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DK0771197T3 - Anvendelse af heterocykliske forbindelser som dopamin-D3-ligander - Google Patents

Anvendelse af heterocykliske forbindelser som dopamin-D3-ligander

Info

Publication number
DK0771197T3
DK0771197T3 DK95926896T DK95926896T DK0771197T3 DK 0771197 T3 DK0771197 T3 DK 0771197T3 DK 95926896 T DK95926896 T DK 95926896T DK 95926896 T DK95926896 T DK 95926896T DK 0771197 T3 DK0771197 T3 DK 0771197T3
Authority
DK
Denmark
Prior art keywords
dopamine
pct
ligands
heterocyclic compounds
het
Prior art date
Application number
DK95926896T
Other languages
English (en)
Inventor
Liliane Unger
Hans-Juergen Teschendorf
Beate Hellendahl
Annegret Lansky
Beatrice Rendenbach-Mueller
Alfred Bach
Carsten Wicke
Original Assignee
Abbott Gmbh & Co Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Gmbh & Co Kg filed Critical Abbott Gmbh & Co Kg
Application granted granted Critical
Publication of DK0771197T3 publication Critical patent/DK0771197T3/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Furan Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
DK95926896T 1994-07-15 1995-07-14 Anvendelse af heterocykliske forbindelser som dopamin-D3-ligander DK0771197T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4425146A DE4425146A1 (de) 1994-07-15 1994-07-15 Verwendung heterocyclischer Verbindungen
PCT/EP1995/002782 WO1996002246A1 (de) 1994-07-15 1995-07-14 Verwendung heterocyclischer verbindungen als dopamin-d3 liganden

Publications (1)

Publication Number Publication Date
DK0771197T3 true DK0771197T3 (da) 2003-06-23

Family

ID=6523325

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95926896T DK0771197T3 (da) 1994-07-15 1995-07-14 Anvendelse af heterocykliske forbindelser som dopamin-D3-ligander

Country Status (22)

Country Link
US (1) US6090807A (da)
EP (1) EP0771197B1 (da)
JP (1) JPH10502658A (da)
KR (2) KR970704435A (da)
CN (2) CN1534023A (da)
AT (1) ATE236629T1 (da)
AU (1) AU704839B2 (da)
BG (1) BG63487B1 (da)
BR (1) BR9508296A (da)
CA (1) CA2195242A1 (da)
CZ (1) CZ293126B6 (da)
DE (2) DE4425146A1 (da)
DK (1) DK0771197T3 (da)
ES (1) ES2196072T3 (da)
FI (1) FI970148L (da)
HU (1) HUT77608A (da)
MX (1) MX9700430A (da)
NO (1) NO311683B1 (da)
NZ (1) NZ290388A (da)
PT (1) PT771197E (da)
SI (1) SI9520084B (da)
WO (1) WO1996002246A1 (da)

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US7320979B2 (en) * 2003-04-14 2008-01-22 Abbott Gmbh & Co. Kg. N-[(piperazinyl)hetaryl]arylsulfonamide compounds
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DE10358004A1 (de) 2003-12-11 2005-07-14 Abbott Gmbh & Co. Kg Ketolactam-Verbindungen und ihre Verwendung
US20050137186A1 (en) 2003-12-18 2005-06-23 Abbott Gmbh & Co. Kg. Tetrahydrobenzazepines and their use
JP4982184B2 (ja) 2003-12-18 2012-07-25 アボット ゲーエムベーハー ウント カンパニー カーゲー テトラヒドロベンズアゼピンおよびドーパミンｄ３レセプターの調節におけるこれらの使用
DE102004027358A1 (de) 2004-06-04 2005-12-29 Abbott Gmbh & Co. Kg Pyrimidinverbindungen und ihre Verwendung
DE102004027359A1 (de) * 2004-06-04 2005-12-29 Abbott Gmbh & Co. Kg Pyridin-2-onverbindungen und deren Verwendung
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JP2008526715A (ja) * 2005-01-03 2008-07-24 ユニベルシタ デグリ ストゥディ ディ シエナ 神経精神障害の治療のためのアリールピペラジン誘導体
WO2006081289A2 (en) * 2005-01-25 2006-08-03 Glaxo Group Limited Antibacterial agents
PA8802101A1 (es) 2007-11-02 2009-08-26 Abbott Gmbh & Co Kg Compuestos de 1,2,4-3,5-diona adecuados para el tratamiento de trastornos que responden a la modulación del receptor de dopamina d3
WO2009095438A1 (en) * 2008-02-01 2009-08-06 Neurosearch A/S Novel aryl piperazine derivatives useful as modulators of dopamine and serotonin receptors
WO2010040274A1 (zh) 2008-10-10 2010-04-15 中国人民解放军军事医学科学院毒物药物研究所 新型多巴胺d3受体配体，其制备方法及其医药用途
US9227944B2 (en) 2008-10-10 2016-01-05 Institute Of Pharmacology And Toxicology Academy Of Military Science P.L.A. China Dopamine D3 receptor ligands and preparation and medical uses of the same
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Also Published As

Publication number Publication date
CN1152870A (zh) 1997-06-25
HU9700111D0 (en) 1997-02-28
CZ293126B6 (cs) 2004-02-18
CA2195242A1 (en) 1996-02-01
NZ290388A (en) 2001-04-27
CN1534023A (zh) 2004-10-06
AU704839B2 (en) 1999-05-06
ATE236629T1 (de) 2003-04-15
CZ9697A3 (en) 1997-08-13
FI970148A0 (fi) 1997-01-14
PT771197E (pt) 2003-08-29
BR9508296A (pt) 1998-05-19
HUT77608A (hu) 1998-06-29
KR20040000412A (ko) 2004-01-03
EP0771197A1 (de) 1997-05-07
US6090807A (en) 2000-07-18
NO970163L (no) 1997-03-14
KR970704435A (ko) 1997-09-06
DE59510635D1 (de) 2003-05-15
WO1996002246A1 (de) 1996-02-01
SI9520084A (en) 1997-08-31
EP0771197B1 (de) 2003-04-09
BG101112A (bg) 1998-04-30
JPH10502658A (ja) 1998-03-10
BG63487B1 (bg) 2002-03-29
SI9520084B (sl) 2005-02-28
ES2196072T3 (es) 2003-12-16
FI970148A7 (fi) 1997-01-14
KR100443850B1 (ko) 2004-08-11
NO970163D0 (no) 1997-01-14
NO311683B1 (no) 2002-01-07
DE4425146A1 (de) 1996-01-18
MX9700430A (es) 1998-05-31
AU3111495A (en) 1996-02-16
FI970148L (fi) 1997-01-14

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