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CL2004000898A1 - COMPOUNDS DERIVED FROM TRIAZOLALQUILFENILAMINA OR TRIAZOLALQUILFENILAMIDA REPLACED BY OXAZOL AND ITS PHARMACEUTICALLY ACCEPTABLE SALTS; PREPARATION PROCESS; PHARMACEUTICAL COMPOSITION; AND USE OF THE COMPOUND IN THE TREATMENT OF CANCER. - Google Patents

COMPOUNDS DERIVED FROM TRIAZOLALQUILFENILAMINA OR TRIAZOLALQUILFENILAMIDA REPLACED BY OXAZOL AND ITS PHARMACEUTICALLY ACCEPTABLE SALTS; PREPARATION PROCESS; PHARMACEUTICAL COMPOSITION; AND USE OF THE COMPOUND IN THE TREATMENT OF CANCER.

Info

Publication number
CL2004000898A1
CL2004000898A1 CL200400898A CL2004000898A CL2004000898A1 CL 2004000898 A1 CL2004000898 A1 CL 2004000898A1 CL 200400898 A CL200400898 A CL 200400898A CL 2004000898 A CL2004000898 A CL 2004000898A CL 2004000898 A1 CL2004000898 A1 CL 2004000898A1
Authority
CL
Chile
Prior art keywords
cancer
pharmaceutically acceptable
triazolalquilfenilamina
triazolalquilfenilamida
oxazol
Prior art date
Application number
CL200400898A
Other languages
Spanish (es)
Inventor
Birgit Friebe Walt Bossenmaier
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=33395779&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2004000898(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of CL2004000898A1 publication Critical patent/CL2004000898A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

OBJETIVOS DE LA PRESENTE INVENCION SON LOS COMPUESTOS DE FORMULA (I) SUS SALES FARMACEUTICAMENTE ACEPTABLES, ENANTIOMERICAS, DIASTEREOISOMEROS, Y RACEMATOS, LA PREPARACION DE LOS COMPUESTOS ANTERIORMENTE MENCIONADOS, MEDICAMENTOS QUE LOS CONTIENEN Y SU FABRICACION, ASI COMO EL USO DE LOS COMPUESTOS ANTERIORMENTE MENCIONADOS, EN EL CONTROL O LA PREVENCION DE ENFERMEDADES TALES COMO CANCER.OBJECTIVES OF THE PRESENT INVENTION ARE THE COMPOUNDS OF FORMULA (I) ITS PHARMACEUTICALLY ACCEPTABLE, ENANTIOMERIC, DIASTEREOISOMERAL AND RACEMATE SALES, THE PREPARATION OF THE PREVIOUSLY MENTIONED COMPOUNDS, MEDICATIONS THAT FOLLOW THEM AND THE COMPOSITION OF , IN THE CONTROL OR PREVENTION OF DISEASES SUCH AS CANCER.

CL200400898A 2003-04-30 2004-04-28 COMPOUNDS DERIVED FROM TRIAZOLALQUILFENILAMINA OR TRIAZOLALQUILFENILAMIDA REPLACED BY OXAZOL AND ITS PHARMACEUTICALLY ACCEPTABLE SALTS; PREPARATION PROCESS; PHARMACEUTICAL COMPOSITION; AND USE OF THE COMPOUND IN THE TREATMENT OF CANCER. CL2004000898A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP03009908 2003-04-30

Publications (1)

Publication Number Publication Date
CL2004000898A1 true CL2004000898A1 (en) 2005-03-04

Family

ID=33395779

Family Applications (1)

Application Number Title Priority Date Filing Date
CL200400898A CL2004000898A1 (en) 2003-04-30 2004-04-28 COMPOUNDS DERIVED FROM TRIAZOLALQUILFENILAMINA OR TRIAZOLALQUILFENILAMIDA REPLACED BY OXAZOL AND ITS PHARMACEUTICALLY ACCEPTABLE SALTS; PREPARATION PROCESS; PHARMACEUTICAL COMPOSITION; AND USE OF THE COMPOUND IN THE TREATMENT OF CANCER.

Country Status (20)

Country Link
US (1) US7205326B2 (en)
EP (1) EP1622896B1 (en)
JP (1) JP2006515347A (en)
KR (1) KR100763293B1 (en)
CN (1) CN100345845C (en)
AR (1) AR044098A1 (en)
AT (1) ATE366252T1 (en)
AU (1) AU2004234060A1 (en)
BR (1) BRPI0409951A (en)
CA (1) CA2522809A1 (en)
CL (1) CL2004000898A1 (en)
CO (1) CO5640050A2 (en)
DE (1) DE602004007374T2 (en)
ES (1) ES2290701T3 (en)
MX (1) MXPA05011671A (en)
NO (1) NO20054495L (en)
RU (1) RU2005137033A (en)
TW (1) TW200423931A (en)
WO (1) WO2004096796A1 (en)
ZA (1) ZA200508694B (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200612914A (en) * 2004-03-05 2006-05-01 Hoffmann La Roche Novel oxidized thioether derivatives, their manufacture and use as pharmaceutical agents
FR2876692B1 (en) 2004-10-19 2007-02-23 Sanofi Aventis Sa 2-AMIDO-4-PHENYLTHIAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC USE
US20060116407A1 (en) * 2004-11-22 2006-06-01 Birgit Bossenmaier Amide derivatives
JP2009504586A (en) * 2005-08-08 2009-02-05 エフ.ホフマン−ラ ロシュ アーゲー Pyrazole derivatives, their production and use as pharmaceuticals
CN112920133B (en) * 2021-01-29 2022-09-16 中国医科大学 (E) -4-methyl-2- (4- (trifluoromethyl) styryl) oxazole compound and preparation method and application thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0912562A1 (en) 1996-07-19 1999-05-06 Takeda Chemical Industries, Ltd. Heterocyclic compounds, their production and use
PE20011178A1 (en) 2000-04-07 2001-11-19 Takeda Chemical Industries Ltd HETEROCYCLIC COMPOUNDS AND THEIR PRODUCTION

Also Published As

Publication number Publication date
AR044098A1 (en) 2005-08-24
NO20054495L (en) 2005-11-23
NO20054495D0 (en) 2005-09-28
AU2004234060A1 (en) 2004-11-11
BRPI0409951A (en) 2006-04-25
DE602004007374D1 (en) 2007-08-16
CN100345845C (en) 2007-10-31
MXPA05011671A (en) 2005-12-15
CN1780830A (en) 2006-05-31
EP1622896A1 (en) 2006-02-08
WO2004096796A1 (en) 2004-11-11
CA2522809A1 (en) 2004-11-11
KR20060006070A (en) 2006-01-18
RU2005137033A (en) 2006-06-27
EP1622896B1 (en) 2007-07-04
ES2290701T3 (en) 2008-02-16
KR100763293B1 (en) 2007-10-04
DE602004007374T2 (en) 2008-03-20
JP2006515347A (en) 2006-05-25
ZA200508694B (en) 2007-06-27
US20040254217A1 (en) 2004-12-16
CO5640050A2 (en) 2006-05-31
US7205326B2 (en) 2007-04-17
TW200423931A (en) 2004-11-16
ATE366252T1 (en) 2007-07-15

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