CL2006003737A1 - Uso de compuestos derivados de triazina o pirimidina sustituida, para tratar o prevenir enfermedades mediadas por los receptores de prokineticina 2 tales como trastornos gastrointestinales. - Google Patents
Uso de compuestos derivados de triazina o pirimidina sustituida, para tratar o prevenir enfermedades mediadas por los receptores de prokineticina 2 tales como trastornos gastrointestinales.Info
- Publication number
- CL2006003737A1 CL2006003737A1 CL200603737A CL2006003737A CL2006003737A1 CL 2006003737 A1 CL2006003737 A1 CL 2006003737A1 CL 200603737 A CL200603737 A CL 200603737A CL 2006003737 A CL2006003737 A CL 2006003737A CL 2006003737 A1 CL2006003737 A1 CL 2006003737A1
- Authority
- CL
- Chile
- Prior art keywords
- prokineticin
- triazine
- receptors
- treat
- gastrointestinal disorders
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US75498905P | 2005-12-29 | 2005-12-29 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CL2006003737A1 true CL2006003737A1 (es) | 2008-02-08 |
Family
ID=38017002
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CL200603737A CL2006003737A1 (es) | 2005-12-29 | 2006-12-28 | Uso de compuestos derivados de triazina o pirimidina sustituida, para tratar o prevenir enfermedades mediadas por los receptores de prokineticina 2 tales como trastornos gastrointestinales. |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US20080287445A1 (es) |
| EP (1) | EP1976528A2 (es) |
| JP (1) | JP2009522301A (es) |
| CN (1) | CN101405002A (es) |
| AR (1) | AR058407A1 (es) |
| CA (1) | CA2635845A1 (es) |
| CL (1) | CL2006003737A1 (es) |
| IL (1) | IL192426A0 (es) |
| WO (1) | WO2007079214A2 (es) |
Families Citing this family (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2008016522A2 (en) * | 2006-07-24 | 2008-02-07 | Gilead Sciences, Inc. | Hiv reverse transcriptase inhibitors |
| WO2009042765A1 (en) * | 2007-09-25 | 2009-04-02 | The Regents Of The University Of California | Methods of modulating prokineticin 2 for treatment of stress response and anxiety-related disorders |
| CA2704185C (en) * | 2007-10-30 | 2016-02-16 | Janssen Pharmaceutica N.V. | Amino-heteroaryl-containing prokineticin 1 receptor antagonists |
| WO2009074575A2 (en) | 2007-12-10 | 2009-06-18 | Novartis Ag | Organic compounds |
| US9150546B2 (en) * | 2009-02-13 | 2015-10-06 | Shionogi & Co., Ltd. | Triazine derivative and pharmaceutical composition comprising the same |
| CA2803545A1 (en) * | 2010-06-28 | 2012-01-12 | Janssen Pharmaceutica Nv | Prokineticin 1 receptor antagonists for the treatment of pain |
| EP2604260B1 (en) | 2010-08-10 | 2017-05-10 | Shionogi&Co., Ltd. | Novel heterocyclic derivatives and pharmaceutical composition containing same |
| MX346367B (es) | 2010-08-10 | 2017-03-16 | Shionogi & Co Ltd * | Derivado de triazina y composicion farmaceutica que tiene actividad analgesica que comprende el mismo. |
| CN102321015A (zh) * | 2011-06-30 | 2012-01-18 | 江苏德峰药业有限公司 | 一种抗艾滋病药物奈韦拉平关键中间体 2-(环丙胺基)-3-甲酸吡啶的制备方法 |
| US9550763B2 (en) | 2012-02-09 | 2017-01-24 | Shionogi & Co., Ltd. | Heterocyclic ring and carbocyclic derivative |
| GB201209587D0 (en) | 2012-05-30 | 2012-07-11 | Takeda Pharmaceutical | Therapeutic compounds |
| TWI637949B (zh) | 2013-06-14 | 2018-10-11 | 塩野義製藥股份有限公司 | 胺基三衍生物及含有其等之醫藥組合物 |
| EA029430B1 (ru) | 2013-06-21 | 2018-03-30 | Такеда Фармасьютикл Компани Лимитед | Производные 1-сульфонилпиперидина в качестве модуляторов рецепторов прокинетицина |
| GB201314286D0 (en) | 2013-08-08 | 2013-09-25 | Takeda Pharmaceutical | Therapeutic Compounds |
| KR101862493B1 (ko) | 2013-10-25 | 2018-05-29 | 노파르티스 아게 | Fgfr4 억제제로서의 고리-융합된 비시클릭 피리딜 유도체 |
| GB201320905D0 (en) | 2013-11-27 | 2014-01-08 | Takeda Pharmaceutical | Therapeutic compounds |
| JP6422164B2 (ja) | 2013-12-26 | 2018-11-14 | 塩野義製薬株式会社 | 含窒素6員環誘導体およびそれらを含有する医薬組成物 |
| ES2756748T3 (es) | 2014-10-03 | 2020-04-27 | Novartis Ag | Uso de derivados de piridilo bicíclicos de anillo fusionado como inhibidores de fgfr4 |
| GB201420095D0 (en) | 2014-11-12 | 2014-12-24 | Takeda Pharmaceutical | New use |
| US9802917B2 (en) | 2015-03-25 | 2017-10-31 | Novartis Ag | Particles of N-(5-cyano-4-((2-methoxyethyl)amino)pyridin-2-yl)-7-formyl-6-((4-methyl-2-oxopiperazin-1-yl)methyl)-3,4-dihydro-1,8-naphthyridine-1(2H)-carboxamide |
| EP3287443B1 (en) | 2015-04-24 | 2021-10-27 | Shionogi & Co., Ltd | 6-membered heterocyclic derivative and pharmaceutical composition comprising same |
| JP7212930B2 (ja) * | 2016-04-06 | 2023-01-26 | ザ リージェンツ オブ ザ ユニバーシティ オブ カリフォルニア | プロキネチシン2アゴニストおよびアンタゴニストを使用する概日および日周リズムの障害を処置するための組成物および方法 |
| CN110072862B (zh) | 2016-10-17 | 2022-05-13 | 盐野义制药株式会社 | 二环性含氮杂环衍生物及含有该衍生物的药物组合物 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MXPA05001783A (es) * | 2002-08-13 | 2005-04-25 | Warner Lambert Co | Derivados de pirimidina-2,4-diona como inhibidores de las metaloproteinasas de matriz. |
| WO2004087054A2 (en) * | 2003-03-25 | 2004-10-14 | The Regents Of The University Of California | Methods for modulating gastric secretion using prokineticin receptor antagonists. |
| JP2008534499A (ja) * | 2005-03-24 | 2008-08-28 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | プロキネチシン2受容体アンタゴニストとしてのピリミジンジオン誘導体 |
| MX2007011848A (es) * | 2005-03-24 | 2008-04-22 | Johnson & Johnson | Antagonistas del receptor de procineticina i. |
-
2006
- 2006-12-28 AR ARP060105854A patent/AR058407A1/es unknown
- 2006-12-28 CL CL200603737A patent/CL2006003737A1/es unknown
- 2006-12-28 WO PCT/US2006/049560 patent/WO2007079214A2/en not_active Ceased
- 2006-12-28 CA CA002635845A patent/CA2635845A1/en not_active Abandoned
- 2006-12-28 US US11/646,957 patent/US20080287445A1/en not_active Abandoned
- 2006-12-28 JP JP2008548764A patent/JP2009522301A/ja not_active Withdrawn
- 2006-12-28 CN CNA2006800534962A patent/CN101405002A/zh active Pending
- 2006-12-28 EP EP06848331A patent/EP1976528A2/en not_active Withdrawn
-
2008
- 2008-06-24 IL IL192426A patent/IL192426A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA2635845A1 (en) | 2007-07-12 |
| IL192426A0 (en) | 2009-02-11 |
| US20080287445A1 (en) | 2008-11-20 |
| JP2009522301A (ja) | 2009-06-11 |
| AR058407A1 (es) | 2008-01-30 |
| WO2007079214A2 (en) | 2007-07-12 |
| WO2007079214A3 (en) | 2007-08-30 |
| EP1976528A2 (en) | 2008-10-08 |
| CN101405002A (zh) | 2009-04-08 |
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