CN118974026A - 莱特莫韦中间体及其制备方法 - Google Patents
莱特莫韦中间体及其制备方法 Download PDFInfo
- Publication number
- CN118974026A CN118974026A CN202380024475.1A CN202380024475A CN118974026A CN 118974026 A CN118974026 A CN 118974026A CN 202380024475 A CN202380024475 A CN 202380024475A CN 118974026 A CN118974026 A CN 118974026A
- Authority
- CN
- China
- Prior art keywords
- methoxyphenyl
- trifluoromethyl
- fluoro
- methoxy
- phenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/78—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
- C07D239/84—Nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN202210371221 | 2022-04-01 | ||
| CN2022103712214 | 2022-04-01 | ||
| PCT/CN2023/083173 WO2023185597A1 (fr) | 2022-04-01 | 2023-03-22 | Intermédiaire de letermovir et son procédé de préparation |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN118974026A true CN118974026A (zh) | 2024-11-15 |
Family
ID=88199228
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN202380024475.1A Pending CN118974026A (zh) | 2022-04-01 | 2023-03-22 | 莱特莫韦中间体及其制备方法 |
Country Status (2)
| Country | Link |
|---|---|
| CN (1) | CN118974026A (fr) |
| WO (1) | WO2023185597A1 (fr) |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10319612A1 (de) * | 2003-05-02 | 2004-11-18 | Bayer Healthcare Ag | Substituierte Dihydrochinazoline |
| DE102005027517A1 (de) * | 2005-06-15 | 2006-12-21 | Bayer Healthcare Ag | Verfahren zur Herstellung von Dihydrochinazolinen |
| WO2015088931A1 (fr) * | 2013-12-12 | 2015-06-18 | Merck Sharp & Dohme Corp. | Procédé de préparation de composés quinazoline substitués |
| WO2017091453A1 (fr) * | 2015-11-24 | 2017-06-01 | Merck Sharp & Dohme Corp. | Nouveaux procédés de production de composés de quinazoline substitués à l'aide de catalyseurs de liaison hydrogène |
| IT202000017617A1 (it) * | 2020-07-21 | 2022-01-21 | Olon Spa | Procedimento per la preparazione di un intermedio utilizzato nella sintesi del letermovir |
-
2023
- 2023-03-22 CN CN202380024475.1A patent/CN118974026A/zh active Pending
- 2023-03-22 WO PCT/CN2023/083173 patent/WO2023185597A1/fr not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO2023185597A1 (fr) | 2023-10-05 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PB01 | Publication | ||
| PB01 | Publication | ||
| SE01 | Entry into force of request for substantive examination | ||
| SE01 | Entry into force of request for substantive examination |