DK1196428T3 - 11-beta-aryl-17,17-spirothiolan-substituerede steroider - Google Patents
11-beta-aryl-17,17-spirothiolan-substituerede steroiderInfo
- Publication number
- DK1196428T3 DK1196428T3 DK00948741T DK00948741T DK1196428T3 DK 1196428 T3 DK1196428 T3 DK 1196428T3 DK 00948741 T DK00948741 T DK 00948741T DK 00948741 T DK00948741 T DK 00948741T DK 1196428 T3 DK1196428 T3 DK 1196428T3
- Authority
- DK
- Denmark
- Prior art keywords
- spirothiolane
- beta
- aryl
- substituted steroids
- compounds
- Prior art date
Links
- 150000003431 steroids Chemical class 0.000 title 1
- 238000000034 method Methods 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 1
- 230000001747 exhibiting effect Effects 0.000 abstract 1
- 102000003998 progesterone receptors Human genes 0.000 abstract 1
- 108090000468 progesterone receptors Proteins 0.000 abstract 1
- -1 steroid compounds Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J33/00—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Diabetes (AREA)
- Gynecology & Obstetrics (AREA)
- Pregnancy & Childbirth (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US09/357,923 US6043235A (en) | 1999-07-21 | 1999-07-21 | 11β-aryl-17, 17-spirothiolane-substituted steroids |
| PCT/US2000/019537 WO2001007462A1 (en) | 1999-07-21 | 2000-07-20 | 11β-ARYL-17,17-SPIROTHIOLANE-SUBSTITUTED STEROIDS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1196428T3 true DK1196428T3 (da) | 2005-01-24 |
Family
ID=23407590
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK00948741T DK1196428T3 (da) | 1999-07-21 | 2000-07-20 | 11-beta-aryl-17,17-spirothiolan-substituerede steroider |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US6043235A (da) |
| EP (1) | EP1196428B1 (da) |
| JP (1) | JP4768181B2 (da) |
| KR (1) | KR100616025B1 (da) |
| AT (1) | ATE277071T1 (da) |
| AU (1) | AU774472B2 (da) |
| CA (1) | CA2379995C (da) |
| DE (1) | DE60014096T2 (da) |
| DK (1) | DK1196428T3 (da) |
| ES (1) | ES2228584T3 (da) |
| HK (1) | HK1044542B (da) |
| NO (1) | NO321524B1 (da) |
| PT (1) | PT1196428E (da) |
| WO (1) | WO2001007462A1 (da) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6262042B1 (en) | 1998-05-29 | 2001-07-17 | Research Triangle Institute | 17β-amino and hydroxylamino-11β-arylsteroids and their derivatives having agonist or antagonist hormonal properties |
| AP2949A (en) | 2006-03-07 | 2014-07-31 | Shroff Geeta | Compositions comprising human embryonic stem cellsand their derivatives, methods of use, and method s of preparation |
| KR200451979Y1 (ko) * | 2008-04-11 | 2011-01-24 | 정종오 | 회전형 광고장치 |
| DE102009034367A1 (de) * | 2009-07-20 | 2011-01-27 | Bayer Schering Pharma Aktiengesellschaft | 17-Hydroxy-17-pentafluorethyl-estra-4,9(10)-dien-11-benzyliden-Derivate, Verfahren zu deren Herstellung und deren Verwendung zur Behandlung von Krankheiten |
| DE102009034526A1 (de) * | 2009-07-21 | 2011-02-10 | Bayer Schering Pharma Aktiengesellschaft | 17-Hydroxy-17-pentafluorethyl-estra-4,9(10)-dien-11-ethinylphenyl-Derivate, Verfahren zu deren Herstellung und deren Verwendung zur Behandlung von Krankheiten |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2344286A1 (fr) * | 1976-03-16 | 1977-10-14 | Roussel Uclaf | Nouveaux derives 17-spirosultines, les g-hydroxy acides correspondants, leur procede de preparation et leur application comme medicament |
| FR2374037A1 (fr) * | 1976-10-27 | 1978-07-13 | Roussel Uclaf | Nouveaux derives steroides 17-spirosultines les g-hydroxy acides correspondants, leur procede de preparation et leur application comme medicament |
| ZA929315B (en) * | 1991-12-20 | 1993-05-24 | Akzo Nv | 17-spirofuran-3'-ylidene steroids. |
| IL115659A (en) * | 1994-10-27 | 2000-06-01 | Akzo Nobel Nv | Steroids with a 17-spiromethylene lactone or lactol group process for their preparation and pharmaceutical compositions containing them |
-
1999
- 1999-07-21 US US09/357,923 patent/US6043235A/en not_active Expired - Lifetime
-
2000
- 2000-07-20 AT AT00948741T patent/ATE277071T1/de active
- 2000-07-20 JP JP2001512545A patent/JP4768181B2/ja not_active Expired - Fee Related
- 2000-07-20 ES ES00948741T patent/ES2228584T3/es not_active Expired - Lifetime
- 2000-07-20 DE DE60014096T patent/DE60014096T2/de not_active Expired - Lifetime
- 2000-07-20 DK DK00948741T patent/DK1196428T3/da active
- 2000-07-20 CA CA002379995A patent/CA2379995C/en not_active Expired - Fee Related
- 2000-07-20 KR KR1020027000816A patent/KR100616025B1/ko not_active Expired - Fee Related
- 2000-07-20 EP EP00948741A patent/EP1196428B1/en not_active Expired - Lifetime
- 2000-07-20 HK HK02106120.8A patent/HK1044542B/en not_active IP Right Cessation
- 2000-07-20 AU AU62200/00A patent/AU774472B2/en not_active Ceased
- 2000-07-20 WO PCT/US2000/019537 patent/WO2001007462A1/en not_active Ceased
- 2000-07-20 PT PT00948741T patent/PT1196428E/pt unknown
-
2002
- 2002-01-17 NO NO20020260A patent/NO321524B1/no not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| PT1196428E (pt) | 2005-02-28 |
| NO20020260D0 (no) | 2002-01-17 |
| EP1196428B1 (en) | 2004-09-22 |
| US6043235A (en) | 2000-03-28 |
| KR20020092893A (ko) | 2002-12-12 |
| DE60014096T2 (de) | 2005-10-06 |
| WO2001007462A1 (en) | 2001-02-01 |
| ATE277071T1 (de) | 2004-10-15 |
| JP4768181B2 (ja) | 2011-09-07 |
| AU6220000A (en) | 2001-02-13 |
| ES2228584T3 (es) | 2005-04-16 |
| NO321524B1 (no) | 2006-05-15 |
| KR100616025B1 (ko) | 2006-08-30 |
| AU774472B2 (en) | 2004-07-01 |
| EP1196428A1 (en) | 2002-04-17 |
| CA2379995A1 (en) | 2001-02-01 |
| JP2003531815A (ja) | 2003-10-28 |
| EP1196428A4 (en) | 2002-10-16 |
| NO20020260L (no) | 2002-03-14 |
| DE60014096D1 (de) | 2004-10-28 |
| CA2379995C (en) | 2008-10-14 |
| HK1044542B (en) | 2005-02-25 |
| HK1044542A1 (en) | 2002-10-25 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DK1124842T3 (da) | Betulinsyrederivater anvendelige til behandling af neuroektodermale tumorer | |
| BR0010215A (pt) | Derivados de indolina como antagonistas de progesterona | |
| AU7743001A (en) | Cyclopentanoindoles, compositions containing such compounds and methods of treatment | |
| DK1053239T3 (da) | Gluccocorticoid-selektive, anti-inflammatoriske midler | |
| DE69709938D1 (de) | N-benzylpiperidin- und tetrahydropyridin-derivate | |
| TR200003377T2 (tr) | Estrojenler ile bütünleşik 2-fenil-1-[4-(2-aminoetoksi)benzil]-indol | |
| EP1042352A4 (en) | ANDROGENE STEROID DERIVATIVES AND A METHOD FOR THE PRODUCTION AND USE THEREOF | |
| IL139861A (en) | 17beta-AMINO-AND HYDROXYLAMINO -11 beta - ARYLSTEROID DERIVATIVES, METHODS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME | |
| DE60030410D1 (de) | Steroid sulfataseinhibitoren, verfahren zu ihrer herstellung und ihre verwendung | |
| NO20023276L (no) | Fremgangsmåter fremstilling av betulinsyre | |
| HK1046404A1 (zh) | 用作nmda受体拮抗剂的取代的吡咯烷-2，3，4-三酮-3-肟衍生物 | |
| DK1196428T3 (da) | 11-beta-aryl-17,17-spirothiolan-substituerede steroider | |
| BR9713176A (pt) | Benzotiofenos amorfos,métodos de preparação e métodos de uso | |
| WO2001062765A3 (en) | Small molecule modulators of g protein-coupled receptor six | |
| DK0559706T3 (da) | 2 beta,19-methylenamino-broforbundne steroider som aromataseinhibitorer. | |
| DK1165595T3 (da) | Leverspecifikke galdesyre-derivater af glucocorticoid-receptorantangonisten RU486 | |
| AU6832498A (en) | Substituted benzyl oximino compounds | |
| ATE265418T1 (de) | Neue substituierte 3-phenoxy- und 3- phenylalkyloxy-2-phenyl-propylamine | |
| AU3894399A (en) | Benzocarbazole and indenoindole derived estrogenic agents | |
| DK1235850T3 (da) | Umættede 14,15-cyclopropano-androstaner, fremgangsmåde til deres fremstilling og farmaceutiske præparater indeholdende disse forbindelser | |
| MX9707832A (es) | 1-fenil-3-pirazolcarboxilamidas que actuan sobre los receptores de neurotensina. |