CL2012000595A1 - Composición antihelmíntica granular con levamisol hci y uno o más antihelmínticos seleccionados imidazotiazoles,lactonas macrocíclicas y praziquantel,un agente humectante y,opcionalmente,un agente de suspensión;sistema de dosificación;método de preparación de una formulación de suministro líquido;y un método para formar una composición antíhelmíntica. - Google Patents
Composición antihelmíntica granular con levamisol hci y uno o más antihelmínticos seleccionados imidazotiazoles,lactonas macrocíclicas y praziquantel,un agente humectante y,opcionalmente,un agente de suspensión;sistema de dosificación;método de preparación de una formulación de suministro líquido;y un método para formar una composición antíhelmíntica.Info
- Publication number
- CL2012000595A1 CL2012000595A1 CL2012000595A CL2012000595A CL2012000595A1 CL 2012000595 A1 CL2012000595 A1 CL 2012000595A1 CL 2012000595 A CL2012000595 A CL 2012000595A CL 2012000595 A CL2012000595 A CL 2012000595A CL 2012000595 A1 CL2012000595 A1 CL 2012000595A1
- Authority
- CL
- Chile
- Prior art keywords
- anthelmintic composition
- imidazothiazoles
- praziquantel
- anthelmintics
- granular
- Prior art date
Links
- 230000000507 anthelmentic effect Effects 0.000 title 3
- 239000000203 mixture Substances 0.000 title 3
- 238000000034 method Methods 0.000 title 2
- FSVJFNAIGNNGKK-UHFFFAOYSA-N 2-[cyclohexyl(oxo)methyl]-3,6,7,11b-tetrahydro-1H-pyrazino[2,1-a]isoquinolin-4-one Chemical compound C1C(C2=CC=CC=C2CC2)N2C(=O)CN1C(=O)C1CCCCC1 FSVJFNAIGNNGKK-UHFFFAOYSA-N 0.000 title 1
- UMZCLZPXPCNKML-UHFFFAOYSA-N 2h-imidazo[4,5-d][1,3]thiazole Chemical class C1=NC2=NCSC2=N1 UMZCLZPXPCNKML-UHFFFAOYSA-N 0.000 title 1
- HLFSDGLLUJUHTE-SNVBAGLBSA-N Levamisole Chemical compound C1([C@H]2CN3CCSC3=N2)=CC=CC=C1 HLFSDGLLUJUHTE-SNVBAGLBSA-N 0.000 title 1
- 229940124339 anthelmintic agent Drugs 0.000 title 1
- 239000000921 anthelmintic agent Substances 0.000 title 1
- 238000009472 formulation Methods 0.000 title 1
- 150000002596 lactones Chemical class 0.000 title 1
- 229960001614 levamisole Drugs 0.000 title 1
- 239000007788 liquid Substances 0.000 title 1
- 229960002957 praziquantel Drugs 0.000 title 1
- 239000000375 suspending agent Substances 0.000 title 1
- 239000000080 wetting agent Substances 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
- A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1611—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Inorganic Chemistry (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| NZ57954609 | 2009-09-07 | ||
| NZ57954509 | 2009-09-07 | ||
| NZ57954409 | 2009-09-07 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CL2012000595A1 true CL2012000595A1 (es) | 2012-12-14 |
Family
ID=43648938
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CL2012000595A CL2012000595A1 (es) | 2009-09-07 | 2012-03-06 | Composición antihelmíntica granular con levamisol hci y uno o más antihelmínticos seleccionados imidazotiazoles,lactonas macrocíclicas y praziquantel,un agente humectante y,opcionalmente,un agente de suspensión;sistema de dosificación;método de preparación de una formulación de suministro líquido;y un método para formar una composición antíhelmíntica. |
Country Status (10)
| Country | Link |
|---|---|
| US (2) | US11253593B2 (es) |
| EP (1) | EP2475430B1 (es) |
| AR (1) | AR079409A1 (es) |
| AU (8) | AU2010290829A1 (es) |
| BR (1) | BR112012005127B1 (es) |
| CA (2) | CA3040719C (es) |
| CL (1) | CL2012000595A1 (es) |
| ES (1) | ES2667026T3 (es) |
| WO (1) | WO2011027333A1 (es) |
| ZA (1) | ZA201207975B (es) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2482526A (en) * | 2010-08-05 | 2012-02-08 | Fiona Anne Macdonald | Praziquantel suspendable powder as an immersion fish treatment for parasites |
| NZ722695A (en) * | 2014-02-04 | 2021-12-24 | Argenta Innovation Ltd | Ectoparasite formulation |
| RU2669377C2 (ru) * | 2015-03-18 | 2018-10-11 | Федеральное государственное бюджетное научное учреждение Якутский научно-исследовательский институт сельского хозяйства | Способ комплексного лечения паразитарных болезней домашних северных оленей |
| KR102419769B1 (ko) | 2016-08-11 | 2022-07-13 | 아다미스 파마슈티칼스 코포레이션 | 약물 조성물 |
| NZ760663A (en) | 2017-06-26 | 2025-11-28 | Boehringer Ingelheim Animal Health Usa Inc | Dual active parasiticidal granule compositions, methods and uses thereof |
| EP3720844A4 (en) | 2017-12-08 | 2021-08-11 | Adamis Pharmaceuticals Corporation | MEDICINAL COMPOSITIONS |
| IT202000022126A1 (it) * | 2020-09-18 | 2022-03-18 | Nutrilinea S R L | Procedimento per preparare formulazioni solide comprendenti un composto idrofobico disperdibili in un liquido a freddo e relative formulazioni solide |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3626070A (en) * | 1968-03-20 | 1971-12-07 | Du Pont | Substituted 2-aminobenzimidazoles as anthelmintics |
| DE19654079A1 (de) * | 1996-12-23 | 1998-06-25 | Bayer Ag | Endo-ekto-parasitizide Mittel |
| AU772988B2 (en) * | 1999-06-04 | 2004-05-13 | Elanco Tiergesundheit Ag | Stable biocidal compositions |
| US20040151759A1 (en) * | 2002-08-16 | 2004-08-05 | Douglas Cleverly | Non-animal product containing veterinary formulations |
| NZ523128A (en) * | 2002-12-12 | 2006-01-27 | Ashmont Holdings Ltd | Anthelmintic formulations containing avermectins and or milbemycins |
| AU2003900505A0 (en) * | 2003-02-05 | 2003-02-20 | Jurox Pty Ltd | Anthelmintic composition |
| GB2403407B (en) * | 2003-07-03 | 2006-12-13 | Michael Hilary Burke | Palatable oral anthelmintic composition |
| WO2005016356A1 (en) * | 2003-08-08 | 2005-02-24 | The Hartz Mountain Corporation | Improved anthelmintic formulations |
| KR20070008686A (ko) * | 2004-04-07 | 2007-01-17 | 인터벳 인터내셔널 비.브이. | 벤지미다졸, 아버멕틴 및 프라지콴텔의 효능성 조성물 및이의 사용 방법 |
| NZ552040A (en) * | 2006-12-13 | 2009-04-30 | Bomac Research Ltd | Veterinary formulation comprising an anthelmintic compound and glyceryl acetate |
| PT2217241T (pt) * | 2007-11-07 | 2018-06-11 | Rigel Pharmaceuticals Inc | Granulação por via húmida utilizando um agente sequestrante de água |
| AU2008324095A1 (en) * | 2007-11-09 | 2009-05-14 | Intervet International B.V. | Anthelmintic combination |
| WO2011075592A1 (en) * | 2009-12-17 | 2011-06-23 | Merial Limited | Compositions comprising macrocyclic lactone compounds and spirodioxepinoindoles |
-
2010
- 2010-09-07 CA CA3040719A patent/CA3040719C/en active Active
- 2010-09-07 CA CA2777225A patent/CA2777225C/en active Active
- 2010-09-07 BR BR112012005127-0A patent/BR112012005127B1/pt active IP Right Grant
- 2010-09-07 ES ES10813424.8T patent/ES2667026T3/es active Active
- 2010-09-07 EP EP10813424.8A patent/EP2475430B1/en active Active
- 2010-09-07 AR ARP100103280A patent/AR079409A1/es not_active Application Discontinuation
- 2010-09-07 AU AU2010290829A patent/AU2010290829A1/en not_active Abandoned
- 2010-09-07 WO PCT/IB2010/054005 patent/WO2011027333A1/en not_active Ceased
-
2012
- 2012-03-06 CL CL2012000595A patent/CL2012000595A1/es unknown
- 2012-03-07 US US13/414,495 patent/US11253593B2/en active Active
- 2012-10-23 ZA ZA2012/07975A patent/ZA201207975B/en unknown
-
2016
- 2016-10-07 AU AU2016238922A patent/AU2016238922A1/en not_active Abandoned
-
2018
- 2018-09-05 AU AU2018226427A patent/AU2018226427A1/en not_active Abandoned
-
2020
- 2020-04-27 AU AU2020202781A patent/AU2020202781B2/en active Active
-
2021
- 2021-02-12 AU AU2021200921A patent/AU2021200921A1/en not_active Abandoned
- 2021-02-12 AU AU2021200922A patent/AU2021200922A1/en not_active Abandoned
-
2022
- 2022-01-07 US US17/571,084 patent/US20220125924A1/en not_active Abandoned
- 2022-01-11 AU AU2022200149A patent/AU2022200149B2/en active Active
- 2022-11-11 AU AU2022268388A patent/AU2022268388A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| AU2021200921A1 (en) | 2021-03-04 |
| AU2010290829A1 (en) | 2012-04-26 |
| CA2777225C (en) | 2019-06-11 |
| AU2016238922A1 (en) | 2016-12-15 |
| AR079409A1 (es) | 2012-01-25 |
| BR112012005127B1 (pt) | 2020-10-27 |
| ZA201207975B (en) | 2013-06-26 |
| US20220125924A1 (en) | 2022-04-28 |
| AU2022200149A1 (en) | 2022-02-10 |
| EP2475430A4 (en) | 2013-05-15 |
| US11253593B2 (en) | 2022-02-22 |
| AU2020202781A1 (en) | 2020-05-14 |
| CA2777225A1 (en) | 2011-03-10 |
| BR112012005127A2 (pt) | 2016-05-03 |
| AU2020202781B2 (en) | 2021-05-13 |
| AU2022200149B2 (en) | 2023-06-15 |
| CA3040719A1 (en) | 2011-03-10 |
| AU2021200922A1 (en) | 2021-03-04 |
| CA3040719C (en) | 2022-06-14 |
| ES2667026T3 (es) | 2018-05-09 |
| EP2475430B1 (en) | 2018-01-24 |
| EP2475430A1 (en) | 2012-07-18 |
| WO2011027333A1 (en) | 2011-03-10 |
| AU2018226427A1 (en) | 2018-09-27 |
| US20120238516A1 (en) | 2012-09-20 |
| AU2022268388A1 (en) | 2022-12-15 |
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