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DK0607193T3 - Antifugale triazolderivater - Google Patents

Antifugale triazolderivater

Info

Publication number
DK0607193T3
DK0607193T3 DK92920368T DK92920368T DK0607193T3 DK 0607193 T3 DK0607193 T3 DK 0607193T3 DK 92920368 T DK92920368 T DK 92920368T DK 92920368 T DK92920368 T DK 92920368T DK 0607193 T3 DK0607193 T3 DK 0607193T3
Authority
DK
Denmark
Prior art keywords
pct
image
antifugal
date apr
triazole derivatives
Prior art date
Application number
DK92920368T
Other languages
Danish (da)
English (en)
Inventor
Andrew Simon Bell
Kenneth Richardson
Peter John Whittle
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of DK0607193T3 publication Critical patent/DK0607193T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62Oxygen or sulfur atoms
    • C07D213/70Sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Cephalosporin Compounds (AREA)
  • Pyridine Compounds (AREA)
DK92920368T 1991-10-10 1992-10-01 Antifugale triazolderivater DK0607193T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB919121456A GB9121456D0 (en) 1991-10-10 1991-10-10 Triazole antifungal agents
PCT/EP1992/002278 WO1993007139A1 (fr) 1991-10-10 1992-10-01 Angents antifongiques contenant du triazole

Publications (1)

Publication Number Publication Date
DK0607193T3 true DK0607193T3 (da) 2000-10-09

Family

ID=10702663

Family Applications (1)

Application Number Title Priority Date Filing Date
DK92920368T DK0607193T3 (da) 1991-10-10 1992-10-01 Antifugale triazolderivater

Country Status (13)

Country Link
US (1) US5541203A (fr)
EP (1) EP0607193B1 (fr)
JP (1) JPH07502022A (fr)
AT (1) ATE196293T1 (fr)
CA (1) CA2118937C (fr)
DE (1) DE69231445T2 (fr)
DK (1) DK0607193T3 (fr)
ES (1) ES2149777T3 (fr)
FI (1) FI108131B (fr)
GB (1) GB9121456D0 (fr)
GR (1) GR3034769T3 (fr)
PT (1) PT100942B (fr)
WO (1) WO1993007139A1 (fr)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9317491D0 (en) * 1993-08-23 1993-10-06 Fujisawa Pharmaceutical Co New compound and a process for preparation thereof
NZ270418A (en) * 1994-02-07 1997-09-22 Eisai Co Ltd Polycyclic triazole & imidazole derivatives, antifungal compositions
GB9512961D0 (en) * 1995-06-26 1995-08-30 Pfizer Ltd Antifungal agents
GB9605705D0 (en) * 1996-03-19 1996-05-22 Pfizer Ltd Therapeutic agents
KR100889937B1 (ko) 2007-08-06 2009-03-20 한미약품 주식회사 보리코나졸의 제조방법
GB2452049A (en) * 2007-08-21 2009-02-25 Alpharma Aps Process for the preparation of voriconazole
KR20180095109A (ko) * 2011-06-19 2018-08-24 비아멧 파마슈티컬즈(엔씨), 인코포레이티드 금속효소 억제제 화합물
CA2839769A1 (fr) 2011-06-19 2012-12-27 Viamet Pharmaceuticals, Inc. Composes inhibiteurs de metalloenzymes
EA026209B1 (ru) * 2012-01-20 2017-03-31 Ваймет Фармасьютикалс, Инк. Соединения, ингибирующие металлоферменты
TWI561515B (en) * 2012-03-16 2016-12-11 Viamet Pharmaceuticals Inc Metalloenzyme inhibitor compounds
AU2016265932B2 (en) 2015-05-18 2020-10-08 Viamet Pharmaceuticals (NC), Inc. Antifungal compounds
EP3544427A4 (fr) * 2016-11-22 2020-04-29 Dow Agrosciences Llc Composés fongicides et mélanges de régulation des champignons dans les céréales
AR110209A1 (es) * 2016-11-22 2019-03-06 Viamet Pharmaceuticals Inc Uso de un compuesto de difluoro-(2-hidroxipropil)piridina como fungicida para el control de hongos fitopatógenos en maíz
AU2017365179B2 (en) 2016-11-22 2021-09-02 Corteva Agriscience Llc Fungicidal compounds and mixtures for fungal control in cereals
WO2018098216A1 (fr) * 2016-11-22 2018-05-31 Vps-3, Inc. Utilisation d'un composé difluoro-(2-hydroxypropyl)pyridine en tant que fongicide pour lutter contre les champignons phytopathogènes de l'orge
US20190297888A1 (en) * 2016-11-22 2019-10-03 Dow Agrosciences Llc Fungicidal compounds and mixtures for fungal control in cereals
JP2019535756A (ja) * 2016-11-22 2019-12-12 ダウ アグロサイエンシィズ エルエルシー 殺真菌組成物および穀類における真菌防除のための混合物
CN110621157A (zh) * 2016-11-22 2019-12-27 美国陶氏益农公司 二氟-(2-羟基丙基)吡啶化合物作为用于防治稻子的植物病原真菌的杀真菌剂的用途
CN109996443A (zh) * 2016-11-22 2019-07-09 美国陶氏益农公司 二氟-(2-羟基丙基)吡啶化合物作为用于防治小麦的植物病原真菌的杀真菌剂的用途
RU2019118636A (ru) * 2016-11-22 2020-12-25 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Фунгицидные соединения и смеси для борьбы с грибковыми заболеваниями зерновых культур
AR110210A1 (es) * 2016-11-22 2019-03-06 Viamet Pharmaceuticals Inc Uso de un compuesto de difluoro-(2-hidroxipropil)piridina como fungicida para el control de la mancha foliar en remolacha azucarera

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE322526C (de) * 1918-08-31 1920-07-01 Hermann Meyer Sicherheitskettenverschluss fuer Korridortueren u. dgl.
EP0158741A3 (fr) * 1980-11-19 1986-02-12 Imperial Chemical Industries Plc Intermédiaires pour composés fongicides triazoles ou imidazoles
ES523184A0 (es) * 1982-06-17 1985-04-01 Pfizer Un procedimiento para la preparacion de un compuesto dotado de propiedades fungicidas
DE3245504A1 (de) * 1982-12-09 1984-06-14 Bayer Ag, 5090 Leverkusen Fungizide mittel, deren herstellung und verwendung
US4952232A (en) * 1987-04-29 1990-08-28 E. I. Du Pont De Nemours And Company Antifungal carbinols
DE3813841A1 (de) * 1987-06-03 1988-12-15 Bayer Ag Heterocyclische hydroxyethylazole
DE3732385A1 (de) * 1987-09-25 1989-04-06 Bayer Ag Hydroxyalkylcyclopropyl1-1,2,4-triazolyl- oder -imidazolyl-derivate und ihre verwendung als antimykotische mittel
EP0440608A1 (fr) * 1987-12-17 1991-08-14 E.I. Du Pont De Nemours And Company Carbinols antifongiques
NO171272C (no) * 1988-03-04 1993-02-17 Sankyo Co Analogifremgangsmaate til fremstilling av terapeutisk aktive 1,2,4-triazolforbindelser
GB8819308D0 (en) * 1988-08-13 1988-09-14 Pfizer Ltd Triazole antifungal agents
GB9002375D0 (en) * 1990-02-02 1990-04-04 Pfizer Ltd Triazole antifungal agents

Also Published As

Publication number Publication date
DE69231445D1 (de) 2000-10-19
CA2118937C (fr) 1998-04-28
CA2118937A1 (fr) 1993-04-15
EP0607193A1 (fr) 1994-07-27
GB9121456D0 (en) 1991-11-27
JPH07502022A (ja) 1995-03-02
ES2149777T3 (es) 2000-11-16
DE69231445T2 (de) 2001-01-11
EP0607193B1 (fr) 2000-09-13
GR3034769T3 (en) 2001-02-28
WO1993007139A1 (fr) 1993-04-15
FI941644L (fi) 1994-04-08
PT100942A (pt) 1993-10-29
FI941644A0 (fi) 1994-04-08
FI108131B (fi) 2001-11-30
ATE196293T1 (de) 2000-09-15
US5541203A (en) 1996-07-30
PT100942B (pt) 1999-07-30

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