CL2007003723A1 -
SUBSTITUTED CYCLICAL OR HETEROCICLIC COMPOUNDS, NON-STEROID MODULATORS OF THE PROGESTERONE RECEIVER; PHARMACEUTICAL COMPOSITION; AND USE TO TREAT AND / OR PREVENT GYNECOLOGICAL DISEASES SUCH AS ENDOMETRIOSIS AND DISMENORREA, DEPENDENT TUMORS
- Google Patents
SUBSTITUTED CYCLICAL OR HETEROCICLIC COMPOUNDS, NON-STEROID MODULATORS OF THE PROGESTERONE RECEIVER; PHARMACEUTICAL COMPOSITION; AND USE TO TREAT AND / OR PREVENT GYNECOLOGICAL DISEASES SUCH AS ENDOMETRIOSIS AND DISMENORREA, DEPENDENT TUMORS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE102007023614Aexternal-prioritypatent/DE102007023614A1/en
Application filed by Bayer Schering Pharma AgfiledCriticalBayer Schering Pharma Ag
Publication of CL2007003723A1publicationCriticalpatent/CL2007003723A1/en
CL2007003723A2006-12-212007-12-20
SUBSTITUTED CYCLICAL OR HETEROCICLIC COMPOUNDS, NON-STEROID MODULATORS OF THE PROGESTERONE RECEIVER; PHARMACEUTICAL COMPOSITION; AND USE TO TREAT AND / OR PREVENT GYNECOLOGICAL DISEASES SUCH AS ENDOMETRIOSIS AND DISMENORREA, DEPENDENT TUMORS
CL2007003723A1
(en)
New amide compounds used for treatment of gynecological diseases e.g. endometriosis, for female fertility control and female hormone replacement therapy, has general formula
SUBSTITUTED CYCLICAL OR HETEROCICLIC COMPOUNDS, NON-STEROID MODULATORS OF THE PROGESTERONE RECEIVER; PHARMACEUTICAL COMPOSITION; AND USE TO TREAT AND / OR PREVENT GYNECOLOGICAL DISEASES SUCH AS ENDOMETRIOSIS AND DISMENORREA, DEPENDENT TUMORS
COMPOUNDS DERIVED FROM INDOL-3-PROPIONIC ACID; PHARMACEUTICAL COMPOSITION; AND USE IN THE TREATMENT OF DISEASES SUCH AS HYPERLIPIDEMIA, HYPERTENSION; AMONG OTHER.
COMPOUNDS DERIVED FROM QUINAZOLINA SUBSTITUTES, INHIBITORS OF QUINASA; PHARMACEUTICAL COMPOSITION; AND USE IN THE TREATMENT OF DISEASES SUCH AS CANCER, ATEROSCLEROSIS AND ARTHRITIS.
ARIL-SUBSTITUTED HETEROCICLIC COMPOUNDS, TYPE I CANNABINOID RECEIVER MODULATORS (CB1); PREPARATION PROCESS; PHARMACEUTICAL COMPOSITION; AND USE IN THE TREATMENT OF SUCH DISEASES AS METABOLIC DISORDERS AND COGNITIVE DISORDERS.
COMPOUNDS DERIVED FROM REPLACED INDOL, INHIBITORS OF THE 5-LIPOXYGENASE ACTIVATING PROTEIN (FLAP); PHARMACEUTICAL COMPOSITION; AND USE IN THE TREATMENT OF SUCH DISEASES AS COPD, CARDIOVASCULAR DISEASE AND INFLAMMATION.
COMPOUNDS DERIVED FROM BENCIMIDAZOL; PREPARATION PROCEDURE; PHARMACEUTICAL COMPOSITIONS; AND USE FOR THE TREATMENT AND / OR PROFILAXIS OF DISEASES MODULATED WITH FXR AGONISTS, SUCH AS DISLIPIDEMIAS, DIABETES, CANCER, OSTEOPOROSIS AND E
Compounds derived from 4,5-dihydro-oxazol-2-ylamine; preparation procedure; pharmaceutical composition; and its use for the treatment of Alzheimer's disease.
COMPOUNDS DERIVED FROM AZAESPIRO; PREPARATION PROCEDURE; PHARMACEUTICAL COMPOSITION; AND ITS USE TO PREVENT AND TREAT ANXIETY, DEPRESSIVE DISORDERS, AMONG OTHER DISEASES.
Compounds derived from carboxamide and urea comprising aromatic substituted pyrazole, vanilloid receptor binders; pharmaceutical composition that includes them; and its use in the treatment and / or prophylaxis of pain, migraine, parkinson's disease, gastrointestinal disorders, osteoporosis, among other diseases.
COMPOUNDS DERIVED FROM PROGESTERONA, ANTAGONISTS OF THE PROGESTERONE RECEIVER; PHARMACEUTICAL COMPOSITION; AND USE FOR THE TREATMENT OF ENDOMETRIOSIS, MYOMAS OR TUMORS DEPENDENT ON HORMONES.
COMPOUNDS DERIVED FROM 1H-INDOL-2-CARBOXAMIDE; PREPARATION PROCEDURE, PHARMACEUTICAL COMPOSITION; AND USE FOR THE TREATMENT AND / OR PREVENTION OF DISEASES ASSOCIATED WITH THE MODULATION OF H3 RECEPTORS AS OBESITY, TYPE II DIABETES AND
COMPOUNDS DERIVED FROM SUBSTITUTED AMIDAS; PROCESS FOR THE PREPARATION OF SUCH COMPOUNDS; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH COMPOUNDS; AND ITS USE FOR THE TREATMENT OF INSOMNIUM, SEXUAL DYSFUNCTION, SCHIZOPHRENIA, BETWEEN OTHER SICK
CRYSTAL FORMS OF THE HEMI ALISQUIRENE FUMARATE; PREPARATION PROCEDURE; PHARMACEUTICAL COMPOSITION THAT INCLUDES SUCH CRYSTAL FORMS; AND ITS USE TO TREAT DISEASES THAT ARE MODULATED WITH AT1 RECEIVER BLOCK, SUCH AS REGULATION