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CN1496737A - Method for treating inflammation of muscular skeleton and connective tissue - Google Patents

Method for treating inflammation of muscular skeleton and connective tissue Download PDF

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Publication number
CN1496737A
CN1496737A CNA2003101017637A CN200310101763A CN1496737A CN 1496737 A CN1496737 A CN 1496737A CN A2003101017637 A CNA2003101017637 A CN A2003101017637A CN 200310101763 A CN200310101763 A CN 200310101763A CN 1496737 A CN1496737 A CN 1496737A
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patient
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L・迪安・帕克斯
L·迪安·帕克斯
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李 毅
李毅
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Abstract

A method of treating said musculoskeletal and connective tissue inflammations including osteoarthritis and associated articular and periarticular inflammations, and non-articular Rheumatism including capsulitis, tendonitis, fibrositis, and perarticular inflammations is disclosed. The method includes administering to a patient of a therapeutically effective amount of a composition comprising 13-cis-retinoic acid. Preferably, the treatment method includes administering to a patient of an initial dosage of a composition comprising 13-cis-retinoic acid for an initial treatment period, and thereafter administering a maintenance dosage of the composition.

Description

A kind of method for the treatment of muscle skeleton and ICT
Technical field
The present invention relates to a kind of method for the treatment of muscle skeleton and ICT.More particularly, this method is used the 13-cis-retinoic acid and is treated muscle skeleton and ICT effectively, this muscle skeleton comprises osteoarthritis and joint and the periarthritis disease relevant with osteoarthritis with ICT, and nonarticular rheumatism, nonarticular rheumatism comprises capsulitis, tendinitis, fibrositis and periarthritis disease.
Background technology
Muscle skeleton and ICT are a large amount of crowds' of infringement common diseases.Some common muscle skeletons comprise osteoarthritis and joint and the periarthritis disease relevant with osteoarthritis with ICT, and nonarticular rheumatism, and nonarticular rheumatism comprises capsulitis, tendinitis, fibrositis and periarthritis disease.
Osteoarthritis is a kind of the most common arthritis type, is more common in the old people.Osteoarthritis is a kind of joint disease of main invasion and attack cartilage.Cartilage is the smooth tissue that intraarticular covers epiphysis.Healthy cartilage can make skeleton slide mutually freely, the energy that vibrations are produced in the time of also can the absorbing bodily motion.When osteoarthritis takes place when, the top layer disintegrate wearing and tearing of cartilage.This makes and the mutual friction of subchondral skeleton phase causes pain, swelling and joint movement disorder.As time goes on, the joint will be out of shape.In addition, also can grow bony spur at the edge in joint.Fritter bone or cartilage can come off, and float in the joint space.This can cause more serious pain and damage.The people who suffers from osteoarthritis generally has the symptom of arthralgia and limitation of activity.Different with the arthritis of other types is that osteoarthritis is only encroached on the joint, and does not encroach on the internal.
Osteoarthritis is one of common cause that causes adult's physical disabilities.In the U.S., there are more than 2,000 ten thousand people may suffer from this disease.Some youngsters are suffered from osteoarthritis owing to the joint is injured, but osteoarthritis mainly betides the old people.In fact, in the crowd below 65 years old, at least one joint that surpasses the people of half suffers from the osteoarthritis of making a definite diagnosis through X-ray.Because U.S. old people's number is in continuous increase, so osteoarthritis patient's number also is constantly to increase.The men and women all can suffer from this disease.
The measure of treatment osteoarthritis at present comprises exercise, endo-medicine, rest, joint maintenance, surgical operation, pain relief technology, alternative medicine and controlling body weight etc.The medicine of treatment osteoarthritis commonly used comprises nonsteroidal anti-inflammatory agent (NSAIDs), as aspirin, Advil (ibuprofen), Motrin IB (ibuprofen), Aleve (naproxen sodium), ketoprofen; The local pain that directly applies to skin is alleviated Emulsion, wiping agent and spray (as capsaicin Emulsion); Cortical steroid, a kind of natural in vivo synthetic or as the powerful antiinflammatory hormone of medicine synthetic, be injected into usually and encroached on the joint, with respite pain; And hyaluronic acid, a kind of novel drugs that is used for joint injection is used for the treatment of the knee osteoarthritis.Adopt surgical operation can reproduce (polishing) surface of bone, restore skeleton and joint replacement.For some patients, surgical operation helps to alleviate pain and the deformity due to the osteoarthritis.Osteoarthritis is a kind of chronic disease, although multiple medicine has been used for the treatment of this disease, this is not effective aspect sick to these medicines in long-term control and prevention.
A kind of most common form of capsulitis is an adhesive capsulitis, is also referred to as " congealed shoulder ", and the pain of this disease can cause the movable serious forfeiture of shoulder.Its symptom mainly is that pain and the range of motion that the serious inflammation by joint capsule causes dwindles.When motion reached the limit of range of activity, shoulder was understood pain usually, and the aggravation at night.The reason of this disease is not also understood now.There is a kind of theory to think what autoimmune response caused.Adhesive capsulitis can be secondary to other damages, and these damages make the shoulder can not normal activity.After a common example is wrist fractures, may need to place sling to reach several weeks arm, so just limit the activity of shoulder.In addition, when other shoulder illness occurring, " congealed shoulder " also can take place.Sometimes, problem such as tear such as bursitis, bump syndrome or local rotator cuff and also can cause congealed shoulder.
Usually, before solving basic problem, must at first treat adhesive capsulitis to recover the shoulder activity.The treatment of congealed shoulder may baffle or slowly.Initial treatment also can be used anti-inflammatory drug at reducing inflammation and adopting the stretching, extension scheme to increase the shoulder range of activity.Startup and lasting physiotherapy also are important to recover the shoulder activity.Injection cortisone and long-acting anesthetis also can control inflammation preferably, and make the stretching, extension therapeutic scheme more effective.Most of cases finally can improve.But generally, the range of activity of shoulder can not recovered fully.
Tendinitis be with tendon on the skeleton adhere to the place pain be a kind of inflammation of feature.The tendinitis predilection site comprises shoulder rotator cuff (spinal column and biceps tendon); Wrist extensor (lateral epicondylitis and tennis) and ancon musculus flexor (middle epicondylitis) adhere to the place; The ilium shin band of patellar ligament, state portion tendon and knee; Shank ossa tibiale posterius tendon adhere to place's (outer shin inflammation); The heel string of heel.Tendinitis is caused by excessive use mostly.Usually can observe the pathological change that conforms to chronic inflammatory disease.Also can observe with the cellular atrophy is the tissue degeneratiaon of feature.Calcium salt can precipitate (as calcific tendinitis) along the direction of tendon, and shoulder is modal site of pathological change.Chronic tendinitis can cause tendon to die down and the Secondary cases fracture.Middle age is the most responsive to the development of tendinitis.
The purpose of Drug therapy tendinitis is pain management and reduces inflammation.Existing treatment measure comprises nonsteroidal anti-inflammatory agent (NSAIDs), splinting or fixation; And the lignocaine/steroid injection around the tendon.Non-steroidal antiinflammatory drugs comprises ibuprofen, flurbiprofen, naproxen, mefenamic acid, ketoprofen, indometacin and piroxicam.
Fibrositis is a kind of more common nonarticular rheumatism.It may be partial or disperse that fiber is knitted class.The dispersivity fibrositis that occurs in a plurality of positions of health is also referred to as fibromyalgia.Fibrositis is and muscle and the disease that contiguous connective tissue is touched a tender spot, pain is relevant that it shows as the pain at fibrous tissue, muscle, tendon, ligament and other position with fibromyalgia.Any fibrillar muscle is organized all effected, but the fibrillar muscle of occipitalia, cervical region, shoulder, chest, back and thigh organize be subject to especially the infringement.For fibromyalgia, can discern " trigger point " that different focuses are touched a tender spot, and General Symptoms can often occur also as fatigue, insomnia and depression.
The pain of fibrositis and sore spot feature are attributable to Several Factors.At first, the local inflammation that may exist virus to cause.This as the back or cervical region got flu.The myalgia of general is to be caused by the general toxin in the blood due to the viral infection, and this viral infection also can betide other position usually except the muscle or joint capsule place that occur in pain.In addition, a common cause of local trigger point formation is so-called " referred pain ".Is by wound in the many joints that link to each other with spinal column as the strain or the common site of spraining the inflammation that causes.Because these joints are near the nerve sheath of the nerve that spreads out from spinal cord, these nerve sheath that are called as " dura mater " can be upset and pain or be inflamed.When these pathological changes took place, problem did not just lie in and has been subjected to infringement place, but is deep in the inflammation intraarticular and nerve sheath.If pain and tenderness continue a plurality of months, will cause chronic pain and ankylosis.Above-mentioned mechanism can occur in a plurality of different parts of health.Ancon, heel, back, cervical region and the shoulder relevant with the painful trigger point is common site of pathological change.The existing measure of treatment fibrositis comprises cortisone injection, nonsteroidal anti-inflammatory agent (NSAIDs) and physiotherapy.For fibromyalgia, the treatment measure comprises that the tricyclic antidepressants, exercise and the oneself that are used for relaxed muscle and improve sleep quality loosen.
Many muscle skeletons and ICT are chronic, and can cause the afunction of chronic local pain and affected areas.These diseases are patient harm from the health not only, and influences their economy and life style.Economic implication comprises that medical expense and the disabled salary that causes descend.To the influence of life style comprise that depression, anxiety, helplessness, daily routines are limited, work limit, daily family is happy and the forfeiture of responsibility.
Sell by the Hoffmann-La Roch company of New Jersey nanotesla profit, trade mark is Accutane The 13-cis-retinoic acid, be that usually said tretinoin is also referred to as Accutane, described 13-cis-retinoic acid is as the dermatological medicament of part or oral application, and is long ago just known, and this medicament can be used for treating acne vulgaris and other several dermatosiss.The 13-cis-retinoic acid can suppress the effect and the keratinization of sebaceous gland.Accutane The definite mechanism of action of treatment acne is not also understood.Because tretinoin is a kind of teratogen, and the relevant mutagenesis of medicine is therewith arranged, so it only is used for the treatment of the invalid serious acne of additive method.
Since 1992, occurred about the bibliographical information of 13-cis-retinoic acid to the latent effect of Human Prostate Cancer Cells.U.S. Patent number 5,612,354 (Sanzet etc.) have disclosed the method that a kind of treatment suffers from hyperplasia and is divided into the mammalian diseases of feature unusually, and this method comprises that by the quinoline that (the 1H-pyrroles-1-ylmethyl) of mammal whole body or local application effective dose replaced the 13-cis-retinoic acid treats.Because the quinoline that (1H-pyrroles-1-ylmethyl) replaces has the ability that postpones retinoic acid metabolism, so be considered to be used for the treatment of acne.
As mentioned above, obviously, the medicine that can treat muscle skeleton and ICT is effectively still had very big demand.The medicine of a kind of energy long-term control muscle skeleton and ICT, the existing disease progression of inhibition and prophylaxis of acute symptomatic recurrence has the important medical meaning for millions upon millions of patients that suffer from described disease.
Summary of the invention
In one embodiment, the present invention relates to a kind of method for the treatment of muscle skeleton and ICT.Described inflammation comprises osteoarthritis and joint and the periarthritis disease relevant with osteoarthritis, and nonarticular rheumatism, and described nonarticular rheumatism comprises capsulitis, tendinitis, fibrositis and periarthritis disease.Described method comprises that the compositions that contains the 13-cis-retinoic acid with effective therapeutic dose is applied to the patient.Described compositions also contains pharmaceutical carrier, and can powder, the form of pill, capsule, tablet and liquid exists.Under the preferred situation, the method for described treatment muscle skeleton and ICT comprises the steps: to use described compositions preliminary dosage, that contain the 13-cis-retinoic acid in the preliminary treatment phase to the patient; Subsequently, to the patient use maintenance dose contain the 13-cis-retinoic acid described compositions, described muscle skeleton comprises osteoarthritis and joint and the periarthritis disease relevant with osteoarthritis with ICT, and nonarticular rheumatism, described nonarticular rheumatism comprises capsulitis, tendinitis, fibrositis and periarthritis disease.
In another embodiment, the present invention relates to a kind of osteoarthritis for the treatment of and reach the joint relevant with osteoarthritis and the combined method of periarthritis disease and nonarticular rheumatism, described nonarticular rheumatism comprises capsulitis, tendinitis, fibrositis and periarthritis disease.Described combination therapy has adopted the traditional method of treatment muscle skeleton and ICT, and uses compositions effective therapeutic dose, that contain the 13-cis-retinoic acid to the patient.
So, the purpose of this invention is to provide treatment muscle skeleton and ICT and a kind of medicine of associated symptom.
By hereinafter the statement the specific embodiment and additional claim as can be known, the above and other objects and advantages of the present invention are conspicuous.
The specific embodiment
In one embodiment, the present invention relates to a kind of method for the treatment of muscle skeleton and ICT.The muscle skeleton that is suitable for comprises osteoarthritis and joint and the periarthritis disease relevant with osteoarthritis without limitation with the ICT type, and the nonarticular rheumatism that comprises capsulitis, tendinitis, fibrositis and periarthritis disease.Described method comprises to the patient uses a kind of compositions effective therapeutic dose, that contain the 13-cis-retinoic acid.The scope of described effective therapeutic dose is daily to take in about 80 milligrams of the about 10-of 13-cis-retinoic acid (about 1.1 milligrams of the about 0.14-of every kg body weight).
Described compositions also contains pharmaceutical carrier.Common pharmaceutical carrier comprises liquid carrier, as the analog of oral liquids such as water, ethylene glycol, oil, ethanol, syrup and suspension, syrup, elixir and solution; Solid carrier is as analog such as starch, saccharide, Kaolin, lubricant, binding agent, disintegrating agent and powder, pill, capsule and tablets; Other pharmaceutical carriers well known in the art.The compositions that is used for purpose of the present invention can exist with various form, as powder, pill, capsule, tablet and medicinal liquid etc.Although because of its convenience preferred oral preparation, be to use other suitable general administering modes also to can be used for purpose of the present invention.
The 13-cis-retinoic acid is a kind of commercial medicine, and its trade mark is Accutane , produce by the sharp Hoffmann-La Roche of New Jersey nanotesla company, be used for the treatment of some dermatosis.Accutane Three kinds of available dosage forms are arranged, the Perle of promptly 10 milligrams, 20 milligrams and 40 milligrams.
Preferred Therapeutic Method comprises two treatment phases: tentatively treat the phase and keep the treatment phase.At first, in preliminary treatment, the patient takes the 13-cis-retinoic acid of preliminary dosage, about 10 days to about 5 months its medicine time.Subsequently, this patient takes the 13-cis-retinoic acid of lower maintenance dose.
The preferred preliminary treatment phase is about 2-3 week because as surpass 2-3 week, some side effect of this medicine, as tenderness, xerosis cutis, the lip of fiber-muscle-old injury of skeleton system chap, eyes are dry and astringent and nose drying etc. will take place.If tentatively these side effect appear in the treatment phase, then after beginning to take maintenance dose, described side effect can weaken usually.If but side effect does not appear in the patient, then can prolong the preliminary treatment phase, to strengthen the effect of this medicine treatment muscle skeleton and ICT.But in 20 weeks of continuous administration when the 13-cis-retinoic acid is used for the treatment of the patient who suffers from serious acne at present, based on this, according to the individual patients reaction and the state of an illness, the preliminary treatment phase of the present invention can be longer than several weeks basically.
Low keep dosage two functions are arranged.At first, after the preliminary treatment, the treatment of using maintenance dose needs several time-of-weeks to control existing muscle skeleton and ICT, and the existing inflammation disease of inhibition further develops deterioration.The second, the long term maintenance dosed administration can prevent the recurrence of muscle skeleton and ICT, and described inflammation is clinically often with various chronic muscle skeletons and ICT.Under the therefore preferred situation, answer the chronic administration maintenance dose.
Dosage should be decided according to patient's body weight.Preliminary dosage is the 13-cis-retinoic acid (about 1.1 milligrams of the about 0.14-of every kg body weight) of about 10-80 milligram every day.For body weight is the ordinary people of 160 pounds (72.6 kilograms) approximately, and average preliminary dosage is about 40 milligrams of every day.Maintenance dose was to take the about 10-80 milligram of 13-cis-retinoic acid (about 1.1 milligrams of the about 0.14-of every kg body weight) every 3-7 days.For body weight approximately is 160 pounds ordinary people, average maintenance dose be every 3-7 days about 40 milligrams.Be starkly lower than or be higher than the people of average weight for child or body weight, should correspondingly adjust its dosage.
Patient's dosage every day can be taken disposable or in batches.Because Accutane The i.e. Perle of 10 milligrams, 20 milligrams and 40 milligrams of three kinds of commercial dosage forms is arranged, so, take one 40 milligrams capsule every day but preliminary dosage is 40 milligrams patient, or take two 20 milligrams capsule every day, or take 4 10 milligrams capsule every day.The dosage of keeping treatment is the same.For simplicity, during keeping treatment, the patient took 40 milligrams dosage in every approximately 3-7 days one time.
Have now found that, use method of the present invention to treat after, the state of an illness that the patient who suffers from muscle skeleton and ICT after diagnosing obtains is in various degree improved.Visible improvement comprises and having alleviated because of for example muscle skeleton of affected body parts such as cervical vertebra, shoulder, hands, buttocks and neck and pain and the tenderness that ICT causes; Alleviate arthroncus; Eliminate the other fibrocalcific tuberosity of cervical vertebra vertebra; Alleviate ankylosis and enlarge range of activity; Recover physical ability.In addition, use above-mentioned Therapeutic Method, do not observe serious adverse.
Clinical effectiveness based on this medicine, think now, the 13-cis-retinoic acid can be controlled muscle skeleton and ICT, eliminate and reinvent joint and the periarticular pathological changes that causes by described disease, comprising: it is plump and eliminate the bone fibres cartilage lesion of peripheral region, joint to decompose ligament and joint capsule, and reinvents the pathological changes that described disease causes and make it to be tending towards more normal structure.The detailed mechanism of 13-cis-retinoic acid treatment muscle skeleton and ICT still belongs to unknown at present.
Importantly, have been found that now by secular hanging down and keep dosed administration, the 13-cis-retinoic acid can provide the long-term control to muscle skeleton and ICT, suppress existing inflammation disease and further worsen, and prevent the acute relapse of described chronic muscle skeleton and ICT.Consider that the number of suffering from this type of common chronic disease is more, and the forfeiture of health natural functions can occur lack effectively long-term prevention of described disease and control, so the present invention to have the important medical meaning with PD in addition.
In another embodiment, method of the present invention can be used as the ancillary method of other traditional therapies that are used for the treatment of muscle skeleton and ICT.Described traditional method comprises cortisone injection, surgical operation therapy, uses nonsteroidal anti-inflammatory agent and physiotherapy to general.Using of the 13-cis-retinoic acid of effective dose can be used for auxiliary other traditional remedies, and can be used for improving overall therapeutic effect.Using the 13-cis-retinoic acid can carry out simultaneously with traditional remedies, for example carries out with cortisone or hyaluronic acid injection; Use with conventional medicaments such as nonsteroidal anti-inflammatory agent, chondroitin sulfate and glycosamines; Or carry out with physiotherapy.13-cis-retinoic acid therapy of the present invention also can be carried out before operation or after the operation.
Embodiment 1 to embodiment 3 for example understands the clinical effectiveness of above-mentioned Therapeutic Method.Write out a prescription to the patient and to carry out preliminary treatment recited above and to keep treatment.It should be noted that the weight in patients described in the example all in the average weight scope, therefore, has adopted 40 milligrams mean dose.Should also be noted that because take Accutane Can cause photosensitivity, so, enjoined all patients to avoid sun exposure fully in the preliminary treatment phase with in last or two weeks after keeping the treatment beginning.
Embodiment 1:
1988, white race male patient's joint disease outbreak that 62 years old, health are roughly healthy, its affected part only is a hand.Main site of pathological change is once in the tip interphalangeal joint (IP joint) of fracture in 1980.Symptom has edema and swelling, with the tenderness of aggravation year by year.This tenderness is more and more obvious, to such an extent as in 1994, this patient can not wave because of pain.In addition, because finger swelling and tightening, the carrying out property obstacle of clenching fist appears in the patient.
X-ray examination finds that articular cavity attenuates and the interphalangeal joint capsular swelling.The lab testing result is normal.The patient is suffered from osteoarthritis companion tendinitis by diagnosis.
Atomic or absolutely void at several treatment measure effects that this patient adopts, these treatment measures comprise aspirin (every day 2-5 grain 325 milligrams pill); Motrin TM(ibuprofen) and Naprosyn TM(naproxen); And glycosamine/chondroitin sulfate.
In April, 1997, because of another disease, this patient begins to take Accutane (13-cis-retinoic acid, Hoffmann-La Roche company, nanotesla profit, New Jersey), preliminary dosage is about 40 milligrams Accutane every day , continue 21 days, then a week 2 times (Monday and Fridays) is taken about 40 milligrams maintenance dose.In some months subsequently, the patient notices that its hand state of an illness obtains progressively, stable improvement, and the stiff and pain of the shoulder that is caused by the right side old wound of shoulder rotator cuff also is improved.In addition, the patient is also noted that its cervical vertebra touches a tender spot and also slowly improve (be subjected to serious whiplash in the nineteen sixty-eight traffic accident after, its cervical vertebra touch a tender spot last very long), and with the expansion and the other fibrocalcific nodular elimination of cervical vertebra vertebra of range of activity (ROM).
Because patient's osteoarthritis and tendinitis are able to obvious improvement, the patient continues the Accutane of above-mentioned maintenance dose Treatment so far.Except occurring side effect such as lip, chapped skin in early days, other health side effect do not appear.In the preliminary treatment phase, notice the right shoulder pain that principal characteristic once occurs adding, but disappeared afterwards.Blood samples of patients is biochemical and the hematological examination result is normal always.
This patient's whole health is improved greatly, and the weak disease of any never again muscle skeleton occurs.
Embodiment 2:
69 years old, the retired warrant officer of naval, white race male old man are suffered from struvite osteoarthritis and rheumatism by diagnosis.Its symptom comprises the arthralgia that continues 6-10.In 1992, the right buttocks of arthralgia invasion and attack patient was subjected to the torment of pain of buttock deeply when the patient works at first.1994, cervical region and left shoulder pain progressively appearred in the patient.The X-ray examination result shows the cervical vertebra calcification.In addition, patient's shoulder is suffered from the rotator cuff wound by diagnosis.1997, touching a tender spot appearred in patient's hand when playing golf.After this patient's hand state of an illness further worsens, and the floating bloated and difficulty of clenching fist of finger occurs.But patient's blood biochemical is normal.
The patient adopted aspirin and Motrin in the past TMTreatment, but have little effect.And have only of short duration effect with glycosamine/chondroitin sulfate extract for treating.Naturopathy just part has been alleviated the hand state of an illness.Because the hand swing and the difficulty of clenching fist, the patient worry can not such as own institute hopes often be engaged in golf sports, even be forced to consideration and abandon this motion.
This patient adopts the treatment of 13-cis-retinoic acid on May 1st, 2002, and preliminary dosage is about 40 milligrams of Accutane every day , continue 14 days, then week 2 times is used about 40 milligrams maintenance dose to the patient.After the treatment through 7 weeks altogether, patient's shoulder pain complete obiteration (annotate: in the 13-cis-retinoic acid treatment phase, the patient continues naturopathy is carried out in this zone), it is normal that range of activity is recovered, cervical region and pain of buttock almost completely disappear (ending in August, 2002).Under situation about playing golf continuously 3-4 days, patient's hand still has slight tenderness.But the floating the symptom bloated and difficulty of clenching fist of hand has disappeared.Because health is significantly improved, patient's golf obstacle rank drops to 9 by 11.
After the patient takes the 13-cis-retinoic acid, have only slight side reaction, what comprise former of dry and some left shoulders of skin, lip adds principal characteristic pain, and these side reactions had disappeared afterwards.
Embodiment 3:
A white race male peasant of 61 years old has the pain in hand history that relates to finger in more than 10 year, with interphalangeal joint swelling and tenderness.The hand illness makes its work and the difficulty that plays golf.He is suffered from osteoarthritis by diagnosis.
This patient begins to carry out the treatment of 13-cis-retinoic acid April calendar year 2001, preliminary dosage about 400 milligrams of Accutane every day , continuing 21 days, week 2 times is used about 40 milligrams maintenance dose to the patient subsequently.After treating for 10 weeks, patient's symptom begins to improve, and comprises the expansion with range of activity of alleviating of finger swelling and tenderness symptom.Follow-up 6 the middle of the month continuous administration maintenance dose, its doing well,improving is kept.
Patient's hematological results is all normal before and after treatment.Except skin and lip drying, the patient does not have other side reaction.These side reactions have disappeared behind the picked-up maintenance dose.
Though shown and described the preferred embodiments of the invention, should be understood that except the concrete embodiment that shows and describe herein, the present invention can also adopt other modes to implement here.And, in described embodiment, without prejudice to as the prerequisite of the basic thought of following additional claims of the present invention and principle under, can and arrange to do some change to the form of each several part.

Claims (10)

1. the compositions that comprises the 13-cis-retinoic acid is used for the treatment of purposes in the medicine of muscle skeleton and ICT in preparation.
2. purposes as claimed in claim 1, wherein said compositions also contains a kind of pharmaceutical carrier.
3. purposes as claimed in claim 2, the existence form of wherein said compositions is selected from the group of being made up of powder, pill, capsule, tablet and liquid.
4. purposes as claimed in claim 1, wherein said muscle skeleton comprises osteoarthritis and relevant arthritis and periarthritis disease with ICT, and nonarticular rheumatism, wherein said nonarticular rheumatism comprises capsulitis, tendinitis, fibrositis and periarthritis disease.
5. purposes as claimed in claim 1, wherein the treatment to described muscle skeleton and ICT comprises the preliminary treatment phase and keeps the treatment phase.
6. purposes as claimed in claim 5, wherein the preliminary dosage in the preliminary treatment phase is that per kg body weight per day is used about 0.14 milligram-Yue 1.1 milligrams of 13-cis-retinoic acids.
7. purposes as claimed in claim 5, the wherein said preliminary treatment phase is about 10 days to 5 months.
8. purposes as claimed in claim 5, wherein said compositions are that every 3-7 days every kg body weight are used about 0.14 milligram-Yue 1.1 milligrams of 13-cis-retinoic acids at the maintenance dose of keeping the treatment phase.
9. purposes as claimed in claim 1, wherein said treatment comprise with the traditional therapy of treatment muscle skeleton and ICT and are used in combination the compositions that comprises the 13-cis-retinoic acid.
10. purposes as claimed in claim 9, wherein said traditional therapy comprise cortisone injection, hyaluronic acid injection, surgical operation therapy, use nonsteroidal anti-inflammatory agent and physiotherapy to general.
CNA2003101017637A 2002-10-23 2003-10-23 Method for treating inflammation of muscular skeleton and connective tissue Pending CN1496737A (en)

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Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN116546982A (en) * 2020-05-24 2023-08-04 李兆阳 Retinoic acid compositions and methods thereof

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN116546982A (en) * 2020-05-24 2023-08-04 李兆阳 Retinoic acid compositions and methods thereof

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