DK1007517T3 - Fremgangsmåde til fremstilling af 5-hydroxymethylthiazoler - Google Patents
Fremgangsmåde til fremstilling af 5-hydroxymethylthiazolerInfo
- Publication number
- DK1007517T3 DK1007517T3 DK98942099T DK98942099T DK1007517T3 DK 1007517 T3 DK1007517 T3 DK 1007517T3 DK 98942099 T DK98942099 T DK 98942099T DK 98942099 T DK98942099 T DK 98942099T DK 1007517 T3 DK1007517 T3 DK 1007517T3
- Authority
- DK
- Denmark
- Prior art keywords
- preparation
- hydroxymethylthiazole
- compound
- formula
- hydroxymethylthiazoles
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 4
- WKBQQWDVVHGWDB-UHFFFAOYSA-N 1,3-thiazol-5-ylmethanol Chemical class OCC1=CN=CS1 WKBQQWDVVHGWDB-UHFFFAOYSA-N 0.000 title 1
- CDBYLPFSWZWCQE-UHFFFAOYSA-L Sodium Carbonate Chemical compound [Na+].[Na+].[O-]C([O-])=O CDBYLPFSWZWCQE-UHFFFAOYSA-L 0.000 abstract 2
- 239000002253 acid Substances 0.000 abstract 2
- 125000005843 halogen group Chemical group 0.000 abstract 2
- -1 hydroxymethylthiazole compound Chemical class 0.000 abstract 2
- JNHDLNXNYPLBMJ-UHFFFAOYSA-N 1,3-thiazol-2-ylmethanol Chemical compound OCC1=NC=CS1 JNHDLNXNYPLBMJ-UHFFFAOYSA-N 0.000 abstract 1
- 229940126214 compound 3 Drugs 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 229910000029 sodium carbonate Inorganic materials 0.000 abstract 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D277/24—Radicals substituted by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US08/921,399 US5959118A (en) | 1997-08-29 | 1997-08-29 | Process for the preparation of 5-hydroxymethylthiazoles |
| PCT/US1998/017100 WO1999011636A1 (fr) | 1997-08-29 | 1998-08-18 | Procede de preparation de 5-hydroxymethylthiazoles |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1007517T3 true DK1007517T3 (da) | 2004-02-09 |
Family
ID=25445373
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK98942099T DK1007517T3 (da) | 1997-08-29 | 1998-08-18 | Fremgangsmåde til fremstilling af 5-hydroxymethylthiazoler |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US5959118A (fr) |
| EP (1) | EP1007517B1 (fr) |
| JP (1) | JP2002510331A (fr) |
| AT (1) | ATE251616T1 (fr) |
| CA (1) | CA2294089A1 (fr) |
| DE (1) | DE69818837T2 (fr) |
| DK (1) | DK1007517T3 (fr) |
| ES (1) | ES2209198T3 (fr) |
| PT (1) | PT1007517E (fr) |
| WO (1) | WO1999011636A1 (fr) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1313624B1 (it) | 1999-09-21 | 2002-09-09 | Archimica Spa Ora Clariant Lif | Procedimento per la sintesi del ritonavir |
| CN101863853B (zh) * | 2009-12-28 | 2012-12-19 | 安徽贝克联合制药有限公司 | 一锅煮法制备5-羟甲基噻唑工艺 |
| BR112020008124A2 (pt) | 2017-10-27 | 2020-10-06 | Syngenta Participations Ag | composições de controle de vetores, métodos e produtos utilizando as mesmas |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3299083A (en) * | 1967-01-17 | Processes for preparing hydroxy- methylthiazole | ||
| US2332906A (en) * | 1939-10-03 | 1943-10-26 | Foldi Zolten | Process for preparation of sulphonamide derivatives |
| DE3631538A1 (de) * | 1986-09-17 | 1988-03-24 | Bayer Ag | Verfahren zur herstellung von 2-chlor-5-chlormethylthiazol |
| US5696270A (en) * | 1989-05-23 | 1997-12-09 | Abbott Laboratories | Intermediate for making retroviral protease inhibiting compounds |
| US5354866A (en) * | 1989-05-23 | 1994-10-11 | Abbott Laboratories | Retroviral protease inhibiting compounds |
| PT793659E (pt) * | 1994-11-22 | 2001-07-31 | Abbott Lab | Processo para a preparacao fr 5-hidroximetiltiazolo |
| DE19520612A1 (de) * | 1995-06-06 | 1996-12-12 | Bayer Ag | Verfahren zur Herstellung von Benzylalkohol |
| WO1997010226A1 (fr) * | 1995-09-11 | 1997-03-20 | Novartis Ag | Procede de preparation d'un compose a base de 2-chloro-5-chloromethyl-thiazole |
| GB9518824D0 (en) * | 1995-09-14 | 1995-11-15 | Fine Organics Ltd | Preparation of substituted thiazoles |
| DE19547076A1 (de) * | 1995-12-18 | 1997-06-19 | Bayer Ag | Verbessertes Verfahren zur Herstellung von 5-Hydroxymethylthiazol |
| US8013167B1 (en) * | 1995-12-21 | 2011-09-06 | Syngenta Crop Protection, Inc. | Process for the preparation of 2-chloro-5-chloromethyl-thiazole |
| US6265585B1 (en) * | 1997-01-22 | 2001-07-24 | Syngenta Crop Protection, Inc. | Process for the preparation of thiazole derivatives |
| US5773625A (en) * | 1997-10-02 | 1998-06-30 | Abbott Laboratories | Process for the preparation of disubstituted carbonates |
-
1997
- 1997-08-29 US US08/921,399 patent/US5959118A/en not_active Expired - Lifetime
-
1998
- 1998-08-18 CA CA002294089A patent/CA2294089A1/fr not_active Abandoned
- 1998-08-18 JP JP51684099A patent/JP2002510331A/ja not_active Ceased
- 1998-08-18 AT AT98942099T patent/ATE251616T1/de not_active IP Right Cessation
- 1998-08-18 DK DK98942099T patent/DK1007517T3/da active
- 1998-08-18 DE DE69818837T patent/DE69818837T2/de not_active Expired - Fee Related
- 1998-08-18 PT PT98942099T patent/PT1007517E/pt unknown
- 1998-08-18 WO PCT/US1998/017100 patent/WO1999011636A1/fr not_active Ceased
- 1998-08-18 ES ES98942099T patent/ES2209198T3/es not_active Expired - Lifetime
- 1998-08-18 EP EP98942099A patent/EP1007517B1/fr not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| PT1007517E (pt) | 2004-03-31 |
| EP1007517B1 (fr) | 2003-10-08 |
| US5959118A (en) | 1999-09-28 |
| EP1007517A1 (fr) | 2000-06-14 |
| WO1999011636A1 (fr) | 1999-03-11 |
| DE69818837T2 (de) | 2004-07-22 |
| DE69818837D1 (de) | 2003-11-13 |
| CA2294089A1 (fr) | 1999-03-11 |
| ATE251616T1 (de) | 2003-10-15 |
| ES2209198T3 (es) | 2004-06-16 |
| JP2002510331A (ja) | 2002-04-02 |
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