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CL2012000114A1 - Proceso para la preparacion de compuestos derivados de 5-amino-benzonorbornadieno donde se hacer reaccionar un compuesto de 5-halo-benzonorbornadieno con una bencilamina en prensecia de un catalizador de paladio. - Google Patents

Proceso para la preparacion de compuestos derivados de 5-amino-benzonorbornadieno donde se hacer reaccionar un compuesto de 5-halo-benzonorbornadieno con una bencilamina en prensecia de un catalizador de paladio.

Info

Publication number
CL2012000114A1
CL2012000114A1 CL2012000114A CL2012000114A CL2012000114A1 CL 2012000114 A1 CL2012000114 A1 CL 2012000114A1 CL 2012000114 A CL2012000114 A CL 2012000114A CL 2012000114 A CL2012000114 A CL 2012000114A CL 2012000114 A1 CL2012000114 A1 CL 2012000114A1
Authority
CL
Chile
Prior art keywords
benzonorbornadiene
benzylamine
halo
amino
preparation
Prior art date
Application number
CL2012000114A
Other languages
English (en)
Inventor
Hans Tobler
Harald Walter
Josef Ehrenfreund
Camilla Corsi
Fanny Giordano
Martin Zeller
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of CL2012000114A1 publication Critical patent/CL2012000114A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/62—Preparation of compounds containing amino groups bound to a carbon skeleton by cleaving carbon-to-nitrogen, sulfur-to-nitrogen, or phosphorus-to-nitrogen bonds, e.g. hydrolysis of amides, N-dealkylation of amines or quaternary ammonium compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/24—Preparation of compounds containing amino groups bound to a carbon skeleton by reductive alkylation of ammonia, amines or compounds having groups reducible to amino groups, with carbonyl compounds
    • C07C209/28—Preparation of compounds containing amino groups bound to a carbon skeleton by reductive alkylation of ammonia, amines or compounds having groups reducible to amino groups, with carbonyl compounds by reduction with other reducing agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/23—Preparation of halogenated hydrocarbons by dehalogenation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/26—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton
    • C07C17/30—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by a Diels-Alder synthesis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/35—Preparation of halogenated hydrocarbons by reactions not affecting the number of carbon or of halogen atoms in the reaction
    • C07C17/354—Preparation of halogenated hydrocarbons by reactions not affecting the number of carbon or of halogen atoms in the reaction by hydrogenation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/04—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups
    • C07C209/06—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups by substitution of halogen atoms
    • C07C209/10—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups by substitution of halogen atoms with formation of amino groups bound to carbon atoms of six-membered aromatic rings or from amines having nitrogen atoms bound to carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/24—Preparation of compounds containing amino groups bound to a carbon skeleton by reductive alkylation of ammonia, amines or compounds having groups reducible to amino groups, with carbonyl compounds
    • C07C209/26—Preparation of compounds containing amino groups bound to a carbon skeleton by reductive alkylation of ammonia, amines or compounds having groups reducible to amino groups, with carbonyl compounds by reduction with hydrogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/68—Preparation of compounds containing amino groups bound to a carbon skeleton from amines, by reactions not involving amino groups, e.g. reduction of unsaturated amines, aromatisation, or substitution of the carbon skeleton
    • C07C209/70—Preparation of compounds containing amino groups bound to a carbon skeleton from amines, by reactions not involving amino groups, e.g. reduction of unsaturated amines, aromatisation, or substitution of the carbon skeleton by reduction of unsaturated amines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/43—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C211/57—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings being part of condensed ring systems of the carbon skeleton
    • C07C211/60—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings being part of condensed ring systems of the carbon skeleton containing a ring other than a six-membered aromatic ring forming part of at least one of the condensed ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/43—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C211/57—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings being part of condensed ring systems of the carbon skeleton
    • C07C211/61—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings being part of condensed ring systems of the carbon skeleton with at least one of the condensed ring systems formed by three or more rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C25/00—Compounds containing at least one halogen atom bound to a six-membered aromatic ring
    • C07C25/18—Polycyclic aromatic halogenated hydrocarbons
    • C07C25/22—Polycyclic aromatic halogenated hydrocarbons with condensed rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C25/00—Compounds containing at least one halogen atom bound to a six-membered aromatic ring
    • C07C25/24—Halogenated aromatic hydrocarbons with unsaturated side chains
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/09—Geometrical isomers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/56—Ring systems containing bridged rings
    • C07C2603/58—Ring systems containing bridged rings containing three rings
    • C07C2603/60—Ring systems containing bridged rings containing three rings containing at least one ring with less than six members
    • C07C2603/66—Ring systems containing bridged rings containing three rings containing at least one ring with less than six members containing five-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Catalysts (AREA)

Abstract

Proceso para la preparación de compuestos derivados de 5-amino-benzonorborneno que comprende hacer reaccionar un compuesto derivado de 5-halo-benzonorborneno con una bencilamina en presencia de una catalizador de paladio.
CL2012000114A 2005-12-12 2012-01-13 Proceso para la preparacion de compuestos derivados de 5-amino-benzonorbornadieno donde se hacer reaccionar un compuesto de 5-halo-benzonorbornadieno con una bencilamina en prensecia de un catalizador de paladio. CL2012000114A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP05027072 2005-12-12
EP06008248 2006-04-21

Publications (1)

Publication Number Publication Date
CL2012000114A1 true CL2012000114A1 (es) 2012-08-31

Family

ID=37946810

Family Applications (2)

Application Number Title Priority Date Filing Date
CL2010000015A CL2010000015A1 (es) 2005-12-12 2010-01-08 Proceso de preparacion de un amino benzonorbornadieno por reaccion entre un halo benzonorbornadieno y una bencilamina en presencia de una base y una cantidad catalitica de al menos un complejo de paladio, (divisional sol. n° 3444-06).
CL2012000114A CL2012000114A1 (es) 2005-12-12 2012-01-13 Proceso para la preparacion de compuestos derivados de 5-amino-benzonorbornadieno donde se hacer reaccionar un compuesto de 5-halo-benzonorbornadieno con una bencilamina en prensecia de un catalizador de paladio.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
CL2010000015A CL2010000015A1 (es) 2005-12-12 2010-01-08 Proceso de preparacion de un amino benzonorbornadieno por reaccion entre un halo benzonorbornadieno y una bencilamina en presencia de una base y una cantidad catalitica de al menos un complejo de paladio, (divisional sol. n° 3444-06).

Country Status (21)

Country Link
US (1) US7781615B2 (es)
EP (5) EP2316809B1 (es)
JP (1) JP5144533B2 (es)
KR (1) KR101364220B1 (es)
CN (3) CN101360703B (es)
AR (1) AR058302A1 (es)
AU (1) AU2006326289B2 (es)
BR (1) BRPI0619629B1 (es)
CA (1) CA2631973C (es)
CL (2) CL2010000015A1 (es)
CR (1) CR10052A (es)
DK (1) DK1963251T3 (es)
EA (1) EA014275B1 (es)
EC (1) ECSP088525A (es)
EG (1) EG25547A (es)
ES (1) ES2391904T3 (es)
IL (3) IL191760A (es)
IN (1) IN2015DN00818A (es)
PL (1) PL1963251T3 (es)
TW (1) TWI396676B (es)
WO (1) WO2007068417A2 (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL1963251T3 (pl) * 2005-12-12 2013-01-31 Syngenta Participations Ag Proces wytwarzania amin
EA019915B1 (ru) 2007-09-20 2014-07-30 Басф Се Фунгицидная композиция для борьбы с фитопатогенными вредными грибами
KR20110026018A (ko) 2008-07-04 2011-03-14 바스프 에스이 치환된 1-메틸피라졸-4-일카르복스아닐리드를 포함하는 살진균 혼합물
US9115043B2 (en) 2008-10-27 2015-08-25 Syngenta Crop Protection, Llc Process for the preparation of benzonorbornenes
MX2011006425A (es) 2008-12-24 2011-07-20 Syngenta Ltd Metodos para la preparacion de fungicidas.
CN102858749B (zh) * 2010-04-20 2014-07-02 先正达参股股份有限公司 吡唑羧酸酰胺的制备方法
WO2012065947A1 (en) 2010-11-15 2012-05-24 Bayer Cropscience Ag 5-halogenopyrazolecarboxamides
RU2493145C1 (ru) * 2012-10-02 2013-09-20 Федеральное государственное бюджетное образовательное учреждение высшего профессионального образования "Волгоградский государственный технический университет" (ВолгГТУ) Способ получения 2-(аминоалкил)-3-(аминофенил)бицикло[2.2.1]гептанов
WO2014158614A1 (en) 2013-03-14 2014-10-02 Dow Agrosciences Llc Broadleaf crop control with 6-arylpicoline carboxylic acids, 2-arylpyrimidine carboxylic acids, or salts or esters thereof
US11560384B2 (en) 2017-05-04 2023-01-24 University Of Utah Research Foundation Benzonorbornadiene derivatives and reactions thereof

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1086978A (en) * 1965-09-21 1967-10-11 Shionogi & Co Improvements in or relating to the preparation of 7-oxobenzonorbornene derivatives
JPH075487B2 (ja) 1985-11-14 1995-01-25 住友化学工業株式会社 １―ブロモ―２―クロロ―４―フルオロベンゼンの製造法
US7223879B2 (en) 1998-07-10 2007-05-29 Massachusetts Institute Of Technology Ligands for metals and improved metal-catalyzed processes based thereon
WO2002076922A1 (en) * 2001-03-16 2002-10-03 Idemitsu Kosan Co., Ltd. Method for producing aromatic amino compound
JP4219622B2 (ja) * 2002-06-11 2009-02-04 独立行政法人科学技術振興機構 ベンザイン化合物の新規製造法
PL375353A1 (en) 2002-08-22 2005-11-28 Syngenta Participations Ag Chemical compounds
GB0224316D0 (en) * 2002-10-18 2002-11-27 Syngenta Participations Ag Chemical compounds
PL1963251T3 (pl) * 2005-12-12 2013-01-31 Syngenta Participations Ag Proces wytwarzania amin

Also Published As

Publication number Publication date
TWI396676B (zh) 2013-05-21
EP2316809A1 (en) 2011-05-04
CA2631973C (en) 2015-02-03
IL218350A0 (en) 2012-04-30
EA014275B1 (ru) 2010-10-29
EP2316813B1 (en) 2013-04-03
EP2316815A1 (en) 2011-05-04
CN104151132B (zh) 2016-07-06
PL1963251T3 (pl) 2013-01-31
AU2006326289B2 (en) 2011-12-22
CL2010000015A1 (es) 2010-07-02
WO2007068417A3 (en) 2007-10-04
EP1963251B1 (en) 2012-08-15
CN102516086B (zh) 2014-10-22
BRPI0619629A2 (pt) 2011-10-04
IL218351A0 (en) 2012-04-30
EP2316814A1 (en) 2011-05-04
CN104151132A (zh) 2014-11-19
EP2316813A1 (en) 2011-05-04
KR20080077011A (ko) 2008-08-20
EP2316809B1 (en) 2014-06-18
US7781615B2 (en) 2010-08-24
IL218351A (en) 2014-05-28
CA2631973A1 (en) 2007-06-21
US20090221856A1 (en) 2009-09-03
KR101364220B1 (ko) 2014-02-21
ECSP088525A (es) 2008-07-30
CN101360703B (zh) 2012-07-18
DK1963251T3 (da) 2012-11-26
IN2015DN00818A (es) 2015-07-10
EG25547A (en) 2012-02-15
JP2009518346A (ja) 2009-05-07
CN101360703A (zh) 2009-02-04
ES2391904T3 (es) 2012-11-30
AR058302A1 (es) 2008-01-30
TW200800854A (en) 2008-01-01
JP5144533B2 (ja) 2013-02-13
EP1963251A2 (en) 2008-09-03
IL191760A (en) 2014-05-28
WO2007068417A2 (en) 2007-06-21
EA200870038A1 (ru) 2008-10-30
CR10052A (es) 2008-09-17
CN102516086A (zh) 2012-06-27
AU2006326289A1 (en) 2007-06-21
BRPI0619629B1 (pt) 2016-03-01
IL191760A0 (en) 2008-12-29

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