DK1163241T3 - Zolpidemsalte - Google Patents
ZolpidemsalteInfo
- Publication number
- DK1163241T3 DK1163241T3 DK00913159T DK00913159T DK1163241T3 DK 1163241 T3 DK1163241 T3 DK 1163241T3 DK 00913159 T DK00913159 T DK 00913159T DK 00913159 T DK00913159 T DK 00913159T DK 1163241 T3 DK1163241 T3 DK 1163241T3
- Authority
- DK
- Denmark
- Prior art keywords
- zolpidem
- salt
- exhibiting
- excluding
- minute
- Prior art date
Links
- ZAFYATHCZYHLPB-UHFFFAOYSA-N zolpidem Chemical compound N1=C2C=CC(C)=CN2C(CC(=O)N(C)C)=C1C1=CC=C(C)C=C1 ZAFYATHCZYHLPB-UHFFFAOYSA-N 0.000 title abstract 3
- 229960001475 zolpidem Drugs 0.000 title abstract 2
- 230000001747 exhibiting effect Effects 0.000 abstract 1
- 239000012458 free base Substances 0.000 abstract 1
- 238000010438 heat treatment Methods 0.000 abstract 1
- 230000008018 melting Effects 0.000 abstract 1
- 238000002844 melting Methods 0.000 abstract 1
- -1 salt zolpidem tartrate Chemical class 0.000 abstract 1
- 229960005111 zolpidem tartrate Drugs 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Anesthesiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US12649499P | 1999-03-25 | 1999-03-25 | |
| EP99203478A EP1038875B1 (fr) | 1999-03-25 | 1999-10-22 | Dérivés d'imidazopyridine et procédé pour leur préparation |
| US09/449,974 US6242460B1 (en) | 1999-03-25 | 1999-11-26 | Zolpidem salt forms |
| PCT/NL2000/000171 WO2000058310A1 (fr) | 1999-03-25 | 2000-03-13 | Sels de zolpidem |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1163241T3 true DK1163241T3 (da) | 2005-10-10 |
Family
ID=27240136
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK00913159T DK1163241T3 (da) | 1999-03-25 | 2000-03-13 | Zolpidemsalte |
Country Status (9)
| Country | Link |
|---|---|
| EP (1) | EP1163241B1 (fr) |
| AT (1) | ATE297924T1 (fr) |
| AU (1) | AU3464200A (fr) |
| DE (1) | DE60020814T2 (fr) |
| DK (1) | DK1163241T3 (fr) |
| ES (1) | ES2240074T3 (fr) |
| NL (1) | NL1014634C1 (fr) |
| PT (1) | PT1163241E (fr) |
| WO (1) | WO2000058310A1 (fr) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2003518016A (ja) * | 1999-11-22 | 2003-06-03 | エギシュ ヂョヂセルヂャール エルテー | 6−メチル−2−(4−メチル−フェニル)−イミダゾ[1,2−a]ピリジン−3−(N,N−ジメチル−アセトアミド)の製法及び中間体 |
| EP1600159A1 (fr) * | 2000-04-24 | 2005-11-30 | Teva Pharmaceutical Industries Ltd | Procédé de synthèse de dérivés differentes de zolpidem hemitartrat |
| SK16372002A3 (sk) * | 2000-04-24 | 2003-04-01 | Teva Pharmaceutical Industries Ltd. | Zolpidem hemitartrát |
| WO2006008636A2 (fr) * | 2004-07-16 | 2006-01-26 | Ranbaxy Laboratories Limited | Nouveau polymorphe d'hemitartrate de zolpidem |
| US20080293946A1 (en) * | 2005-10-03 | 2008-11-27 | Cheng Brian K | Process for Preparing Zolpidem Hemitartrate and Tartrate Polymorphs |
| CN116283957A (zh) * | 2021-12-03 | 2023-06-23 | 山东新时代药业有限公司 | 唑吡坦水合物及其制备方法 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2492382A1 (fr) * | 1980-10-22 | 1982-04-23 | Synthelabo | Derives d'imidazo (1,2-a) pyridine, leur preparation et leur application en therapeutique |
| FR2600650B1 (fr) * | 1986-06-27 | 1988-09-09 | Synthelabo | Procede de preparation d'imidazopyridines et composes intermediaires |
-
2000
- 2000-03-13 WO PCT/NL2000/000171 patent/WO2000058310A1/fr not_active Ceased
- 2000-03-13 AT AT00913159T patent/ATE297924T1/de not_active IP Right Cessation
- 2000-03-13 EP EP00913159A patent/EP1163241B1/fr not_active Expired - Lifetime
- 2000-03-13 AU AU34642/00A patent/AU3464200A/en not_active Abandoned
- 2000-03-13 NL NL1014634A patent/NL1014634C1/nl not_active IP Right Cessation
- 2000-03-13 ES ES00913159T patent/ES2240074T3/es not_active Expired - Lifetime
- 2000-03-13 DE DE60020814T patent/DE60020814T2/de not_active Expired - Fee Related
- 2000-03-13 PT PT00913159T patent/PT1163241E/pt unknown
- 2000-03-13 DK DK00913159T patent/DK1163241T3/da active
Also Published As
| Publication number | Publication date |
|---|---|
| DE60020814T2 (de) | 2006-05-04 |
| ATE297924T1 (de) | 2005-07-15 |
| ES2240074T3 (es) | 2005-10-16 |
| PT1163241E (pt) | 2005-08-31 |
| DE60020814D1 (de) | 2005-07-21 |
| AU3464200A (en) | 2000-10-16 |
| EP1163241B1 (fr) | 2005-06-15 |
| WO2000058310A1 (fr) | 2000-10-05 |
| EP1163241A1 (fr) | 2001-12-19 |
| NL1014634C1 (nl) | 2000-08-03 |
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