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DK0594291T3 - Fremgangsmåder til fremstilling af 13-etherderivater af milbemyciner og mellemprodukter dertil - Google Patents

Fremgangsmåder til fremstilling af 13-etherderivater af milbemyciner og mellemprodukter dertil

Info

Publication number
DK0594291T3
DK0594291T3 DK93306899T DK93306899T DK0594291T3 DK 0594291 T3 DK0594291 T3 DK 0594291T3 DK 93306899 T DK93306899 T DK 93306899T DK 93306899 T DK93306899 T DK 93306899T DK 0594291 T3 DK0594291 T3 DK 0594291T3
Authority
DK
Denmark
Prior art keywords
intermediates
group
milbemycins
preparation
methods
Prior art date
Application number
DK93306899T
Other languages
English (en)
Inventor
Mitsugi Shibano
Mutsuo Suzuki
Shunshi Kojima
Original Assignee
Sankyo Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sankyo Co filed Critical Sankyo Co
Application granted granted Critical
Publication of DK0594291T3 publication Critical patent/DK0594291T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biochemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK93306899T 1992-09-01 1993-09-01 Fremgangsmåder til fremstilling af 13-etherderivater af milbemyciner og mellemprodukter dertil DK0594291T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP23344492 1992-09-01
JP26366092 1992-10-01
JP32284792 1992-12-02

Publications (1)

Publication Number Publication Date
DK0594291T3 true DK0594291T3 (da) 2003-01-27

Family

ID=27331997

Family Applications (1)

Application Number Title Priority Date Filing Date
DK93306899T DK0594291T3 (da) 1992-09-01 1993-09-01 Fremgangsmåder til fremstilling af 13-etherderivater af milbemyciner og mellemprodukter dertil

Country Status (13)

Country Link
US (2) US5461168A (da)
EP (1) EP0594291B1 (da)
JP (1) JP2654337B2 (da)
KR (1) KR0161541B1 (da)
AT (1) ATE229960T1 (da)
AU (1) AU666750B2 (da)
CA (1) CA2105251C (da)
DE (1) DE69332577T2 (da)
DK (1) DK0594291T3 (da)
ES (1) ES2186672T3 (da)
NZ (1) NZ248559A (da)
PT (1) PT594291E (da)
TW (1) TW262474B (da)

Families Citing this family (165)

* Cited by examiner, † Cited by third party
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JP4499847B2 (ja) * 1998-05-25 2010-07-07 三井化学アグロ株式会社 ミルベマイシン類の１３−エステル誘導体の製造法
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DE69332577T2 (de) 2003-11-20
NZ248559A (en) 1995-05-26
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US5625078A (en) 1997-04-29
EP0594291B1 (en) 2002-12-18
HK1010371A1 (en) 1999-06-17
PT594291E (pt) 2003-03-31
AU4497993A (en) 1994-03-10
CA2105251A1 (en) 1994-03-02
ES2186672T3 (es) 2003-05-16
AU666750B2 (en) 1996-02-22
EP0594291A1 (en) 1994-04-27
JP2654337B2 (ja) 1997-09-17
KR940007038A (ko) 1994-04-26
TW262474B (da) 1995-11-11
KR0161541B1 (ko) 1998-12-01
US5461168A (en) 1995-10-24
JPH06220068A (ja) 1994-08-09
CA2105251C (en) 2004-12-07

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