CO5160333A1 - TETRAZINE DERIVATIVES PESTICIDLY ACTIVE AND COMPOSITION THAT CONTAINS THEM - Google Patents
TETRAZINE DERIVATIVES PESTICIDLY ACTIVE AND COMPOSITION THAT CONTAINS THEMInfo
- Publication number
- CO5160333A1 CO5160333A1 CO00044621A CO00044621A CO5160333A1 CO 5160333 A1 CO5160333 A1 CO 5160333A1 CO 00044621 A CO00044621 A CO 00044621A CO 00044621 A CO00044621 A CO 00044621A CO 5160333 A1 CO5160333 A1 CO 5160333A1
- Authority
- CO
- Colombia
- Prior art keywords
- carbon atoms
- alkyl
- haloalkyl
- cycloalkyl
- alkylene
- Prior art date
Links
- 150000004905 tetrazines Chemical class 0.000 title 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 32
- 125000000217 alkyl group Chemical group 0.000 abstract 6
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 5
- 125000001188 haloalkyl group Chemical group 0.000 abstract 5
- 125000003545 alkoxy group Chemical group 0.000 abstract 4
- 125000002947 alkylene group Chemical group 0.000 abstract 4
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical compound [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 abstract 3
- 229910052799 carbon Inorganic materials 0.000 abstract 3
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 2
- 125000003118 aryl group Chemical group 0.000 abstract 2
- 125000001072 heteroaryl group Chemical group 0.000 abstract 2
- 229910052760 oxygen Inorganic materials 0.000 abstract 2
- -1 N (R8) 2 Chemical group 0.000 abstract 1
- 125000003342 alkenyl group Chemical group 0.000 abstract 1
- 125000004450 alkenylene group Chemical group 0.000 abstract 1
- 125000000304 alkynyl group Chemical group 0.000 abstract 1
- 125000004419 alkynylene group Chemical group 0.000 abstract 1
- 125000004429 atom Chemical group 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000000000 cycloalkoxy group Chemical group 0.000 abstract 1
- 125000004438 haloalkoxy group Chemical group 0.000 abstract 1
- 125000005347 halocycloalkyl group Chemical group 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- KIWSYRHAAPLJFJ-DNZSEPECSA-N n-[(e,2z)-4-ethyl-2-hydroxyimino-5-nitrohex-3-enyl]pyridine-3-carboxamide Chemical compound [O-][N+](=O)C(C)C(/CC)=C/C(=N/O)/CNC(=O)C1=CC=CN=C1 KIWSYRHAAPLJFJ-DNZSEPECSA-N 0.000 abstract 1
- 229910052717 sulfur Inorganic materials 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/713—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with four or more nitrogen atoms as the only ring hetero atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
- C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D257/08—Six-membered rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
La presente invención se refiere a compuestos de la fórmula general:<EMI FILE="00044621_1" ID="1" IMF=JPEG >en donde:T-V es -N=N- ó -NH-NH-; X1 es R1;X2 y X3 son cada uno independientemente del otro, H ó R1;R1 es, por ejemplo, halógeno, CN, NO2, alquilo de 1 a 6 átomos de carbono, cicloalquilo de 3 a 8 átomos de carbono, haloalquilo de 1 a 6 átomos de carbono, halocicloalquilo de 3 a 8 átomos de carbono, alcoxilo de 1 a 6 átomos de carbono, cicloalcoxilo de 3 a 8 átomos de carbono, o haloalcoxilo de 1 a 6 átomos de carbono;Ar1 es arilo o heteroarilo insustituido o mono- a tetra-sustituido;Ar2 es arilo o heteroarilo insustituido o mono- a penta-sustituido;A es un solo enlace, alquileno de 1 a 12 átomos de carbono, O, O(alquileno de 1 a 12 átomos de carbono), S(O)n, S(O)n(alquileno de 1 a 12 átomos de carbono), alquenileno de 2 a 8 átomos de carbono,alquinileno de 2 a 8 átomos de carbono; NR6, NR6(alquileno de 1 a 12 átomos de carbono), ó C(=Z); Z es O, NR4, NNR4R5 ó NOR4;R2 es H, alquilo de 1 a 6 átomos de carbono, o cicloalquilo de 3 a 8 átomos de carbono; R4 y R5 son cada uno independientemente del otro, H, alquilo de 1 a 6 átomos de carbono, o haloalquilo de 1 a 6 átomos de carbono;R6 es H, alquilo de 1 a 6 átomos de carbono, cicloalquilo de 3 a 8 átomos de carbono, haloalquilo de 1 a 6 átomos de carbono, alquenilo de 2 a 8 átomos de carbono, alquinilo de 2 a 8 átomos de carbono, arilalquilo de 1 a 6 átomos de carbono, (CH2)pC(0)R7 ó alcoxilo de 1 a 6 átomos de carbono-alquilo de 2 a 6 .átomos de carbono;R7 es H, alquilo de 1 a 6 átomos de carbono, cicloalquilo de 3 a 8 átomos de carbono, haloalquilo de 1 a 6 átomos de carbono, alcoxilo de 1 a 6 átomos de carbono, N(R8)2, ó alcoxilo de 1 a 6 átomos de carbono-alquilo de 2 a 6 átomos de carbono;R8 es H, alquilo de 1 a 6 átomos de carbono, cicloalquilo de 3 a 8 átomos de carbono, haloalquilo de 1 a 6 átomos de carbono, o arilalquilo de 1 a 6 átomos de carbono;n es 0, 1, ó 2;The present invention relates to compounds of the general formula: <EMI FILE = "00044621_1" ID = "1" MFI = JPEG> wherein: T-V is -N = N- or -NH-NH-; X1 is R1; X2 and X3 are each independently of each other, H or R1; R1 is, for example, halogen, CN, NO2, alkyl of 1 to 6 carbon atoms, cycloalkyl of 3 to 8 carbon atoms, haloalkyl of 1 to 6 carbon atoms, halocycloalkyl of 3 to 8 carbon atoms, alkoxy of 1 to 6 carbon atoms, cycloalkoxy of 3 to 8 carbon atoms, or haloalkoxy of 1 to 6 carbon atoms; Ar1 is unsubstituted aryl or heteroaryl or mono- to tetra-substituted; Ar2 is unsubstituted aryl or heteroaryl or mono- to penta-substituted; A is a single bond, alkylene of 1 to 12 carbon atoms, O, O (alkylene of 1 to 12 carbon atoms) , S (O) n, S (O) n (alkylene of 1 to 12 carbon atoms), alkenylene of 2 to 8 carbon atoms, alkynylene of 2 to 8 carbon atoms; NR6, NR6 (alkylene of 1 to 12 carbon atoms), or C (= Z); Z is O, NR4, NNR4R5 or NOR4; R2 is H, alkyl of 1 to 6 carbon atoms, or cycloalkyl of 3 to 8 carbon atoms; R4 and R5 are each independently of each other, H, alkyl of 1 to 6 carbon atoms, or haloalkyl of 1 to 6 carbon atoms; R6 is H, alkyl of 1 to 6 carbon atoms, cycloalkyl of 3 to 8 atoms carbon, haloalkyl of 1 to 6 carbon atoms, alkenyl of 2 to 8 carbon atoms, alkynyl of 2 to 8 carbon atoms, arylalkyl of 1 to 6 carbon atoms, (CH2) pC (0) R7 or alkoxy of 1 to 6 carbon atoms-alkyl of 2 to 6 carbon atoms; R7 is H, alkyl of 1 to 6 carbon atoms, cycloalkyl of 3 to 8 carbon atoms, haloalkyl of 1 to 6 carbon atoms, alkoxy of 1 to 6 carbon atoms, N (R8) 2, or alkoxy of 1 to 6 carbon atoms-alkyl of 2 to 6 carbon atoms; R8 is H, alkyl of 1 to 6 carbon atoms, cycloalkyl of 3 to 8 carbon atoms, haloalkyl of 1 to 6 carbon atoms, or arylalkyl of 1 to 6 carbon atoms, n is 0, 1, or 2;
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH114899 | 1999-06-21 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CO5160333A1 true CO5160333A1 (en) | 2002-05-30 |
Family
ID=4203614
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CO00044621A CO5160333A1 (en) | 1999-06-21 | 2000-06-15 | TETRAZINE DERIVATIVES PESTICIDLY ACTIVE AND COMPOSITION THAT CONTAINS THEM |
Country Status (6)
| Country | Link |
|---|---|
| EP (1) | EP1187818A1 (en) |
| JP (1) | JP2003502413A (en) |
| AU (1) | AU5405600A (en) |
| CO (1) | CO5160333A1 (en) |
| EG (1) | EG22089A (en) |
| WO (1) | WO2000078739A1 (en) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN105104407B (en) * | 2012-03-10 | 2017-06-16 | 陕西韦尔奇作物保护有限公司 | A kind of Efficient insecticidal composition |
| CN102702122B (en) * | 2012-05-16 | 2014-05-14 | 南通大学 | Method for preparing tetrazine by oxidizing dihydro tetrazine |
| CN105130962B (en) * | 2015-09-06 | 2017-09-26 | 浙江博仕达作物科技有限公司 | A kind of tetrazine pyrazoles acaricide |
| CN105061399B (en) * | 2015-09-06 | 2017-03-22 | 青岛科技大学 | Fluorine-containing tetrazine pyridine compounds and application thereof |
| CN105037329B (en) * | 2015-09-06 | 2017-03-22 | 青岛科技大学 | Fluorine-containing tetrazine pyrazol acaricide |
| WO2018006795A1 (en) * | 2016-07-05 | 2018-01-11 | 广州再极医药科技有限公司 | Aromatic acetylene or aromatic ethylene compound, intermediate, preparation method, pharmaceutical composition and use thereof |
| CN109988144B (en) | 2017-12-29 | 2024-07-05 | 广州再极医药科技有限公司 | Aromatic vinyl or aromatic ethyl derivative, preparation method, intermediate, pharmaceutical composition and application thereof |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CY1243A (en) * | 1978-05-25 | 1984-06-29 | Fbc Ltd | Acaricidal and ovicidal heterocyclic compounds and compositions and process for their preparation |
| EP0029657A3 (en) * | 1979-11-16 | 1981-08-26 | Fbc Limited | Pesticidal tetrazines, their use and compositions, processes for their preparation and preparation intermediates |
| DE3173083D1 (en) * | 1980-03-22 | 1986-01-16 | Fbc Ltd | Pesticidal heterocyclic compounds, processes for preparing them, compositions containing them, and their use |
| HU212613B (en) * | 1993-07-21 | 1996-09-30 | Chinoin Gyogyszer Es Vegyeszet | Tetrazine-derivatives, process for production of the compounds, acaricidal,larvicidal and ovicidal compositions containing the compounds as active ingredient and process for their production and their use |
-
2000
- 2000-06-15 CO CO00044621A patent/CO5160333A1/en unknown
- 2000-06-19 JP JP2001504905A patent/JP2003502413A/en active Pending
- 2000-06-19 EP EP00938800A patent/EP1187818A1/en not_active Withdrawn
- 2000-06-19 EG EG20000788A patent/EG22089A/en active
- 2000-06-19 WO PCT/EP2000/005627 patent/WO2000078739A1/en not_active Ceased
- 2000-06-19 AU AU54056/00A patent/AU5405600A/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2000078739A1 (en) | 2000-12-28 |
| EP1187818A1 (en) | 2002-03-20 |
| AU5405600A (en) | 2001-01-09 |
| JP2003502413A (en) | 2003-01-21 |
| EG22089A (en) | 2002-07-31 |
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