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CL2017002299A1 - Combinaciones de dosis fija y formulaciones comprendiendo etc-1002 y ezetimiba y métodos para tratar o reducir el riesgo de enfermedades cardiovasculares - Google Patents

Combinaciones de dosis fija y formulaciones comprendiendo etc-1002 y ezetimiba y métodos para tratar o reducir el riesgo de enfermedades cardiovasculares

Info

Publication number
CL2017002299A1
CL2017002299A1 CL2017002299A CL2017002299A CL2017002299A1 CL 2017002299 A1 CL2017002299 A1 CL 2017002299A1 CL 2017002299 A CL2017002299 A CL 2017002299A CL 2017002299 A CL2017002299 A CL 2017002299A CL 2017002299 A1 CL2017002299 A1 CL 2017002299A1
Authority
CL
Chile
Prior art keywords
ezetimibe
treat
methods
cardiovascular diseases
risk
Prior art date
Application number
CL2017002299A
Other languages
English (en)
Inventor
Roger Schofield Newton
Noah Laban Rosenberg
Diane Elaine Macdougall
Original Assignee
Esperion Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=56920255&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2017002299(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Esperion Therapeutics Inc filed Critical Esperion Therapeutics Inc
Publication of CL2017002299A1 publication Critical patent/CL2017002299A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/20Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/194Carboxylic acids, e.g. valproic acid having two or more carboxyl groups, e.g. succinic, maleic or phthalic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

<p>Se divulga aquí composiciones comprendiendo dosis fijas de ETC-1002 y Ezetimiba. También se divulga aquí métodos para usar dosis fijas de ETC-1002 y Ezetimiba. Los usos incluyen métodos para tratar enfermedades cardiovasculares o reducir el riesgo de enfermedades cardiovasculares en un sujeto. Los usos también incluyen métodos para tratar la hipercolesterolemia en un sujeto.</p>
CL2017002299A 2015-03-13 2017-09-12 Combinaciones de dosis fija y formulaciones comprendiendo etc-1002 y ezetimiba y métodos para tratar o reducir el riesgo de enfermedades cardiovasculares CL2017002299A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201562133128P 2015-03-13 2015-03-13
US201562250921P 2015-11-04 2015-11-04

Publications (1)

Publication Number Publication Date
CL2017002299A1 true CL2017002299A1 (es) 2018-03-16

Family

ID=56920255

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2017002299A CL2017002299A1 (es) 2015-03-13 2017-09-12 Combinaciones de dosis fija y formulaciones comprendiendo etc-1002 y ezetimiba y métodos para tratar o reducir el riesgo de enfermedades cardiovasculares

Country Status (18)

Country Link
US (3) US10912751B2 (es)
EP (1) EP3267989A4 (es)
JP (2) JP6940411B2 (es)
KR (1) KR102370582B1 (es)
CN (2) CN107530307A (es)
AU (3) AU2016233485B2 (es)
BR (1) BR112017019358A2 (es)
CA (1) CA2978204A1 (es)
CL (1) CL2017002299A1 (es)
IL (1) IL254194A0 (es)
MA (1) MA42616A (es)
MX (2) MX392182B (es)
PH (1) PH12017501625A1 (es)
RU (2) RU2766085C2 (es)
SG (2) SG10201908500UA (es)
UA (1) UA123355C2 (es)
WO (1) WO2016149191A1 (es)
ZA (1) ZA201706919B (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102370582B1 (ko) 2015-03-13 2022-03-04 에스페리온 테라피유틱스 인코포레이티드 Etc1002 및 에제티미브를 포함하는 고정 용량 조합 및 제형 및 심혈관 질환의 치료 또는 이의 위험의 감소 방법
MA41793A (fr) 2015-03-16 2018-01-23 Esperion Therapeutics Inc Associations de doses fixes comprenant du etc1002 et une ou plusieurs statines permettant de traiter ou de réduire un risque cardiovasculaire
WO2018148417A1 (en) * 2017-02-08 2018-08-16 Esperion Therapeutics, Inc. Triplet combination formulations and methods of treating or reducing the risk of cardiovascular disease
US20180338922A1 (en) * 2017-05-26 2018-11-29 Esperion Therapeutics, Inc. Fixed dose formulations
WO2019179494A1 (zh) * 2018-03-23 2019-09-26 深圳市塔吉瑞生物医药有限公司 取代的十五烷二酸化合物及药物组合物及其用途
US20210322375A1 (en) * 2018-08-27 2021-10-21 Esperion Therapeutics, Inc. Combination drug formulations for treating patients with cardiovascular disease and associated conditions
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US20240226049A1 (en) * 2023-01-09 2024-07-11 Esperion Therapeutics, Inc. Methods of treatment using bempedoic acid

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Also Published As

Publication number Publication date
ZA201706919B (en) 2022-03-30
UA123355C2 (uk) 2021-03-24
CA2978204A1 (en) 2016-09-22
EP3267989A1 (en) 2018-01-17
US11744816B2 (en) 2023-09-05
KR20180006887A (ko) 2018-01-19
JP2021193105A (ja) 2021-12-23
NZ736344A (en) 2024-08-30
AU2016233485A1 (en) 2017-11-02
JP2018507901A (ja) 2018-03-22
RU2022102472A (ru) 2022-03-15
SG11201707497UA (en) 2017-10-30
US10912751B2 (en) 2021-02-09
MX2017011499A (es) 2018-03-26
CN114099496A (zh) 2022-03-01
US20240398746A1 (en) 2024-12-05
AU2016233485B2 (en) 2021-05-20
MX2022005469A (es) 2022-06-02
US20210361605A1 (en) 2021-11-25
RU2017136180A3 (es) 2019-09-19
EP3267989A4 (en) 2018-11-07
MA42616A (fr) 2021-05-19
JP7295179B2 (ja) 2023-06-20
US20180064671A1 (en) 2018-03-08
KR102370582B1 (ko) 2022-03-04
AU2024202106A1 (en) 2024-05-02
AU2021218120A1 (en) 2021-09-09
CN107530307A (zh) 2018-01-02
RU2766085C2 (ru) 2022-02-07
BR112017019358A2 (pt) 2018-05-08
JP6940411B2 (ja) 2021-09-29
SG10201908500UA (en) 2019-11-28
PH12017501625A1 (en) 2018-02-12
IL254194A0 (en) 2017-10-31
RU2017136180A (ru) 2019-04-15
MX392182B (es) 2025-03-21
WO2016149191A1 (en) 2016-09-22

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