CN115701997A - Btk抑制剂治疗疾病的用途 - Google Patents
Btk抑制剂治疗疾病的用途 Download PDFInfo
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- CN115701997A CN115701997A CN202180043292.5A CN202180043292A CN115701997A CN 115701997 A CN115701997 A CN 115701997A CN 202180043292 A CN202180043292 A CN 202180043292A CN 115701997 A CN115701997 A CN 115701997A
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- btk inhibitor
- neuromyelitis optica
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Abstract
公开了BTK抑制剂治疗疾病的用途。具体公开了BTK抑制剂在制备预防或治疗视神经脊髓炎谱系疾病的药物中的用途。
Description
PCT国内申请，说明书已公开。
Claims (10)
- PCT国内申请，权利要求书已公开。
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN2020107964821 | 2020-08-10 | ||
| CN202010796482 | 2020-08-10 | ||
| CN202110295378 | 2021-03-19 | ||
| CN2021102953789 | 2021-03-19 | ||
| PCT/CN2021/111726 WO2022033460A1 (zh) | 2020-08-10 | 2021-08-10 | Btk抑制剂治疗疾病的用途 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN115701997A true CN115701997A (zh) | 2023-02-14 |
| CN115701997B CN115701997B (zh) | 2024-09-13 |
Family
ID=80246908
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN202180043292.5A Active CN115701997B (zh) | 2020-08-10 | 2021-08-10 | Btk抑制剂治疗疾病的用途 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20230270743A1 (zh) |
| EP (1) | EP4193995A4 (zh) |
| JP (1) | JP2023536944A (zh) |
| KR (1) | KR20230050363A (zh) |
| CN (1) | CN115701997B (zh) |
| CA (1) | CA3188003A1 (zh) |
| TW (1) | TW202214250A (zh) |
| WO (1) | WO2022033460A1 (zh) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2024192765A1 (en) * | 2023-03-23 | 2024-09-26 | Brown University | First in class use of the crth2 antagonist in treating neuromyelitis optica spectrum disorder (nmosd) and relevant autoimmune cns disorders |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW202408524A (zh) * | 2022-05-10 | 2024-03-01 | 大陸商瑞石生物醫藥有限公司 | Ｂｔｋ抑制劑用於治療疾病的用途 |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN106573001A (zh) * | 2014-07-07 | 2017-04-19 | 永恒生物科技公司 | 作为蛋白激酶抑制剂的氨基哒嗪酮化合物 |
| WO2017118277A1 (zh) * | 2016-01-05 | 2017-07-13 | 江苏恒瑞医药股份有限公司 | 一种btk激酶抑制剂的结晶形式及其制备方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20240070721A (ko) * | 2015-06-03 | 2024-05-21 | 프린시피아 바이오파마, 인코퍼레이티드 | 티로신 키나제 억제제 |
| WO2018005849A1 (en) * | 2016-06-29 | 2018-01-04 | Principia Biopharma Inc. | Modified release formulations of 2-[3-[4-amino-3-(2-fluoro-4-phenoxy-phenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl]-4-methyl-4-[4-(oxetan-3-yl)piperazin-1-yl]pent-2-enenitrile |
| WO2019126759A1 (en) * | 2017-12-22 | 2019-06-27 | Convelo Therapeutics, Inc. | Compounds and methods of promoting myelination |
| CN110772521A (zh) * | 2018-07-31 | 2020-02-11 | 苏州亚盛药业有限公司 | Bcl-2抑制剂或Bcl-2/Bcl-xL抑制剂与BTK抑制剂的组合产品及其用途 |
| CN111499642A (zh) * | 2019-01-31 | 2020-08-07 | 江苏恒瑞医药股份有限公司 | 吡咯并[2,3-d]哒嗪-7-酮类衍生物的可药用盐、晶型及其制备方法 |
-
2021
- 2021-08-10 KR KR1020237007341A patent/KR20230050363A/ko active Pending
- 2021-08-10 JP JP2023507702A patent/JP2023536944A/ja not_active Withdrawn
- 2021-08-10 CA CA3188003A patent/CA3188003A1/en active Pending
- 2021-08-10 US US18/019,465 patent/US20230270743A1/en active Pending
- 2021-08-10 TW TW110129478A patent/TW202214250A/zh unknown
- 2021-08-10 WO PCT/CN2021/111726 patent/WO2022033460A1/zh not_active Ceased
- 2021-08-10 EP EP21855512.6A patent/EP4193995A4/en active Pending
- 2021-08-10 CN CN202180043292.5A patent/CN115701997B/zh active Active
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN106573001A (zh) * | 2014-07-07 | 2017-04-19 | 永恒生物科技公司 | 作为蛋白激酶抑制剂的氨基哒嗪酮化合物 |
| WO2017118277A1 (zh) * | 2016-01-05 | 2017-07-13 | 江苏恒瑞医药股份有限公司 | 一种btk激酶抑制剂的结晶形式及其制备方法 |
Non-Patent Citations (1)
| Title |
|---|
| 王炜: "Btk/NF-κB信号通路及相关细胞因子在视神经脊髓炎谱系疾病中作用机制探", 《中国优秀博硕士学位论文全文数据库（硕士）医药卫生科技辑》, no. 1, pages 1 - 2 * |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2024192765A1 (en) * | 2023-03-23 | 2024-09-26 | Brown University | First in class use of the crth2 antagonist in treating neuromyelitis optica spectrum disorder (nmosd) and relevant autoimmune cns disorders |
Also Published As
| Publication number | Publication date |
|---|---|
| KR20230050363A (ko) | 2023-04-14 |
| WO2022033460A1 (zh) | 2022-02-17 |
| EP4193995A1 (en) | 2023-06-14 |
| TW202214250A (zh) | 2022-04-16 |
| US20230270743A1 (en) | 2023-08-31 |
| CA3188003A1 (en) | 2022-02-17 |
| JP2023536944A (ja) | 2023-08-30 |
| EP4193995A4 (en) | 2024-08-21 |
| CN115701997B (zh) | 2024-09-13 |
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