CY1116689T1 - Imidazole derivatives as inhibitors of the PDE10A enzyme - Google Patents
Imidazole derivatives as inhibitors of the PDE10A enzymeInfo
- Publication number
- CY1116689T1 CY1116689T1 CY20151100805T CY151100805T CY1116689T1 CY 1116689 T1 CY1116689 T1 CY 1116689T1 CY 20151100805 T CY20151100805 T CY 20151100805T CY 151100805 T CY151100805 T CY 151100805T CY 1116689 T1 CY1116689 T1 CY 1116689T1
- Authority
- CY
- Cyprus
- Prior art keywords
- present
- subject
- compound
- formula
- effective amount
- Prior art date
Links
- 101001072037 Homo sapiens cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A Proteins 0.000 title abstract 2
- 239000003112 inhibitor Substances 0.000 title abstract 2
- 150000002460 imidazoles Chemical class 0.000 title 1
- 229940079865 intestinal antiinfectives imidazole derivative Drugs 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 6
- 238000000034 method Methods 0.000 abstract 4
- 239000003937 drug carrier Substances 0.000 abstract 1
- 206010013663 drug dependence Diseases 0.000 abstract 1
- 208000015122 neurodegenerative disease Diseases 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 208000020016 psychiatric disease Diseases 0.000 abstract 1
- 208000011117 substance-related disease Diseases 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Η παρούσα εφεύρεση απευθύνεται σε ενώσεις (I) οι οποίες είναι αναστολείς του ενζύμου PDE10A. Η εφεύρεση παρέχει μία φαρμακευτική σύνθεση η οποία περιλαμβάνει μία θεραπευτικά δραστική ποσότητα μίας ενώσεως της εφευρέσεως και έναν φαρμακευτικά αποδεκτό φορέα. Η παρούσα εφεύρεση παρέχει επίσης διαδικασίες παρασκευής των ενώσεων του τύπου I. Η παρούσα εφεύρεση περαιτέρω παρέχει μία μέθοδο αγωγής ενός ατόμου που πάσχει από μία νευροεκφυλιστική διαταραχή που περιλαμβάνει τη χορήγηση στο άτομο μίας θεραπευτικά δραστικής ποσότητας μίας ενώσεως του τύπου I. Η παρούσα εφεύρεση παρέχει επίσης μία μέθοδο αγωγής ενός ατόμου που πάσχει από τοξικομανία που περιλαμβάνει τη χορήγηση στο άτομο μίας θεραπευτικά δραστικής ποσότητας μίας ενώσεως του τύπου I. Η παρούσα εφεύρεση περαιτέρω παρέχει μία μέθοδο αγωγής, ενός ατόμου που πάσχει από μία ψυχιατρική διαταραχή που περιλαμβάνει τη χορήγηση στο άτομο μίας θεραπευτικά δραστικής ποσότητας μίας ενώσεως του τύπου I.The present invention is directed to compounds (I) which are inhibitors of the PDE10A enzyme. The invention provides a pharmaceutical composition comprising a therapeutically effective amount of a compound of the invention and a pharmaceutically acceptable carrier. The present invention also provides processes for the preparation of compounds of formula I. The present invention further provides a method of treating a subject suffering from a neurodegenerative disorder comprising administering to the subject a therapeutically effective amount of a compound of formula I. The present invention also provides a method of treating an individual suffering from drug dependence comprising administering to the subject a therapeutically effective amount of a compound of formula I. The present invention further provides a method of treatment g, a subject suffering from a psychiatric disorder comprising administering to the subject a therapeutically effective amount of a compound of formula I.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US41535610A | 2010-11-19 | 2010-11-19 | |
| DKPA201001045 | 2010-11-19 | ||
| EP11793325.9A EP2640731B9 (en) | 2010-11-19 | 2011-11-18 | Imidazole derivatives as pde10a enzyme inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CY1116689T1 true CY1116689T1 (en) | 2017-03-15 |
Family
ID=58459777
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CY20151100805T CY1116689T1 (en) | 2010-11-19 | 2015-09-14 | Imidazole derivatives as inhibitors of the PDE10A enzyme |
Country Status (1)
| Country | Link |
|---|---|
| CY (1) | CY1116689T1 (en) |
-
2015
- 2015-09-14 CY CY20151100805T patent/CY1116689T1/en unknown
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