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DK0579785T3 - Substituerede benzhydrylaminer som tlslutningsmolekyler til fastfasepeptidsyntese - Google Patents

Substituerede benzhydrylaminer som tlslutningsmolekyler til fastfasepeptidsyntese

Info

Publication number
DK0579785T3
DK0579785T3 DK92917473.8T DK92917473T DK0579785T3 DK 0579785 T3 DK0579785 T3 DK 0579785T3 DK 92917473 T DK92917473 T DK 92917473T DK 0579785 T3 DK0579785 T3 DK 0579785T3
Authority
DK
Denmark
Prior art keywords
pct
solid phase
substituted
phase peptide
peptide synthesis
Prior art date
Application number
DK92917473.8T
Other languages
Danish (da)
English (en)
Inventor
Michal Lebl
Marcel Patek
Original Assignee
Michal Lebl
Marcel Patek
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Michal Lebl, Marcel Patek filed Critical Michal Lebl
Application granted granted Critical
Publication of DK0579785T3 publication Critical patent/DK0579785T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/16—Oxytocins; Vasopressins; Related peptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/26—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
    • C07C317/32—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/04—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
    • C07K1/042—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers characterised by the nature of the carrier
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/02—Ortho- or ortho- and peri-condensed systems
    • C07C2603/04—Ortho- or ortho- and peri-condensed systems containing three rings
    • C07C2603/06—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members
    • C07C2603/10—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings
    • C07C2603/12—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings only one five-membered ring
    • C07C2603/18—Fluorenes; Hydrogenated fluorenes
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Analytical Chemistry (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK92917473.8T 1991-04-12 1992-04-10 Substituerede benzhydrylaminer som tlslutningsmolekyler til fastfasepeptidsyntese DK0579785T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CS911030A CS103091A3 (en) 1991-04-12 1991-04-12 Protected substituted benzhydrylamines as shoulders for the synthesis ofpeptides on solid phase, process of their preparation and use

Publications (1)

Publication Number Publication Date
DK0579785T3 true DK0579785T3 (da) 1996-10-28

Family

ID=5343649

Family Applications (1)

Application Number Title Priority Date Filing Date
DK92917473.8T DK0579785T3 (da) 1991-04-12 1992-04-10 Substituerede benzhydrylaminer som tlslutningsmolekyler til fastfasepeptidsyntese

Country Status (12)

Country Link
US (2) US5684131A (fr)
EP (1) EP0579785B1 (fr)
JP (1) JP3634356B2 (fr)
AT (1) ATE139995T1 (fr)
CA (1) CA2109433C (fr)
CS (1) CS103091A3 (fr)
DE (1) DE69211990T2 (fr)
DK (1) DK0579785T3 (fr)
ES (1) ES2089548T3 (fr)
GR (1) GR3020463T3 (fr)
HU (1) HU222239B1 (fr)
WO (1) WO1992018144A1 (fr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0751779B1 (fr) * 1993-06-21 2001-12-19 Selectide Corporation Elements de liaison pouvant etre coupes de maniere selective, bases sur des esters de l'acide iminodiacetique
ES2115543B1 (es) * 1996-08-06 1999-02-16 Lipotec Sa Procedimiento para la obtencion de carbetocina y sus sales de adicion de acido farmaceuticamente aceptables o complejos de la misma.
GB9620202D0 (en) * 1996-09-27 1996-11-13 Rhone Poulenc Agriculture New herbicides
GB9621985D0 (en) 1996-10-22 1996-12-18 Peptide Therapeutics Ltd A solid-phase technology for the preparation of libraries of bi-directally functionalised drug-like molecules
AU1589099A (en) * 1997-11-18 1999-06-07 Rhone-Poulenc Rorer Pharmaceuticals Inc. Functionalized resin for the synthesis of amides and peptides
AU734992B2 (en) * 1997-11-26 2001-06-28 Medivir Uk Ltd A solid-phase technology for the preparation of combinatorial libraries through amide-bond anchoring
EP2275540B1 (fr) 1999-04-09 2016-03-23 Kyowa Hakko Kirin Co., Ltd. Procédé de contrôle de l'activité de molécule fonctionnelle immunologique

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3963701A (en) * 1972-04-17 1976-06-15 Richardson-Merrell Inc. Substituted benzhydryl lactamimide derivatives
FR2595695B1 (fr) * 1986-03-12 1988-12-02 Synthelabo Derives de n-(((hydroxy-2 phenyl) (phenyl) methylene) amino-2) ethyl) acetamide, leur preparation et leur application en therapeutique
ES2003864A4 (es) * 1986-12-24 1988-12-01 Monsanto Co Resina soporte para la sintesis de peptidos en fase solida.
ES2061714T3 (es) * 1987-12-22 1994-12-16 Hoechst Ag Grupos de anclaje inestables frente a acidos para la sintesis de amidas peptidicas mediante el metodo en fase solida.
JP2815362B2 (ja) * 1988-02-29 1998-10-27 中外製薬株式会社 ベンズヒドリルアミン誘導体及びその製法

Also Published As

Publication number Publication date
HU222239B1 (hu) 2003-05-28
HU9302867D0 (en) 1993-12-28
GR3020463T3 (en) 1996-10-31
DE69211990D1 (de) 1996-08-08
US5891995A (en) 1999-04-06
ATE139995T1 (de) 1996-07-15
HUT70198A (en) 1995-09-28
US5684131A (en) 1997-11-04
EP0579785A4 (en) 1994-07-06
EP0579785B1 (fr) 1996-07-03
JPH06506940A (ja) 1994-08-04
CA2109433C (fr) 2006-07-11
CS103091A3 (en) 1992-10-14
JP3634356B2 (ja) 2005-03-30
DE69211990T2 (de) 1996-11-28
EP0579785A1 (fr) 1994-01-26
WO1992018144A1 (fr) 1992-10-29
CA2109433A1 (fr) 1992-10-13
ES2089548T3 (es) 1996-10-01

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Legal Events

Date Code Title Description
AHB Application shelved due to non-payment