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CU20110054A7 - HETEROARIL AMIDA DERIVATIVES AND THEIR USES AS GLUCOQUINASE ACTIVATORS - Google Patents

HETEROARIL AMIDA DERIVATIVES AND THEIR USES AS GLUCOQUINASE ACTIVATORS

Info

Publication number
CU20110054A7
CU20110054A7 CU20110054A CU20110054A CU20110054A7 CU 20110054 A7 CU20110054 A7 CU 20110054A7 CU 20110054 A CU20110054 A CU 20110054A CU 20110054 A CU20110054 A CU 20110054A CU 20110054 A7 CU20110054 A7 CU 20110054A7
Authority
CU
Cuba
Prior art keywords
activators
glucoquinase
heteroaril
amida
derivatives
Prior art date
Application number
CU20110054A
Other languages
Spanish (es)
Inventor
Meihua Mike Tu
Jeffrey Allen Pfefferkorn
John William Benbow
Jihong Lou
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Priority to CU20110054A priority Critical patent/CU20110054A7/en
Publication of CU20110054A7 publication Critical patent/CU20110054A7/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente invención proporciona compuestos de Fórmula (1A) ESPACIO PARA LA FÓRMULA que actúan como activadores de glucoquinasa; composiciones farmacéuticas de los mismos; y métodos para tratar enfermedades, trastornos o afecciones mediadas por glucoquinasa. X, Y, Z, R1, R2, R3 y R4 son como se han descrito en la presente memoria.The present invention provides compounds of Formula (1A) FORMULA SPACE that act as glucokinase activators; pharmaceutical compositions thereof; and methods for treating diseases, disorders or conditions mediated by glucokinase. X, Y, Z, R1, R2, R3 and R4 are as described herein.

CU20110054A 2011-03-11 2011-03-11 HETEROARIL AMIDA DERIVATIVES AND THEIR USES AS GLUCOQUINASE ACTIVATORS CU20110054A7 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CU20110054A CU20110054A7 (en) 2011-03-11 2011-03-11 HETEROARIL AMIDA DERIVATIVES AND THEIR USES AS GLUCOQUINASE ACTIVATORS

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CU20110054A CU20110054A7 (en) 2011-03-11 2011-03-11 HETEROARIL AMIDA DERIVATIVES AND THEIR USES AS GLUCOQUINASE ACTIVATORS

Publications (1)

Publication Number Publication Date
CU20110054A7 true CU20110054A7 (en) 2011-12-28

Family

ID=45508750

Family Applications (1)

Application Number Title Priority Date Filing Date
CU20110054A CU20110054A7 (en) 2011-03-11 2011-03-11 HETEROARIL AMIDA DERIVATIVES AND THEIR USES AS GLUCOQUINASE ACTIVATORS

Country Status (1)

Country Link
CU (1) CU20110054A7 (en)

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