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DK0745083T3 - 2-Heteroaryl-5, 11-dihydro-6H-dipyrido[3, 2-b:2', 3'-e][1, 4]diazepiner og deres anvendelse til forebyggelse eller behandli - Google Patents

2-Heteroaryl-5, 11-dihydro-6H-dipyrido[3, 2-b:2', 3'-e][1, 4]diazepiner og deres anvendelse til forebyggelse eller behandli

Info

Publication number
DK0745083T3
DK0745083T3 DK95910286T DK95910286T DK0745083T3 DK 0745083 T3 DK0745083 T3 DK 0745083T3 DK 95910286 T DK95910286 T DK 95910286T DK 95910286 T DK95910286 T DK 95910286T DK 0745083 T3 DK0745083 T3 DK 0745083T3
Authority
DK
Denmark
Prior art keywords
dipyrido
diazepines
dihydro
prevention
treatment
Prior art date
Application number
DK95910286T
Other languages
English (en)
Inventor
Karl D Hargrave
Terence A Kelly
Suresh R Kapadia
John R Proudfoot
Daniel W Mcneil
Usha R Patel
Mario G Cardozo
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Application granted granted Critical
Publication of DK0745083T3 publication Critical patent/DK0745083T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/04Immunostimulants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C09DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
    • C09BORGANIC DYES OR CLOSELY-RELATED COMPOUNDS FOR PRODUCING DYES, e.g. PIGMENTS; MORDANTS; LAKES
    • C09B57/00Other synthetic dyes of known constitution

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK95910286T 1994-02-18 1995-02-17 2-Heteroaryl-5, 11-dihydro-6H-dipyrido[3, 2-b:2', 3'-e][1, 4]diazepiner og deres anvendelse til forebyggelse eller behandli DK0745083T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US19824294A 1994-02-18 1994-02-18
US35641594A 1994-12-14 1994-12-14
PCT/US1995/001993 WO1995022545A1 (en) 1994-02-18 1995-02-17 2-HETEROARYL-5,11-DIHYDRO-6H-DIPYRIDO[3,2-b:2',3'-e][1,4]DIAZEPINES AND THEIR USE IN THE PREVENTION OR TREATMENT OF HIV INFECTION

Publications (1)

Publication Number Publication Date
DK0745083T3 true DK0745083T3 (da) 1999-01-25

Family

ID=26893601

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95910286T DK0745083T3 (da) 1994-02-18 1995-02-17 2-Heteroaryl-5, 11-dihydro-6H-dipyrido[3, 2-b:2', 3'-e][1, 4]diazepiner og deres anvendelse til forebyggelse eller behandli

Country Status (15)

Country Link
EP (1) EP0745083B1 (da)
JP (1) JPH09509179A (da)
KR (1) KR970701190A (da)
CN (1) CN1043347C (da)
AT (1) ATE166353T1 (da)
AU (1) AU690646B2 (da)
CA (1) CA2183571A1 (da)
CO (1) CO4340691A1 (da)
DE (1) DE69502587T2 (da)
DK (1) DK0745083T3 (da)
ES (1) ES2118575T3 (da)
PL (1) PL181323B1 (da)
RU (1) RU2142464C1 (da)
TW (1) TW327171B (da)
WO (1) WO1995022545A1 (da)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5705499A (en) * 1995-10-06 1998-01-06 Boehringer Ingelheim Pharmaceuticals, Inc. 8-arylalkyl- and 8-arylheteroalkyl-5,11-dihydro-6H-dipyrido 3,2-B:2',3'-e! 1!diazepines and their use in the treatment of HIV-1 infection
US5747488A (en) * 1996-01-30 1998-05-05 Boehringer Ingelheim Pharmaceuticals, Inc. 2-aryl-5,11-dihydro-6H-dipyrido 3,2-B:2',3'-E! 1, 4!diazepines and their use in the treatment of HIV infection
CA2288787A1 (en) 1997-05-22 1998-11-26 G.D. Searle And Co. Pyrazole derivatives as p38 kinase inhibitors
US6514977B1 (en) 1997-05-22 2003-02-04 G.D. Searle & Company Substituted pyrazoles as p38 kinase inhibitors
US6979686B1 (en) 2001-12-07 2005-12-27 Pharmacia Corporation Substituted pyrazoles as p38 kinase inhibitors
US6716836B2 (en) * 2001-03-22 2004-04-06 Boehringer Ingelheim (Canada) Ltd. Non-nucleoside reverse transcriptase inhibitors
EP1737852A2 (en) * 2004-04-13 2007-01-03 Icagen, Inc. Polycyclic pyridines as potassium ion channel modulators
WO2005121140A1 (en) 2004-06-09 2005-12-22 Glaxo Group Limited Pyrrolopyridine derivatives
US8017781B2 (en) 2005-11-15 2011-09-13 Vertex Pharmaceuticals Incorporated Azaindazoles useful as inhibitors of kinases
WO2014060381A1 (de) 2012-10-18 2014-04-24 Bayer Cropscience Ag Heterocyclische verbindungen als schädlingsbekämpfungsmittel
US20150284380A1 (en) 2012-10-31 2015-10-08 Bayer Cropscience Ag Novel heterocyclic compounds as pest control agents

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3122670A1 (de) * 1981-06-06 1982-12-23 Dr. Karl Thomae Gmbh, 7950 Biberach "neue 1,4,9,10-tetrahydro-pyrazolo(4,3-e) pyrido(3,2-b)(1,4)diazepin-10-one, verfahren zu ihrer herstellung und ihre verwendung zur herstellung von pharmazeutischen wirkstoffen"
EP0410148B1 (en) * 1989-06-28 1994-04-06 Boehringer Ingelheim Pharmaceuticals Inc. Novel 5,11-dihydro-6H-dipyrido[3,2-b:2',3'-e][1,4]diazepin-6-ones and thiones and their use in the prevention or treatment of AIDS
CA2030056C (en) * 1989-11-17 1995-10-17 Karl D. Hargrave 5,11-dihydro-6h-dipyrido[3,2-b:2',3'-e][1,4]diazepines and their use in the prevention or treatment of hiv infection
ATE143018T1 (de) * 1991-02-07 1996-10-15 Boehringer Ingelheim Pharma Pyridobenzodiazepine, dipyrido-(3,2-b:2',3'-3> (1,4>-diazepine und deren verwendung in der vorbeugung und behandlung von aids

Also Published As

Publication number Publication date
DE69502587T2 (de) 1998-11-26
MX9603359A (es) 1998-07-31
TW327171B (en) 1998-02-21
KR970701190A (ko) 1997-03-17
AU690646B2 (en) 1998-04-30
EP0745083B1 (en) 1998-05-20
ATE166353T1 (de) 1998-06-15
ES2118575T3 (es) 1998-09-16
JPH09509179A (ja) 1997-09-16
CA2183571A1 (en) 1995-08-24
CN1043347C (zh) 1999-05-12
PL316006A1 (en) 1996-12-23
DE69502587D1 (de) 1998-06-25
CO4340691A1 (es) 1996-07-30
RU2142464C1 (ru) 1999-12-10
WO1995022545A1 (en) 1995-08-24
AU1845795A (en) 1995-09-04
PL181323B1 (pl) 2001-07-31
CN1138861A (zh) 1996-12-25
EP0745083A1 (en) 1996-12-04

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