CL2021003032A1 - Métodos de tratamiento de la urticaria crónica espontánea utilizando un inhibidor de la tirosina quinasa de bruton - Google Patents
Métodos de tratamiento de la urticaria crónica espontánea utilizando un inhibidor de la tirosina quinasa de brutonInfo
- Publication number
- CL2021003032A1 CL2021003032A1 CL2021003032A CL2021003032A CL2021003032A1 CL 2021003032 A1 CL2021003032 A1 CL 2021003032A1 CL 2021003032 A CL2021003032 A CL 2021003032A CL 2021003032 A CL2021003032 A CL 2021003032A CL 2021003032 A1 CL2021003032 A1 CL 2021003032A1
- Authority
- CL
- Chile
- Prior art keywords
- methods
- bruton
- chronic spontaneous
- tyrosine kinase
- kinase inhibitor
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Epidemiology (AREA)
- Dermatology (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente divulgación se relaciona con métodos para el tratamiento de la Urticaria Crónica Espontánea utilizando un compuesto de Fórmula (I) o una sal farmacéuticamente aceptable del mismo. En la presente también se divulga un compuesto de Fórmula (I) o una sal farmacéuticamente aceptable del mismo, para el tratamiento de pacientes con Urticaria Crónica Espontánea, así como también medicamentos, regímenes de dosificación, formulaciones farmacéuticas, formas de dosificación, y kits para utilizar en los usos y métodos divulgados.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962851996P | 2019-05-23 | 2019-05-23 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CL2021003032A1 true CL2021003032A1 (es) | 2022-09-09 |
Family
ID=70918751
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CL2021003032A CL2021003032A1 (es) | 2019-05-23 | 2021-11-17 | Métodos de tratamiento de la urticaria crónica espontánea utilizando un inhibidor de la tirosina quinasa de bruton |
Country Status (22)
| Country | Link |
|---|---|
| US (2) | US12419889B2 (es) |
| EP (2) | EP3972604B1 (es) |
| JP (2) | JP7568651B2 (es) |
| KR (1) | KR20220012281A (es) |
| CN (1) | CN113795255A (es) |
| AU (2) | AU2020280272B2 (es) |
| BR (1) | BR112021022602A2 (es) |
| CA (1) | CA3138081A1 (es) |
| CL (1) | CL2021003032A1 (es) |
| DK (1) | DK3972604T3 (es) |
| ES (1) | ES3039974T3 (es) |
| FI (1) | FI3972604T3 (es) |
| HR (1) | HRP20251001T1 (es) |
| IL (1) | IL286983B1 (es) |
| LT (1) | LT3972604T (es) |
| MX (2) | MX2021013942A (es) |
| PL (1) | PL3972604T3 (es) |
| PT (1) | PT3972604T (es) |
| RS (1) | RS67141B1 (es) |
| SI (1) | SI3972604T1 (es) |
| TW (1) | TWI868139B (es) |
| WO (1) | WO2020234782A1 (es) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2020234782A1 (en) | 2019-05-23 | 2020-11-26 | Novartis Ag | Methods of treating chronic spontaneous urticaria using a bruton's tyrosine kinase inhibitor |
| AU2022337087A1 (en) | 2021-09-03 | 2024-03-14 | Novartis Ag | Lou064 for treating multiple sclerosis |
| EP4448114A1 (en) | 2021-12-14 | 2024-10-23 | Novartis AG | Methods of treatment using lou064 |
| TW202342048A (zh) | 2022-02-28 | 2023-11-01 | 瑞士商諾華公司 | 使用lou064治療化膿性汗腺炎之方法 |
| KR102834740B1 (ko) * | 2023-04-10 | 2025-07-17 | 아주대학교산학협력단 | Hsp10 또는 이의 항체를 유효성분으로 포함하는 만성 자발적 두드러기의 진단을 위한 바이오마커 조성물 |
| WO2024235163A1 (zh) * | 2023-05-12 | 2024-11-21 | 武汉人福创新药物研发中心有限公司 | Btk抑制剂的用途和单剂量药物 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5439377B2 (ja) | 2007-09-14 | 2014-03-12 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | ヒスタミンh4受容体のチエノ−及びフロ−ピリミジン調節物質 |
| US9512084B2 (en) * | 2013-11-29 | 2016-12-06 | Novartis Ag | Amino pyrimidine derivatives |
| WO2015105926A1 (en) | 2014-01-08 | 2015-07-16 | Moderna Therapeutics, Inc. | Polynucleotides for the in vivo production of antibodies |
| WO2016079669A1 (en) * | 2014-11-19 | 2016-05-26 | Novartis Ag | Labeled amino pyrimidine derivatives |
| WO2020234782A1 (en) | 2019-05-23 | 2020-11-26 | Novartis Ag | Methods of treating chronic spontaneous urticaria using a bruton's tyrosine kinase inhibitor |
-
2020
- 2020-05-20 WO PCT/IB2020/054755 patent/WO2020234782A1/en not_active Ceased
- 2020-05-20 DK DK20729204.6T patent/DK3972604T3/da active
- 2020-05-20 SI SI202030651T patent/SI3972604T1/sl unknown
- 2020-05-20 PT PT207292046T patent/PT3972604T/pt unknown
- 2020-05-20 BR BR112021022602A patent/BR112021022602A2/pt unknown
- 2020-05-20 LT LTEPPCT/IB2020/054755T patent/LT3972604T/lt unknown
- 2020-05-20 CA CA3138081A patent/CA3138081A1/en active Pending
- 2020-05-20 US US17/612,778 patent/US12419889B2/en active Active
- 2020-05-20 HR HRP20251001TT patent/HRP20251001T1/hr unknown
- 2020-05-20 EP EP20729204.6A patent/EP3972604B1/en active Active
- 2020-05-20 AU AU2020280272A patent/AU2020280272B2/en active Active
- 2020-05-20 ES ES20729204T patent/ES3039974T3/es active Active
- 2020-05-20 FI FIEP20729204.6T patent/FI3972604T3/fi active
- 2020-05-20 KR KR1020217041089A patent/KR20220012281A/ko active Pending
- 2020-05-20 PL PL20729204.6T patent/PL3972604T3/pl unknown
- 2020-05-20 RS RS20250816A patent/RS67141B1/sr unknown
- 2020-05-20 CN CN202080032000.3A patent/CN113795255A/zh active Pending
- 2020-05-20 EP EP25178785.9A patent/EP4599894A3/en active Pending
- 2020-05-20 JP JP2021568760A patent/JP7568651B2/ja active Active
- 2020-05-20 MX MX2021013942A patent/MX2021013942A/es unknown
- 2020-05-20 IL IL286983A patent/IL286983B1/en unknown
- 2020-05-21 TW TW109116854A patent/TWI868139B/zh active
-
2021
- 2021-11-12 MX MX2024014626A patent/MX2024014626A/es unknown
- 2021-11-17 CL CL2021003032A patent/CL2021003032A1/es unknown
-
2024
- 2024-08-21 JP JP2024139784A patent/JP2024178168A/ja active Pending
-
2025
- 2025-08-27 US US19/311,292 patent/US20250375446A1/en active Pending
- 2025-10-17 AU AU2025252618A patent/AU2025252618A1/en active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| BR112021022602A2 (pt) | 2022-01-04 |
| HRP20251001T1 (hr) | 2025-10-24 |
| JP2024178168A (ja) | 2024-12-24 |
| FI3972604T3 (fi) | 2025-09-01 |
| AU2020280272A1 (en) | 2021-11-18 |
| AU2025252618A1 (en) | 2025-11-06 |
| WO2020234782A1 (en) | 2020-11-26 |
| EP3972604B1 (en) | 2025-06-04 |
| KR20220012281A (ko) | 2022-02-03 |
| US20250375446A1 (en) | 2025-12-11 |
| LT3972604T (lt) | 2025-09-10 |
| IL286983B1 (en) | 2025-09-01 |
| DK3972604T3 (da) | 2025-09-15 |
| RS67141B1 (sr) | 2025-09-30 |
| PL3972604T3 (pl) | 2025-09-22 |
| AU2020280272B2 (en) | 2025-07-24 |
| CA3138081A1 (en) | 2020-11-26 |
| IL286983A (en) | 2021-12-01 |
| JP7568651B2 (ja) | 2024-10-16 |
| ES3039974T3 (en) | 2025-10-28 |
| SI3972604T1 (sl) | 2025-09-30 |
| CN113795255A (zh) | 2021-12-14 |
| TWI868139B (zh) | 2025-01-01 |
| TW202110450A (zh) | 2021-03-16 |
| MX2021013942A (es) | 2022-01-04 |
| JP2022533981A (ja) | 2022-07-27 |
| US12419889B2 (en) | 2025-09-23 |
| EP3972604A1 (en) | 2022-03-30 |
| EP4599894A2 (en) | 2025-08-13 |
| MX2024014626A (es) | 2025-01-09 |
| US20220184074A1 (en) | 2022-06-16 |
| PT3972604T (pt) | 2025-08-26 |
| EP4599894A3 (en) | 2025-11-12 |
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