CL2007000773A1 - Uso de compuestos derivados de diazepina condensada para el tratamiento de un desorden cognitivo como add o adhd;o su uso para tratar spm o pmdd. - Google Patents
Uso de compuestos derivados de diazepina condensada para el tratamiento de un desorden cognitivo como add o adhd;o su uso para tratar spm o pmdd.Info
- Publication number
- CL2007000773A1 CL2007000773A1 CL2007000773A CL2007000773A CL2007000773A1 CL 2007000773 A1 CL2007000773 A1 CL 2007000773A1 CL 2007000773 A CL2007000773 A CL 2007000773A CL 2007000773 A CL2007000773 A CL 2007000773A CL 2007000773 A1 CL2007000773 A1 CL 2007000773A1
- Authority
- CL
- Chile
- Prior art keywords
- diazepine
- condensed
- treatment
- pmdd
- adhd
- Prior art date
Links
- LRANPJDWHYRCER-UHFFFAOYSA-N 1,2-diazepine Chemical compound N1C=CC=CC=N1 LRANPJDWHYRCER-UHFFFAOYSA-N 0.000 title abstract 2
- 208000010877 cognitive disease Diseases 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 title abstract 2
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/498—Pyrazines or piperazines ortho- and peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Anesthesiology (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Uso de compuestos derivados de diazepina condensada en el tratamiento de un desorden cognitivo.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US78565406P | 2006-03-24 | 2006-03-24 | |
| US85127806P | 2006-10-12 | 2006-10-12 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CL2007000773A1 true CL2007000773A1 (es) | 2008-01-25 |
Family
ID=38235219
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CL2007000773A CL2007000773A1 (es) | 2006-03-24 | 2007-03-23 | Uso de compuestos derivados de diazepina condensada para el tratamiento de un desorden cognitivo como add o adhd;o su uso para tratar spm o pmdd. |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US20070225278A1 (es) |
| EP (1) | EP2015749A2 (es) |
| JP (1) | JP2009531431A (es) |
| KR (1) | KR20080105105A (es) |
| AR (1) | AR060088A1 (es) |
| AU (1) | AU2007229491A1 (es) |
| BR (1) | BRPI0709146A2 (es) |
| CA (1) | CA2644618A1 (es) |
| CL (1) | CL2007000773A1 (es) |
| EC (1) | ECSP088764A (es) |
| IL (1) | IL193697A0 (es) |
| MX (1) | MX2008012208A (es) |
| NO (1) | NO20083751L (es) |
| PA (1) | PA8720401A1 (es) |
| PE (1) | PE20080126A1 (es) |
| RU (1) | RU2008135115A (es) |
| TW (1) | TW200806297A (es) |
| WO (1) | WO2007111982A2 (es) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GT200500317A (es) * | 2004-11-05 | 2006-10-27 | Proceso para preparar compuestos de quinolina y productos obtenidos de los mismos | |
| AR051946A1 (es) * | 2004-11-05 | 2007-02-21 | Wyeth Corp | Formulaciones de derivados de [1,4] diazepina [6,7,1-ij] quinolina |
| PE20060939A1 (es) * | 2004-11-05 | 2006-11-10 | Wyeth Corp | Metabolitos derivados de [1,4] diazepin[6,7,1-ij] quinolina y procedimiento de preparacion |
| AR054849A1 (es) * | 2005-07-26 | 2007-07-18 | Wyeth Corp | Diazepinoquinolinas, sintesis de las mismas, e intermediarios para obtenerlas |
| TW200734334A (en) * | 2006-01-13 | 2007-09-16 | Wyeth Corp | Treatment of substance abuse |
| JP2009531435A (ja) * | 2006-03-24 | 2009-09-03 | ワイス | うつ病の治療用の新規な治療組み合わせ |
| CN101405005A (zh) * | 2006-03-24 | 2009-04-08 | 惠氏公司 | 调节膀胱功能的方法 |
| MX2008012092A (es) * | 2006-03-24 | 2008-10-03 | Wyeth Corp | Tratamiento del dolor. |
| CL2008002777A1 (es) * | 2007-09-21 | 2010-01-22 | Wyeth Corp | Metodo de preparacion de compuestos diazepinoquinolinicos quirales por recristalizacion en un sistema de solvente ternario. |
Family Cites Families (46)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3158619A (en) * | 1962-06-14 | 1964-11-24 | Searle & Co | Certain sulfur-containing ortho-fused polycyclic pyrazole derivatives |
| US3235564A (en) * | 1964-03-27 | 1966-02-15 | Searle & Co | Intermediates to certain sulfur-containing ortho-fused polycyclic pyrazole derivatives |
| US3296252A (en) * | 1964-04-02 | 1967-01-03 | Sandoz Ag | Tetracyclic diazepinone compounds |
| US3335134A (en) * | 1964-04-02 | 1967-08-08 | Sandoz Ag | Certain 3, 4-dihydrofluoreno[1, 9a, 9-e, f]1, 4-diazepin-3(2h)-ones |
| GB1120462A (en) * | 1964-07-06 | 1968-07-17 | Manuf Prod Pharma | 3-alkoxy-2h-fluoreno[1,9-ef]-1,4-diazepine 1-oxides and derivatives thereof |
| US3417101A (en) * | 1964-11-09 | 1968-12-17 | American Home Prod | Fused ring compounds |
| US3329676A (en) * | 1964-11-09 | 1967-07-04 | American Home Prod | Fused 1, 4-diazepine ring systems |
| US3714149A (en) * | 1969-11-03 | 1973-01-30 | Upjohn Co | Pyridobenzodiazepinones |
| US3914250A (en) * | 1974-08-01 | 1975-10-21 | American Home Prod | 1,4-Diazepino{8 6,5,4-jk{9 carbazoles |
| US4880814A (en) * | 1987-11-13 | 1989-11-14 | Abbott Laboratories | 7-cycloalkyl naphthyridines |
| GB8812636D0 (en) * | 1988-05-27 | 1988-06-29 | Glaxo Group Ltd | Chemical compounds |
| US4997831A (en) * | 1988-09-01 | 1991-03-05 | Glaxo Group Limited | Lactam derivatives |
| US5376645A (en) * | 1990-01-23 | 1994-12-27 | University Of Kansas | Derivatives of cyclodextrins exhibiting enhanced aqueous solubility and the use thereof |
| KR0166088B1 (ko) * | 1990-01-23 | 1999-01-15 | . | 수용해도가 증가된 시클로덱스트린 유도체 및 이의 용도 |
| US5565483A (en) * | 1995-06-07 | 1996-10-15 | Bristol-Myers Squibb Company | 3-substituted oxindole derivatives as potassium channel modulators |
| NZ314105A (en) * | 1996-02-02 | 1997-12-19 | Sumitomo Pharma | Guanidine derivative substituted with a substituted indole which is peri condensed with a heterocyclic ring |
| GB9711643D0 (en) * | 1997-06-05 | 1997-07-30 | Janssen Pharmaceutica Nv | Glass thermoplastic systems |
| US6031098A (en) * | 1997-08-11 | 2000-02-29 | California Institute Of Technology | Detection and treatment of duplex polynucleotide damage |
| CA2328197C (en) * | 1998-04-14 | 2007-11-20 | The General Hospital Corporation | Methods for treating neuropsychiatric disorders |
| CO5210925A1 (es) * | 1998-11-17 | 2002-10-30 | Novartis Ag | Derivados de diamino nitroguanidina tetrasustituidos |
| US6503900B2 (en) * | 2000-11-03 | 2003-01-07 | Wyeth | [1,4]diazepino [6,7,1-jk ]carbazoles and derivatives |
| US6858604B2 (en) * | 2000-11-03 | 2005-02-22 | Wyeth | Cyclohepta[b][1,4]diazepino[6,7,1-hi]indoles and derivatives |
| US6777407B2 (en) * | 2000-11-03 | 2004-08-17 | Wyeth | Cyclopenta[b][1,4]diazepino[6,7,1-hi]indoles and derivatives |
| WO2002036596A2 (en) * | 2000-11-03 | 2002-05-10 | Wyeth | CYCLOALKYL[b][1,4]DIAZEPINO[6,7,1-hi]INDOLES AND DERIVATIVES |
| AR031195A1 (es) * | 2000-11-03 | 2003-09-10 | Wyeth Corp | Procedimiento para la preparacion de derivados de 1,2,3,4,8,9,10,10a-octahidro-7bh-ciclopenta (b) (1,4) diazepino (6,7,1) diazepino (6,7,1-hi) indol |
| US6414144B1 (en) * | 2000-11-03 | 2002-07-02 | Wyeth | Process for preparation of cyclopenta[b][1,4]diazepino[6,7,1-hi] indole derivatives |
| AR031200A1 (es) * | 2000-11-03 | 2003-09-10 | Wyeth Corp | Cicloocta [b] [1,4] diazepino [6,7,1-hi] indoles y derivados |
| BR0116429A (pt) * | 2000-12-20 | 2006-05-09 | Bristol Myers Squibb Co | piridoindóis substituìdos como agonistas e antagonistas da serotonina |
| US6849619B2 (en) * | 2000-12-20 | 2005-02-01 | Bristol-Myers Squibb Company | Substituted pyridoindoles as serotonin agonists and antagonists |
| AR033095A1 (es) * | 2001-04-04 | 2003-12-03 | Wyeth Corp | Metodos para el tratamiento de motilidad gastrica hiperactiva |
| BR0211559A (pt) * | 2001-08-06 | 2004-07-13 | Upjohn Co | Compostos, composições de ligantes tetracìclicos terapeuticamente úteis e seus usos |
| EP1436294A1 (en) * | 2001-10-18 | 2004-07-14 | PHARMACIA & UPJOHN COMPANY | Tetracyclic azaindoles and -indolines having serotonin 5-ht2c activity |
| TWI312781B (en) * | 2002-04-25 | 2009-08-01 | [1,4]diazepino[6,7,1-ij]quinoline derivatives as antipsychotic and antiobesity agents | |
| TW200307682A (en) * | 2002-04-25 | 2003-12-16 | Wyeth Corp | 1,2,3,4,7,8-Hexahydro-6H-[1,4]diazepino[6,7,1-ij]quinoline derivatives as antipsychotic and antiobesity agents |
| TW200307540A (en) * | 2002-04-25 | 2003-12-16 | Wyeth Corp | [1, 4]Diazocino[7, 8, 1-hi] indole derivatives as antipsychotic and antiobesity agents |
| US20040235856A1 (en) * | 2003-04-25 | 2004-11-25 | Pfizer Inc | Treatment of incontinence |
| AR051946A1 (es) * | 2004-11-05 | 2007-02-21 | Wyeth Corp | Formulaciones de derivados de [1,4] diazepina [6,7,1-ij] quinolina |
| GT200500317A (es) * | 2004-11-05 | 2006-10-27 | Proceso para preparar compuestos de quinolina y productos obtenidos de los mismos | |
| PE20060939A1 (es) * | 2004-11-05 | 2006-11-10 | Wyeth Corp | Metabolitos derivados de [1,4] diazepin[6,7,1-ij] quinolina y procedimiento de preparacion |
| AR054849A1 (es) * | 2005-07-26 | 2007-07-18 | Wyeth Corp | Diazepinoquinolinas, sintesis de las mismas, e intermediarios para obtenerlas |
| PE20070549A1 (es) * | 2005-10-17 | 2007-06-15 | Wyeth Corp | Tetrahidroquinolinas, su sintesis e intermediarios |
| TW200734334A (en) * | 2006-01-13 | 2007-09-16 | Wyeth Corp | Treatment of substance abuse |
| MX2008012092A (es) * | 2006-03-24 | 2008-10-03 | Wyeth Corp | Tratamiento del dolor. |
| RU2008140136A (ru) * | 2006-03-24 | 2010-04-27 | Вайет (Us) | Новые терапевтические комбинации для лечения или профилактики психотических расстройств |
| JP2009531435A (ja) * | 2006-03-24 | 2009-09-03 | ワイス | うつ病の治療用の新規な治療組み合わせ |
| CL2008002777A1 (es) * | 2007-09-21 | 2010-01-22 | Wyeth Corp | Metodo de preparacion de compuestos diazepinoquinolinicos quirales por recristalizacion en un sistema de solvente ternario. |
-
2007
- 2007-03-23 TW TW096110126A patent/TW200806297A/zh unknown
- 2007-03-23 JP JP2009502880A patent/JP2009531431A/ja not_active Withdrawn
- 2007-03-23 WO PCT/US2007/007209 patent/WO2007111982A2/en not_active Ceased
- 2007-03-23 RU RU2008135115/14A patent/RU2008135115A/ru unknown
- 2007-03-23 EP EP07753807A patent/EP2015749A2/en not_active Withdrawn
- 2007-03-23 MX MX2008012208A patent/MX2008012208A/es not_active Application Discontinuation
- 2007-03-23 US US11/726,924 patent/US20070225278A1/en not_active Abandoned
- 2007-03-23 AR ARP070101210A patent/AR060088A1/es unknown
- 2007-03-23 CA CA002644618A patent/CA2644618A1/en not_active Abandoned
- 2007-03-23 PA PA20078720401A patent/PA8720401A1/es unknown
- 2007-03-23 CL CL2007000773A patent/CL2007000773A1/es unknown
- 2007-03-23 PE PE2007000325A patent/PE20080126A1/es not_active Application Discontinuation
- 2007-03-23 KR KR1020087023339A patent/KR20080105105A/ko not_active Withdrawn
- 2007-03-23 BR BRPI0709146-0A patent/BRPI0709146A2/pt not_active Application Discontinuation
- 2007-03-23 AU AU2007229491A patent/AU2007229491A1/en not_active Abandoned
-
2008
- 2008-08-26 IL IL193697A patent/IL193697A0/en unknown
- 2008-09-01 NO NO20083751A patent/NO20083751L/no not_active Application Discontinuation
- 2008-09-23 EC EC2008008764A patent/ECSP088764A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| MX2008012208A (es) | 2008-10-02 |
| EP2015749A2 (en) | 2009-01-21 |
| AR060088A1 (es) | 2008-05-21 |
| AU2007229491A1 (en) | 2007-10-04 |
| WO2007111982A2 (en) | 2007-10-04 |
| CA2644618A1 (en) | 2007-10-04 |
| KR20080105105A (ko) | 2008-12-03 |
| ECSP088764A (es) | 2008-10-31 |
| PA8720401A1 (es) | 2008-12-18 |
| BRPI0709146A2 (pt) | 2011-06-28 |
| RU2008135115A (ru) | 2010-04-27 |
| PE20080126A1 (es) | 2008-04-07 |
| WO2007111982A3 (en) | 2007-11-15 |
| JP2009531431A (ja) | 2009-09-03 |
| IL193697A0 (en) | 2009-08-03 |
| TW200806297A (en) | 2008-02-01 |
| US20070225278A1 (en) | 2007-09-27 |
| NO20083751L (no) | 2008-10-20 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CL2007000773A1 (es) | Uso de compuestos derivados de diazepina condensada para el tratamiento de un desorden cognitivo como add o adhd;o su uso para tratar spm o pmdd. | |
| CL2007001670A1 (es) | Uso de compuestos derivados de amina para el tratamiento de un trastorno mediado por citoquinas. | |
| CL2008001374A1 (es) | Compuestos derivados de pirazolo pirimidinas, inhibidores de pde9; composicion farmaceutica que comprende a dichos compuetos; utiles en el tratamiento de un trastorno neurodegenerativo y cognitivo tal como la enfermedad de alzheimer y esquizofrenia. | |
| CR20110326A (es) | Compuestos pirazina como inhibidores de fosfodiesterasa 10 | |
| CO6321189A2 (es) | Compuestos de tiazol y oxazol de bencen-sulfonamida | |
| MX360301B (es) | Moleculas pequeñas que contienen boro como agentes antiinflamatorios. | |
| ECSP088782A (es) | Compuestos nuevos | |
| CL2011000527A1 (es) | Compuestos derivados de benzofurano; composicion farmaceutica que los comprende;y su uso en el tratamiento de la hepatitis c. | |
| ECSP099410A (es) | Adsorbente de fosfato a base de hierro (iii)-carbohidrato | |
| CR11488A (es) | 4-fenilpiran 3,5-dionas, 4-feniltiopiran-3,5-dionas y 2-fenilciclohexan-1,3,5-trionas como herbicidas | |
| BRPI0821688A2 (pt) | mistura para o tratamento de fertilizantes contendo uréia | |
| MX354217B (es) | Composiciones y metodos para el tratamiento de leucemia. | |
| PA8740901A1 (es) | Compuestos organicos | |
| CL2007003774A1 (es) | Compuestos derivados de quinazolina sustituidos, inhibidores de quinasa; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como cancer, aterosclerosis y artritis. | |
| CL2009000650A1 (es) | Compuestos derivados de amino-pirazina, inhibidores de cinasa-pi 3; composicion farmaceutica; y uso para el tratamiento de condiciones inflamatorias o alérgicas, tales como enfermedades respiratorias, artritis reumatoide, colitis ulcerativa, entre otras | |
| EA201171367A1 (ru) | Винилиндазолильные соединения | |
| TN2011000187A1 (en) | Organic compounds | |
| SV2009003373A (es) | COMPUESTOS AMINO-5-[-4-(DIFLUOROMETOXI)FENIL SUSTITUIDO]-5- FENILIMIDAZOLONA COMO INHIBIDORES DE ß-SECRETASA REF. AM102759 | |
| UY32384A (es) | Nuevas bencenosulfonamidas como bloqueadores de canales de calcio | |
| EA201101477A1 (ru) | Органические соединения и их применение | |
| GT200900204A (es) | Compuestos complejos de hidrato de carbono y hierro | |
| BR112012006176A2 (pt) | inibidores macrocíclicos de jak | |
| MY150600A (en) | Use of opioid antagonists for treating urinary retention | |
| EA200971068A1 (ru) | Триазолиламинопиримидиновые соединения | |
| MX2009011346A (es) | Tapentadol para tratamiento de dolor con artritis. |