 2001-11-20
SI1296970T1 (sl) 2008-08-31
NO327963B1 (no) 2009-10-26
CA2408292C (en) 2009-11-10
EA200201211A1 (ru) 2003-04-24
ES2301541T3 (es) 2008-07-01
PL358144A1 (en) 2004-08-09

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