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CL2004000304A1 - Uso del acido 4-[1-hidroxi-4-[4-hidroxidifenilmetil)-1-piperidinil]butil]-alfa, alfa-dimetilbenceno acetico o una sal farmaceuticamente aceptable del mismo, para la preparacion de un medicamento util como antihistaminico, en pacientes que padecen un - Google Patents

Uso del acido 4-[1-hidroxi-4-[4-hidroxidifenilmetil)-1-piperidinil]butil]-alfa, alfa-dimetilbenceno acetico o una sal farmaceuticamente aceptable del mismo, para la preparacion de un medicamento util como antihistaminico, en pacientes que padecen un

Info

Publication number
CL2004000304A1
CL2004000304A1 CL200400304A CL2004000304A CL2004000304A1 CL 2004000304 A1 CL2004000304 A1 CL 2004000304A1 CL 200400304 A CL200400304 A CL 200400304A CL 2004000304 A CL2004000304 A CL 2004000304A CL 2004000304 A1 CL2004000304 A1 CL 2004000304A1
Authority
CL
Chile
Prior art keywords
pharmaceutically acceptable
acceptable salt
hydroxidifenylmetil
achetic
piperidinil
Prior art date
Application number
CL200400304A
Other languages
English (en)
Inventor
James K. Woodward
Richard R. Okerholm
Mark G Eller
Bruce E. Mcnutt
Original Assignee
Aventis Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27128589&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2004000304(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Aventis Inc filed Critical Aventis Inc
Publication of CL2004000304A1 publication Critical patent/CL2004000304A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pulmonology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CL200400304A 1992-05-11 2004-02-19 Uso del acido 4-[1-hidroxi-4-[4-hidroxidifenilmetil)-1-piperidinil]butil]-alfa, alfa-dimetilbenceno acetico o una sal farmaceuticamente aceptable del mismo, para la preparacion de un medicamento util como antihistaminico, en pacientes que padecen un CL2004000304A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US88080192A 1992-05-11 1992-05-11
US92289092A 1992-07-31 1992-07-31

Publications (1)

Publication Number Publication Date
CL2004000304A1 true CL2004000304A1 (es) 2005-05-27

Family

ID=27128589

Family Applications (1)

Application Number Title Priority Date Filing Date
CL200400304A CL2004000304A1 (es) 1992-05-11 2004-02-19 Uso del acido 4-[1-hidroxi-4-[4-hidroxidifenilmetil)-1-piperidinil]butil]-alfa, alfa-dimetilbenceno acetico o una sal farmaceuticamente aceptable del mismo, para la preparacion de un medicamento util como antihistaminico, en pacientes que padecen un

Country Status (16)

Country Link
US (7) US6037353A (es)
EP (1) EP0639976B1 (es)
JP (1) JPH07506828A (es)
KR (1) KR950701525A (es)
AT (1) ATE194913T1 (es)
AU (1) AU679910B2 (es)
CA (1) CA2134211C (es)
CL (1) CL2004000304A1 (es)
DE (1) DE69320952T2 (es)
DK (1) DK0639976T3 (es)
ES (1) ES2121084T3 (es)
HU (1) HU223774B1 (es)
MX (1) MX9302704A (es)
NO (1) NO307688B1 (es)
NZ (1) NZ251834A (es)
WO (1) WO1993023047A1 (es)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU223774B1 (hu) * 1992-05-11 2005-01-28 Merrell Dow Pharmaceuticals Inc. Terfenadinszármazékok alkalmazása antihisztamin hatású gyógyszerkészítmények előállítására
PT815860E (pt) 1992-08-03 2006-08-31 Sepracor Inc Carboxilato de terfenadina e tratamento de desordens alergicas.
WO1995010278A1 (en) * 1993-10-15 1995-04-20 Hoechst Marion Roussel, Inc. Treatment of allergic disorders with terfenadine carboxylate
IT1271417B (it) * 1993-10-15 1997-05-28 Erregierre Ind Chim Composti ad attivita' antiistaminica procedimento per la loro preperazione e composizioni farmaceutiche che li contengono.
DE69527429T2 (de) * 1994-05-18 2003-03-20 Aventis Pharmaceuticals Inc., Bridgewater Verfahren zur herstellung von wasserfreien und hydrat-formen von antihistaminischen piperinderivaten, polymerphe und pseudomorphe davon
US20030045722A1 (en) * 1994-05-18 2003-03-06 Henton Daniel R. Processes for preparing anhydrous and hydrate forms of antihistaminic piperidine derivatives, polymorphs and pseudomorphs thereof
AU701042B2 (en) * 1995-02-28 1999-01-21 Aventisub Llc Pharmaceutical composition for piperidinoalkanol compounds
SK283803B6 (sk) * 1997-08-26 2004-02-03 Aventis Pharmaceuticals Inc. Farmaceutický prostriedok vo forme dvojvrstvovej tabletky na kombinovanie piperidinoalkanolu s dekongestantom
US6194431B1 (en) 1998-04-14 2001-02-27 Paul D. Rubin Methods and compositions using terfenadine metabolites in combination with leukotriene inhibitors
US20030021849A1 (en) * 2001-04-09 2003-01-30 Ben-Zion Dolitzky Polymorphs of fexofenadine hydrochloride
US20020177608A1 (en) * 2001-04-09 2002-11-28 Ben-Zion Dolitzky Polymorphs of fexofenadine hydrochloride
EP2316468A1 (en) 2002-02-22 2011-05-04 Shire LLC Delivery system and methods for protecting and administering dextroamphetamine
AU2003248657A1 (en) * 2002-06-10 2003-12-22 Teva Pharmaceutical Industries Ltd. Polymorphic form xvi of fexofenadine hydrochloride
EP1393728A1 (en) * 2002-08-30 2004-03-03 Vrije Universiteit Inverse agonists acting at virus-encoded G protein-coupled receptors
US20050065183A1 (en) * 2003-07-31 2005-03-24 Indranil Nandi Fexofenadine composition and process for preparing
MXPA06012281A (es) * 2004-04-26 2007-07-18 Teva Pharma Formas cristalinas de clorhidrato de fexofenadina y procesos para su preparacion.
EP1685106A2 (en) * 2004-09-28 2006-08-02 Teva Pharmaceutical Industries, Inc. Fexofendadine crystal form and processes for its preparation thereof
US20090076080A1 (en) * 2007-09-19 2009-03-19 Protia, Llc Deuterium-enriched fexofenadine
US20090304826A1 (en) * 2008-05-30 2009-12-10 Fairfield Clinical Trials, Llc Method and composition for dermatoses

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4254129A (en) * 1979-04-10 1981-03-03 Richardson-Merrell Inc. Piperidine derivatives
US4285958A (en) * 1979-04-10 1981-08-25 Richardson-Merrell Inc. 1-Piperidine-alkylene ketones, pharmaceutical compositions thereof and method of use thereof
AR240018A1 (es) * 1987-10-07 1990-01-31 Merrell Pharma Inc Procedimiento para preparar una composicion que comprende derivados de piperidinoalcanol.
US4929605A (en) * 1987-10-07 1990-05-29 Merrell Dow Pharmaceuticals Inc. Pharmaceutical composition for piperidinoalkanol derivatives
HU223774B1 (hu) * 1992-05-11 2005-01-28 Merrell Dow Pharmaceuticals Inc. Terfenadinszármazékok alkalmazása antihisztamin hatású gyógyszerkészítmények előállítására
PT815860E (pt) * 1992-08-03 2006-08-31 Sepracor Inc Carboxilato de terfenadina e tratamento de desordens alergicas.

Also Published As

Publication number Publication date
JPH07506828A (ja) 1995-07-27
MX9302704A (es) 1994-06-30
US6037353A (en) 2000-03-14
HU223774B1 (hu) 2005-01-28
DE69320952D1 (de) 1998-10-15
ATE194913T1 (de) 2000-08-15
US20030055083A1 (en) 2003-03-20
US20100168166A1 (en) 2010-07-01
ES2121084T3 (es) 2002-02-16
US6187791B1 (en) 2001-02-13
CA2134211C (en) 1999-06-29
WO1993023047A1 (en) 1993-11-25
US20060205782A1 (en) 2006-09-14
EP0639976B1 (en) 2000-07-26
US20030130315A1 (en) 2003-07-10
AU679910B2 (en) 1997-07-17
EP0639976A1 (en) 1995-03-01
DK0639976T3 (da) 1999-02-15
NO307688B1 (no) 2000-05-15
US6399632B1 (en) 2002-06-04
AU3973493A (en) 1993-12-13
HUT71402A (en) 1995-11-28
NZ251834A (en) 1997-07-27
DE69320952T2 (de) 1999-05-27
CA2134211A1 (en) 1993-11-25
KR950701525A (ko) 1995-04-28
NO944287L (no) 1994-11-10
NO944287D0 (no) 1994-11-10

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