DK0662952T3 - Fremgangsmåde til stereoselektiv syntese af 3-substituerede 2-sulfonylmethylpropionsyrer samt mellemprodukter - Google Patents
Fremgangsmåde til stereoselektiv syntese af 3-substituerede 2-sulfonylmethylpropionsyrer samt mellemprodukterInfo
- Publication number
- DK0662952T3 DK0662952T3 DK93921894T DK93921894T DK0662952T3 DK 0662952 T3 DK0662952 T3 DK 0662952T3 DK 93921894 T DK93921894 T DK 93921894T DK 93921894 T DK93921894 T DK 93921894T DK 0662952 T3 DK0662952 T3 DK 0662952T3
- Authority
- DK
- Denmark
- Prior art keywords
- pct
- sulfonylmethylpropionic
- intermediates
- acids
- substituted
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- -1 3-substituted 2-sulfonylmethylpropionic acids Chemical class 0.000 title 1
- 230000015572 biosynthetic process Effects 0.000 title 1
- 239000000543 intermediate Substances 0.000 title 1
- 230000000707 stereoselective effect Effects 0.000 title 1
- 238000003786 synthesis reaction Methods 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
- C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
- C07C323/56—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton containing six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C315/00—Preparation of sulfones; Preparation of sulfoxides
- C07C315/02—Preparation of sulfones; Preparation of sulfoxides by formation of sulfone or sulfoxide groups by oxidation of sulfides, or by formation of sulfone groups by oxidation of sulfoxides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C315/00—Preparation of sulfones; Preparation of sulfoxides
- C07C315/04—Preparation of sulfones; Preparation of sulfoxides by reactions not involving the formation of sulfone or sulfoxide groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C317/00—Sulfones; Sulfoxides
- C07C317/44—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
- C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
- C07C323/52—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE4233100A DE4233100A1 (de) | 1992-10-01 | 1992-10-01 | Verfahren zur stereoselektiven Synthese von 3-substituierten 2-Sulfonylmethylpropionsäuren sowie Zwischenprodukte |
| PCT/EP1993/002674 WO1994007850A1 (de) | 1992-10-01 | 1993-09-30 | Verfahren zur stereoselektiven synthese von 3-substituierten 2-sulfonylmethylpropionsäuren sowie zwischenprodukte |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK0662952T3 true DK0662952T3 (da) | 2000-03-13 |
Family
ID=6469439
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK93921894T DK0662952T3 (da) | 1992-10-01 | 1993-09-30 | Fremgangsmåde til stereoselektiv syntese af 3-substituerede 2-sulfonylmethylpropionsyrer samt mellemprodukter |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US5684185A (da) |
| EP (1) | EP0662952B1 (da) |
| JP (1) | JPH08501781A (da) |
| AT (1) | ATE183737T1 (da) |
| AU (1) | AU5110393A (da) |
| CA (1) | CA2146142A1 (da) |
| DE (2) | DE4233100A1 (da) |
| DK (1) | DK0662952T3 (da) |
| ES (1) | ES2137268T3 (da) |
| GR (1) | GR3031695T3 (da) |
| WO (1) | WO1994007850A1 (da) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE69732571T2 (de) * | 1996-09-27 | 2006-01-12 | Pharmacia & Upjohn Co., Kalamazoo | Beta-sulfonyl-hydroxamsäuren als matrix-metalloproteinaseinhibitoren |
| FR2772027B1 (fr) * | 1997-12-10 | 2000-02-04 | Fournier Ind & Sante | Procede de preparation asymetrique de derives de l'acide 2-mercaptomethyl-3-phenyl-propanoique, utilisation pour synthese de principes actifs chiraux |
| EP1392639B1 (en) * | 2001-05-03 | 2008-09-17 | Galileo Laboratories, Inc. | Pyruvate derivatives |
| WO2004009581A1 (ja) * | 2002-07-24 | 2004-01-29 | Mitsui Chemicals, Inc. | ２−アルキル−３−アミノチオフェン誘導体の製造法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4758584A (en) * | 1987-02-05 | 1988-07-19 | Ciba-Geigy Corporation | Antihypertensive 5-amino-4-hydroxyvaleryl derivatives substituted by sulphur-containing groups |
| DE3856166T2 (de) * | 1987-09-29 | 1998-08-06 | Banyu Pharma Co Ltd | N-Acylaminosäurederivate und deren Verwendung |
| US5095031A (en) * | 1990-08-20 | 1992-03-10 | Abbott Laboratories | Indole derivatives which inhibit leukotriene biosynthesis |
| DE4233099A1 (de) * | 1992-10-01 | 1994-04-07 | Hoechst Ag | Verfahren zur stereoselektiven Synthese von 3-substituierten 2-Thiomethylpropionsäuren |
-
1992
- 1992-10-01 DE DE4233100A patent/DE4233100A1/de not_active Withdrawn
-
1993
- 1993-09-30 US US08/411,832 patent/US5684185A/en not_active Expired - Fee Related
- 1993-09-30 ES ES93921894T patent/ES2137268T3/es not_active Expired - Lifetime
- 1993-09-30 JP JP6508713A patent/JPH08501781A/ja active Pending
- 1993-09-30 AU AU51103/93A patent/AU5110393A/en not_active Abandoned
- 1993-09-30 DK DK93921894T patent/DK0662952T3/da active
- 1993-09-30 AT AT93921894T patent/ATE183737T1/de not_active IP Right Cessation
- 1993-09-30 WO PCT/EP1993/002674 patent/WO1994007850A1/de not_active Ceased
- 1993-09-30 CA CA002146142A patent/CA2146142A1/en not_active Abandoned
- 1993-09-30 DE DE59309749T patent/DE59309749D1/de not_active Expired - Fee Related
- 1993-09-30 EP EP93921894A patent/EP0662952B1/de not_active Expired - Lifetime
-
1999
- 1999-11-03 GR GR990402786T patent/GR3031695T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| GR3031695T3 (en) | 2000-02-29 |
| ES2137268T3 (es) | 1999-12-16 |
| CA2146142A1 (en) | 1994-04-14 |
| US5684185A (en) | 1997-11-04 |
| EP0662952B1 (de) | 1999-08-25 |
| JPH08501781A (ja) | 1996-02-27 |
| ATE183737T1 (de) | 1999-09-15 |
| DE59309749D1 (de) | 1999-09-30 |
| AU5110393A (en) | 1994-04-26 |
| EP0662952A1 (de) | 1995-07-19 |
| WO1994007850A1 (de) | 1994-04-14 |
| DE4233100A1 (de) | 1994-04-07 |
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