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DK1073447T3 - N1-modificerede glycopeptider - Google Patents

N1-modificerede glycopeptider

Info

Publication number
DK1073447T3
DK1073447T3 DK99909654T DK99909654T DK1073447T3 DK 1073447 T3 DK1073447 T3 DK 1073447T3 DK 99909654 T DK99909654 T DK 99909654T DK 99909654 T DK99909654 T DK 99909654T DK 1073447 T3 DK1073447 T3 DK 1073447T3
Authority
DK
Denmark
Prior art keywords
modified glycopeptides
glycopeptides
modified
compounds
useful
Prior art date
Application number
DK99909654T
Other languages
English (en)
Inventor
Richard Craig Thompson
Stephen Charles Wilkie
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Application granted granted Critical
Publication of DK1073447T3 publication Critical patent/DK1073447T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DK99909654T 1998-05-01 1999-02-26 N1-modificerede glycopeptider DK1073447T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US8387998P 1998-05-01 1998-05-01
PCT/US1999/004306 WO1999056760A1 (en) 1998-05-01 1999-02-26 N1-modified glycopeptides

Publications (1)

Publication Number Publication Date
DK1073447T3 true DK1073447T3 (da) 2007-09-03

Family

ID=22181253

Family Applications (1)

Application Number Title Priority Date Filing Date
DK99909654T DK1073447T3 (da) 1998-05-01 1999-02-26 N1-modificerede glycopeptider

Country Status (10)

Country Link
US (3) US6670446B1 (da)
EP (1) EP1073447B1 (da)
JP (1) JP4307723B2 (da)
AT (1) ATE361931T1 (da)
AU (1) AU2881399A (da)
CA (1) CA2330619A1 (da)
DE (1) DE69936052T2 (da)
DK (1) DK1073447T3 (da)
ES (1) ES2283107T3 (da)
WO (1) WO1999056760A1 (da)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1073447B1 (en) * 1998-05-01 2007-05-09 Eli Lilly And Company N1-modified glycopeptides
IL140093A0 (en) 1998-12-23 2002-02-10 Advanced Medicine Inc Glycopeptide derivatives and pharmaceutical compositions containing the same
EP1173193A4 (en) * 1999-04-02 2003-01-29 Univ Princeton DES-LEUCYL GLYCOPEPTIDANTIBIOTICS AND METHODS FOR THE PRODUCTION THEREOF
US6699836B2 (en) 1999-04-02 2004-03-02 The Trustees Of Princeton University Vancomycin analogs
DE60114567T2 (de) * 2000-02-11 2006-07-27 Eli Lilly And Co., Indianapolis Selektive acylierung von a82846-glycopeptid-analoge
AR053347A1 (es) 2005-04-06 2007-05-02 Astrazeneca Ab Derivados de [1,3]tiazolo[4,5-d]pirimidin-2(3h)-ona 5,7-sustituidos
UA90707C2 (en) 2005-04-06 2010-05-25 Астразенека Аб Novel 5-substituted 7-amino-[1,3]thiazolo[4,5-d]pyrimidine derivatives
EP1926780B1 (en) 2005-09-22 2013-08-14 Medivas, LLC Bis-( -amino)-diol-diester-containing poly(ester amide) and poly(ester urethane) compositions and methods of use
US8652504B2 (en) 2005-09-22 2014-02-18 Medivas, Llc Solid polymer delivery compositions and methods for use thereof
CN102083862A (zh) 2008-04-01 2011-06-01 康奈尔大学 有机-可溶性壳聚糖盐和由其制备的壳聚糖衍生生物材料

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4698327A (en) 1985-04-25 1987-10-06 Eli Lilly And Company Novel glycopeptide derivatives
US4643987A (en) 1985-08-14 1987-02-17 Eli Lilly And Company Modified glycopeptides
US4639433A (en) 1985-08-14 1987-01-27 Eli Lilly And Company Glycopeptide derivatives
EG18377A (en) 1986-09-19 1993-04-30 Lilly Co Eli Process for preparing glycopeptide antibiotics
US5534420A (en) 1988-07-28 1996-07-09 Eli Lilly And Company Biotransformation of glycopeptide antibiotics
IL96603A (en) 1989-12-13 1998-02-08 Lilly Co Eli Antibacterial glycopeptide derivatives, process for their preparation and pharmaceutical compositions containing them
RU2145609C1 (ru) 1994-01-28 2000-02-20 Эли Лилли Энд Компани Производные гликопептида или их соли, способ получения, фармацевтическая композиция
US5952310A (en) * 1997-05-20 1999-09-14 Eli Lilly And Company Glycopeptide hexapeptides
EP1073447B1 (en) * 1998-05-01 2007-05-09 Eli Lilly And Company N1-modified glycopeptides

Also Published As

Publication number Publication date
CA2330619A1 (en) 1999-11-11
ES2283107T3 (es) 2007-10-16
JP4307723B2 (ja) 2009-08-05
EP1073447A4 (en) 2001-10-04
ATE361931T1 (de) 2007-06-15
EP1073447A1 (en) 2001-02-07
WO1999056760A1 (en) 1999-11-11
DE69936052T2 (de) 2008-01-17
US6670446B1 (en) 2003-12-30
US20060128609A1 (en) 2006-06-15
EP1073447B1 (en) 2007-05-09
US20050037950A1 (en) 2005-02-17
US6939947B2 (en) 2005-09-06
AU2881399A (en) 1999-11-23
DE69936052D1 (de) 2007-06-21
JP2002513764A (ja) 2002-05-14

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