CO5070569A1 - COMPOUND OF AMINOAZOL OR A PHARMACEUTICALLY ACCEPTABLE SALT OF THE SAME AND MEDICINAL PRODUCT CONTAINING THEM - Google Patents
COMPOUND OF AMINOAZOL OR A PHARMACEUTICALLY ACCEPTABLE SALT OF THE SAME AND MEDICINAL PRODUCT CONTAINING THEMInfo
- Publication number
- CO5070569A1 CO5070569A1 CO99031508A CO99031508A CO5070569A1 CO 5070569 A1 CO5070569 A1 CO 5070569A1 CO 99031508 A CO99031508 A CO 99031508A CO 99031508 A CO99031508 A CO 99031508A CO 5070569 A1 CO5070569 A1 CO 5070569A1
- Authority
- CO
- Colombia
- Prior art keywords
- compound
- aminoazol
- pharmaceutically acceptable
- acceptable salt
- same
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 2
- 150000003839 salts Chemical class 0.000 title abstract 2
- QLSWIGRIBOSFMV-UHFFFAOYSA-N 1h-pyrrol-2-amine Chemical compound NC1=CC=CN1 QLSWIGRIBOSFMV-UHFFFAOYSA-N 0.000 title 1
- 229940126601 medicinal product Drugs 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención se relaciona con un compuesto de la fórmula (I):<EMI FILE="99031508_1" ID="1" IMF=JPEG >o una sal de el mismo, métodos para su preparación y composiciones farmacéuticas que los contienen.The present invention relates to a compound of the formula (I): <EMI FILE = "99031508_1" ID = "1" IMF = JPEG> or a salt thereof, methods for its preparation and pharmaceutical compositions containing them.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE1998124175 DE19824175A1 (en) | 1998-05-29 | 1998-05-29 | Amino azole compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CO5070569A1 true CO5070569A1 (en) | 2001-08-28 |
Family
ID=7869385
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CO99031508A CO5070569A1 (en) | 1998-05-29 | 1999-05-21 | COMPOUND OF AMINOAZOL OR A PHARMACEUTICALLY ACCEPTABLE SALT OF THE SAME AND MEDICINAL PRODUCT CONTAINING THEM |
Country Status (4)
| Country | Link |
|---|---|
| AU (1) | AU4501699A (en) |
| CO (1) | CO5070569A1 (en) |
| DE (1) | DE19824175A1 (en) |
| WO (1) | WO1999062892A1 (en) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6191160B1 (en) | 1998-11-10 | 2001-02-20 | Merck & Co., Inc. | Spiro-indolines as Y5 receptor antagonists |
| US6340683B1 (en) | 1999-04-22 | 2002-01-22 | Synaptic Pharmaceutical Corporation | Selective NPY (Y5) antagonists (triazines) |
| US6989379B1 (en) | 1999-04-22 | 2006-01-24 | H. Lundbick A/S | Selective NPY (Y5) antagonists |
| EP1816127A1 (en) | 1999-04-22 | 2007-08-08 | H. Lundbeck A/S | Triazine derivatives for use as selective npy (y5) antagonists |
| US6218408B1 (en) | 1999-06-30 | 2001-04-17 | Synaptic Pharmaceutical Corporation | Selective NPY (Y5) antagonists (bicyclics) |
| US6214853B1 (en) | 1999-06-30 | 2001-04-10 | Synaptic Pharmaceutical Corporation | Selective NPY (Y5) antagonists (bicyclics) |
| US7273880B2 (en) | 1999-06-30 | 2007-09-25 | H. Lunbeck A/S | Selective NPY (Y5) antagonists |
| WO2001017995A1 (en) | 1999-09-10 | 2001-03-15 | Merck & Co., Inc. | Tyrosine kinase inhibitors |
| AU2001246494A1 (en) * | 2000-03-03 | 2001-09-12 | Novartis Ag | Condensed thiazolamines and their use as neuropeptide y5 antagonists |
| CA2450562A1 (en) | 2001-06-22 | 2003-01-03 | Merck & Co., Inc. | Tyrosine kinase inhibitors |
| WO2003051356A1 (en) * | 2001-12-17 | 2003-06-26 | Merck & Co., Inc. | Method for treating circadian rhythm disruptions |
| JP2005526732A (en) | 2002-02-28 | 2005-09-08 | エフ.ホフマン−ラ ロシュ アーゲー | Thiazole derivatives as NPY receptor antagonists |
| US6872724B2 (en) | 2002-07-24 | 2005-03-29 | Merck & Co., Inc. | Polymorphs with tyrosine kinase activity |
| CA2493712A1 (en) * | 2002-08-07 | 2004-02-19 | F. Hoffmann-La Roche Ag | Aminothiazole derivatives as npy5 receptor inhibitors |
| AU2004263312A1 (en) | 2003-08-12 | 2005-02-17 | F. Hoffmann-La Roche Ag | Thiazole derivatives as NPY antagonists |
| AU2004263311A1 (en) | 2003-08-12 | 2005-02-17 | F. Hoffmann-La Roche Ag | 2-amino-5-benzoylthiazole NPY antagonists |
| AR081626A1 (en) | 2010-04-23 | 2012-10-10 | Cytokinetics Inc | AMINO-PYRIDAZINIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM AND USE OF THE SAME TO TREAT CARDIAC AND SKELETIC MUSCULAR DISORDERS |
| US9133123B2 (en) | 2010-04-23 | 2015-09-15 | Cytokinetics, Inc. | Certain amino-pyridines and amino-triazines, compositions thereof, and methods for their use |
| AR081331A1 (en) | 2010-04-23 | 2012-08-08 | Cytokinetics Inc | AMINO- PYRIMIDINES COMPOSITIONS OF THE SAME AND METHODS FOR THE USE OF THE SAME |
| US8759380B2 (en) | 2011-04-22 | 2014-06-24 | Cytokinetics, Inc. | Certain heterocycles, compositions thereof, and methods for their use |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE4326465A1 (en) * | 1993-01-20 | 1995-02-09 | Thomae Gmbh Dr K | Amino acid derivatives, pharmaceutical compositions containing these compounds and process for their preparation |
| DE19544687A1 (en) * | 1995-11-30 | 1997-06-05 | Thomae Gmbh Dr K | Amino acid derivatives, medicaments containing these compounds and processes for their preparation |
| AU7692696A (en) * | 1995-12-01 | 1997-06-27 | Novartis Ag | Heteroaryl derivatives |
| TW399051B (en) * | 1996-01-31 | 2000-07-21 | Ssp Co Ltd | A novel benzoazine thiazolidinedione derivative and pharmaceutical composition for reducing blood glucose |
| TR199902442T2 (en) * | 1997-01-28 | 2000-07-21 | Merck & Co.,Inc. | Thiazole benzenesulfonamides as β3 agonists in the treatment of sugar and obesity. |
| SG72827A1 (en) * | 1997-06-23 | 2000-05-23 | Hoffmann La Roche | Phenyl-and aminophenyl-alkylsulfonamide and urea derivatives |
-
1998
- 1998-05-29 DE DE1998124175 patent/DE19824175A1/en not_active Ceased
-
1999
- 1999-05-21 CO CO99031508A patent/CO5070569A1/en unknown
- 1999-05-27 WO PCT/EP1999/003682 patent/WO1999062892A1/en not_active Ceased
- 1999-05-27 AU AU45016/99A patent/AU4501699A/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO1999062892A1 (en) | 1999-12-09 |
| AU4501699A (en) | 1999-12-20 |
| DE19824175A1 (en) | 1999-12-02 |
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