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CO5560580A2 - Formulaciones de sucralosa para disumular sabores desagradables - Google Patents

Formulaciones de sucralosa para disumular sabores desagradables

Info

Publication number
CO5560580A2
CO5560580A2 CO04015498A CO04015498A CO5560580A2 CO 5560580 A2 CO5560580 A2 CO 5560580A2 CO 04015498 A CO04015498 A CO 04015498A CO 04015498 A CO04015498 A CO 04015498A CO 5560580 A2 CO5560580 A2 CO 5560580A2
Authority
CO
Colombia
Prior art keywords
sucralose
active compound
liquid
disguise
taste
Prior art date
Application number
CO04015498A
Other languages
English (en)
Inventor
David Jaeger
Jay Dickerson
Annabelle Mogavero
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23195896&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO5560580(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of CO5560580A2 publication Critical patent/CO5560580A2/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7012—Compounds having a free or esterified carboxyl group attached, directly or through a carbon chain, to a carbon atom of the saccharide radical, e.g. glucuronic acid, neuraminic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/10—Expectorants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/14—Antitussive agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pulmonology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biochemistry (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Rheumatology (AREA)
  • Otolaryngology (AREA)
  • Pain & Pain Management (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

1.- Una composición farmacéutica que tiene un pH de desde aproximadamente 2.0 a aproximadamente 5.0 que comprendei) una base excipiente líquida que contiene en 100 mI aproximadamente 50 mg a aproximadamente 300 mg de sucralosa para disimular un sabor amargo de cualquier ingrediente activo; yii) al menos un compuesto farmacéuticamente activo seleccionado del grupo que consiste de antihistaminas, descongestionantes, antitusivos, expectorantes, antibióticos, antineoplásticos,medicamentos anti-inflamatorios no esteroidales (NSAIDs) y medicamentos analgésicos, dicho compuesto farmacéuticamente activo disolviéndose o suspendiéndose en la base excipiente líquida.16.- Un método para disimular el sabor de al menos un compuesto activo farmacéuticamente aceptable con sabor desagradable, tal método comprende mezclar tal compuesto farmacéuticamente activo con sabor desagradable en una base excipiente líquida que contiene en 100 ml de base líquida aproximadamente 50 mg a aproximadamente 300 mg de sucralosa para disimular un sabor amargo de cualquier ingrediente activo, en donde la composición tiene un pH desde aproximadamente 2.0 a aproximadamente 5.0.
CO04015498A 2001-07-31 2004-02-23 Formulaciones de sucralosa para disumular sabores desagradables CO5560580A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US30891201P 2001-07-31 2001-07-31

Publications (1)

Publication Number Publication Date
CO5560580A2 true CO5560580A2 (es) 2005-09-30

Family

ID=23195896

Family Applications (1)

Application Number Title Priority Date Filing Date
CO04015498A CO5560580A2 (es) 2001-07-31 2004-02-23 Formulaciones de sucralosa para disumular sabores desagradables

Country Status (13)

Country Link
US (2) US20060121066A1 (es)
EP (1) EP1411955A4 (es)
JP (2) JP2004538309A (es)
AU (1) AU2002324579B2 (es)
BR (1) BR0211794A (es)
CA (1) CA2455939C (es)
CL (1) CL2004000208A1 (es)
CO (1) CO5560580A2 (es)
CR (1) CR7264A (es)
EC (1) ECSP044995A (es)
MX (1) MXPA04001026A (es)
NZ (1) NZ530889A (es)
WO (1) WO2003011306A1 (es)

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JP6565334B2 (ja) * 2014-06-18 2019-08-28 大正製薬株式会社 固形製剤
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Also Published As

Publication number Publication date
AU2002324579B2 (en) 2007-11-15
CA2455939C (en) 2011-03-22
CL2004000208A1 (es) 2005-03-18
ECSP044995A (es) 2004-04-28
JP2010090142A (ja) 2010-04-22
MXPA04001026A (es) 2005-06-20
WO2003011306A1 (en) 2003-02-13
CA2455939A1 (en) 2003-02-13
CR7264A (es) 2004-05-17
BR0211794A (pt) 2004-11-03
NZ530889A (en) 2005-03-24
EP1411955A4 (en) 2006-07-05
US20060121066A1 (en) 2006-06-08
EP1411955A1 (en) 2004-04-28
US20110136851A1 (en) 2011-06-09
JP2004538309A (ja) 2004-12-24

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