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DE60205870D1 - Orale pharmazeutische zusammensetzung aus cefpodoxim-proxetil - Google Patents

Orale pharmazeutische zusammensetzung aus cefpodoxim-proxetil

Info

Publication number
DE60205870D1
DE60205870D1 DE60205870T DE60205870T DE60205870D1 DE 60205870 D1 DE60205870 D1 DE 60205870D1 DE 60205870 T DE60205870 T DE 60205870T DE 60205870 T DE60205870 T DE 60205870T DE 60205870 D1 DE60205870 D1 DE 60205870D1
Authority
DE
Germany
Prior art keywords
pharmaceutical composition
oral pharmaceutical
proxetil
cefpodoxim
cefpodoxim proxetil
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE60205870T
Other languages
English (en)
Other versions
DE60205870T2 (de
Inventor
Mukta Malhotra
Rajeev Shankar Mathur
Rajiv Malik
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Ranbaxy Laboratories Ltd
Original Assignee
Ranbaxy Laboratories Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=11097036&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DE60205870(D1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ranbaxy Laboratories Ltd filed Critical Ranbaxy Laboratories Ltd
Application granted granted Critical
Publication of DE60205870D1 publication Critical patent/DE60205870D1/de
Publication of DE60205870T2 publication Critical patent/DE60205870T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • A61K31/546Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine containing further heterocyclic rings, e.g. cephalothin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DE60205870T 2001-02-27 2002-02-27 Orale pharmazeutische zusammensetzung aus cefpodoxim-proxetil Expired - Fee Related DE60205870T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IN190DE2001 2001-02-27
INDE00001900 2001-02-27
PCT/IB2002/000602 WO2002067943A1 (en) 2001-02-27 2002-02-27 Oral pharmaceutical composition of cefpodoxime proxetil

Publications (2)

Publication Number Publication Date
DE60205870D1 true DE60205870D1 (de) 2005-10-06
DE60205870T2 DE60205870T2 (de) 2006-06-29

Family

ID=11097036

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60205870T Expired - Fee Related DE60205870T2 (de) 2001-02-27 2002-02-27 Orale pharmazeutische zusammensetzung aus cefpodoxim-proxetil

Country Status (14)

Country Link
EP (1) EP1365764B1 (de)
JP (1) JP2004522782A (de)
KR (1) KR20030087009A (de)
CN (1) CN1505515A (de)
AT (1) ATE303149T1 (de)
AU (1) AU2002237462B2 (de)
BR (1) BR0207640A (de)
DE (1) DE60205870T2 (de)
EA (1) EA006974B1 (de)
ES (1) ES2248521T3 (de)
MX (1) MXPA03007678A (de)
NZ (1) NZ527867A (de)
OA (1) OA12687A (de)
WO (1) WO2002067943A1 (de)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6766376B2 (en) 2000-09-12 2004-07-20 Sn Acquisition, L.L.C Streaming media buffering system
ATE415150T1 (de) * 2002-08-16 2008-12-15 Orchid Chemicals & Pharm Ltd Pharmazeutische zusammensetzung mit verzögerte freisetzung enthaltend einen cephalosporin- antibiotikum
AU2002321743A1 (en) * 2002-08-19 2004-03-03 Orchid Health Care Sustained release pharmaceutical composition of a cephalosporin antibiotic
WO2004105728A2 (en) * 2003-05-27 2004-12-09 Ranbaxy Laboratories Limited Solid dispersions of cefpodoxime proxetil and processes for their preparation
JP2008540403A (ja) * 2005-05-05 2008-11-20 ルピン・リミテッド セファロスポリンの安定化経口用医薬組成物
JP2008540691A (ja) * 2005-05-16 2008-11-20 エラン・ファルマ・インターナショナル・リミテッド セファロスポリンを含むナノ粒子および放出制御組成物
US8900637B2 (en) * 2005-12-02 2014-12-02 Lupin Limited Stable taste masked formulations of cephalosporins
WO2008057058A1 (en) * 2006-11-10 2008-05-15 Nobel Ilac Sanayii Ve Ticaret As Oral pharmaceutical compositions
CN101278914B (zh) * 2008-01-02 2010-06-02 海南三叶美好制药有限公司 头孢泊肟酯干混悬剂组合物及其制备方法
TR201001417A1 (tr) * 2010-02-25 2011-09-21 Sanovel İlaç San. Ve Ti̇c. A. Ş. Geliştirilmiş çözünme hızına sahip sefdinir formülasyonu
TR201002878A2 (tr) 2010-04-13 2011-10-21 Bi̇lgi̇ç Mahmut Sefpodoksim proksetil içeren farmasötik bileşimler.
WO2011152805A2 (en) * 2010-06-03 2011-12-08 Mahmut Bilgic Pharmaceutical composition comprising cefpodoxime proxetil and clavulanic acid
TR201007107A1 (tr) * 2010-08-25 2012-03-21 B�Lg�� Mahmut Tat düzenleyici ajan içeren sefpodoksim proksetil formülasyonları.
TR201007106A1 (tr) * 2010-08-25 2012-03-21 Bi̇lgi̇ç Mahmut Sefpodoksim proksetil formülasyonları.
TR201009168A2 (tr) * 2010-11-05 2012-05-21 Bi̇lgi̇ç Mahmut Suda dağılan sefpodoksim proksetil formülasyonları.
EP2647648B1 (de) * 2010-12-03 2017-08-09 Nippon Soda Co., Ltd. Feste Darreichungsform enthaltend eine niedrigviskose HYDROXYALKYLCELLULOSE
WO2013145750A1 (ja) * 2012-03-29 2013-10-03 杏林製薬株式会社 カプセル製剤
ES2717282T3 (es) 2012-07-27 2019-06-20 Redhill Biopharma Ltd Formulaciones y métodos para fabricar formulaciones para su uso en la evacuación colónica
CN103142506B (zh) * 2013-04-03 2015-02-25 天津医药集团津康制药有限公司 一种头孢泊肟酯颗粒剂及其制备方法
US9603804B2 (en) 2013-04-25 2017-03-28 Kyorin Pharmaceutical Co., Ltd. Solid pharmaceutical composition
JP5700740B1 (ja) 2013-04-25 2015-04-15 杏林製薬株式会社 固形医薬組成物
KR101509168B1 (ko) * 2013-06-10 2015-04-06 한국화학연구원 세팔로스포린 항생제의 서방형 제제 및 이를 포함하는 서방형 약제학적 조성물
CN103301075B (zh) * 2013-06-28 2015-11-18 山东罗欣药业集团股份有限公司 一种头孢克肟组合物混悬颗粒剂及其制备方法
JP6292788B2 (ja) * 2013-07-30 2018-03-14 ライオン株式会社 錠剤及び錠剤の製造方法
JP2016204260A (ja) * 2013-10-04 2016-12-08 日本曹達株式会社 錠剤の製造方法
US10154993B2 (en) 2014-10-23 2018-12-18 Kyorin Pharmaceutical Co., Ltd. Solid pharmaceutical composition
CN104771368B (zh) * 2015-04-08 2017-12-22 石家庄四药有限公司 头孢泊肟酯速释制剂及其制备方法
CN113456599A (zh) * 2020-03-30 2021-10-01 洛阳惠中兽药有限公司 一种头孢泊肟酯片的制备方法及其制备的头孢泊肟酯片
CN113952313A (zh) * 2021-08-26 2022-01-21 宁夏医科大学 一种头孢呋辛酯胶囊及其制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4486425A (en) * 1980-09-30 1984-12-04 Sankyo Company Limited 7-[2-(2-Aminothiazol-4-yl)-2-(syn)-methoxyiminoacetamido]-3-methoxymethyl-3-cephem-4-carboxylates
US5929086A (en) * 1996-05-10 1999-07-27 Pharmacia & Upjohn Company Topical administration of antimicrobial agents for the treatment of systemic bacterial diseases
AT500063A1 (de) * 1999-11-23 2005-10-15 Sandoz Ag Beschichtete tablettenkerne
MXPA02012670A (es) * 2000-06-21 2003-10-06 Cubist Pharm Inc Composiciones y metodos para mejorar la absorcion oral de agentes anti-microbianos.

Also Published As

Publication number Publication date
DE60205870T2 (de) 2006-06-29
ATE303149T1 (de) 2005-09-15
MXPA03007678A (es) 2004-03-16
JP2004522782A (ja) 2004-07-29
EA006974B1 (ru) 2006-06-30
ES2248521T3 (es) 2006-03-16
NZ527867A (en) 2004-12-24
CN1505515A (zh) 2004-06-16
EA200300937A1 (ru) 2004-04-29
OA12687A (en) 2006-06-21
WO2002067943A1 (en) 2002-09-06
EP1365764B1 (de) 2005-08-31
BR0207640A (pt) 2004-07-27
EP1365764A4 (de) 2004-08-11
KR20030087009A (ko) 2003-11-12
EP1365764A1 (de) 2003-12-03
AU2002237462B2 (en) 2006-05-18

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Legal Events

Date Code Title Description
8363 Opposition against the patent
8339 Ceased/non-payment of the annual fee