CA2607566A1 - Agonistes vis-a-vis du recepteur peptidique de type glucagon 1 (glp-1) et procedes pharmacologiques d'utilisation - Google Patents

Agonistes vis-a-vis du recepteur peptidique de type glucagon 1 (glp-1) et procedes pharmacologiques d'utilisation Download PDF

Info

Publication number: CA2607566A1
Authority: CA; Canada
Prior art keywords: peptide; lys; diabetes; cys; ala
Prior art date: 2005-05-06
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

CA002607566A

Other languages

English (en)

Inventor

James Whelan

Kevin Lumb

Kevin Clairmont

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Bayer Healthcare LLC

Original Assignee

Individual

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2005-05-06

Filing date

2006-05-05

Publication date

2006-11-16

2006-05-05 Application filed by Individual filed Critical Individual

2006-11-16 Publication of CA2607566A1 publication Critical patent/CA2607566A1/fr

Status Abandoned legal-status Critical Current

Links

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Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/705—Receptors; Cell surface antigens; Cell surface determinants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/28—Insulins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/43—Enzymes; Proenzymes; Derivatives thereof
- A61K38/45—Transferases (2)
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/43—Enzymes; Proenzymes; Derivatives thereof
- A61K38/46—Hydrolases (3)
- A61K38/48—Hydrolases (3) acting on peptide bonds (3.4)
- A61K38/4813—Exopeptidases (3.4.11. to 3.4.19)
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system

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Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical & Material Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Bioinformatics & Cheminformatics (AREA)
Public Health (AREA)
Organic Chemistry (AREA)
Diabetes (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Gastroenterology & Hepatology (AREA)
Immunology (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Epidemiology (AREA)
Endocrinology (AREA)
Hematology (AREA)
Obesity (AREA)
Zoology (AREA)
Emergency Medicine (AREA)
Biophysics (AREA)
Cardiology (AREA)
Child & Adolescent Psychology (AREA)
Cell Biology (AREA)
Toxicology (AREA)
Biochemistry (AREA)
Heart & Thoracic Surgery (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Micro-Organisms Or Cultivation Processes Thereof (AREA)

CA002607566A 2005-05-06 2006-05-05 Agonistes vis-a-vis du recepteur peptidique de type glucagon 1 (glp-1) et procedes pharmacologiques d'utilisation Abandoned CA2607566A1 (fr)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US67872305P	2005-05-06	2005-05-06
US60/678,723		2005-05-06
PCT/US2006/017411 WO2006121860A2 (fr)	2005-05-06	2006-05-05	Agonistes vis-a-vis du recepteur peptidique de type glucagon 1 (glp-1) et procedes pharmacologiques d'utilisation

Publications (1)

Publication Number	Publication Date
CA2607566A1 true CA2607566A1 (fr)	2006-11-16

Family

ID=37397130

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CA002607566A Abandoned CA2607566A1 (fr)	2005-05-06	2006-05-05	Agonistes vis-a-vis du recepteur peptidique de type glucagon 1 (glp-1) et procedes pharmacologiques d'utilisation

Country Status (4)

Country	Link
EP (1)	EP1883419A4 (fr)
JP (1)	JP2008539735A (fr)
CA (1)	CA2607566A1 (fr)
WO (1)	WO2006121860A2 (fr)

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KR102512178B1 (ko)	2011-05-18	2023-03-20	메더리스 다이어비티즈, 엘엘씨	개선된 펩티드 제약
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EP2567959B1 (fr)	2011-09-12	2014-04-16	Sanofi	Dérivés d'amide d'acide 6-(4-hydroxy-phényl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylique en tant qu'inhibiteurs de kinase
WO2013045413A1 (fr)	2011-09-27	2013-04-04	Sanofi	Dérivés d'amide d'acide 6-(4-hydroxyphényl)-3-alkyl-1h-pyrazolo[3,4-b] pyridine-4-carboxylique utilisés comme inhibiteurs de kinase
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CN109456400A (zh)	2012-07-23	2019-03-12	西兰制药公司	胰高血糖素类似物
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US11065304B2 (en)	2012-11-20	2021-07-20	Mederis Diabetes, Llc	Peptide pharmaceuticals for insulin resistance
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AP2016009212A0 (en)	2013-10-17	2016-05-31	Zealand Pharma As	Acylated glucagon analogues
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AU2014345570B2 (en)	2013-11-06	2019-01-24	Zealand Pharma A/S	Glucagon-GLP-1-GIP triple agonist compounds
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2006
- 2006-05-05 EP EP06759154A patent/EP1883419A4/fr not_active Withdrawn
- 2006-05-05 CA CA002607566A patent/CA2607566A1/fr not_active Abandoned
- 2006-05-05 JP JP2008510259A patent/JP2008539735A/ja active Pending
- 2006-05-05 WO PCT/US2006/017411 patent/WO2006121860A2/fr not_active Ceased

Also Published As

Publication number	Publication date
EP1883419A2 (fr)	2008-02-06
WO2006121860A2 (fr)	2006-11-16
EP1883419A4 (fr)	2010-08-04
WO2006121860A3 (fr)	2007-04-12
JP2008539735A (ja)	2008-11-20

Publication	Publication Date	Title
CA2607566A1 (fr)	2006-11-16	Agonistes vis-a-vis du recepteur peptidique de type glucagon 1 (glp-1) et procedes pharmacologiques d'utilisation
WO2006121904A1 (fr)	2006-11-16	Agonistes du recepteur du polypeptide insulinotropique gluco-dependant (gip) et procedes pharmacologiques d'utilisation associes
US7378494B2 (en)	2008-05-27	Pituitary adenylate cyclase activating peptide (PACAP) receptor (VPAC2) agonist peptide
WO2004022004A2 (fr)	2004-03-18	Agonistes modifies du recepteur glp-1 et leurs procedes pharmacologiques d'utilisation
AU2013277372A1 (en)	2014-12-11	Analogs of glucagon exhibiting GIP receptor activity
US20080261863A1 (en)	2008-10-23	Pegylation of Vasoactive Intestinal Peptide (Vip) / Pituitary Adenylate Cyclase Activating Peptide (Pacap) Receptor 2 (Vpac2) Agonists and Methods of Use
WO2006049681A2 (fr)	2006-05-11	Agonistes recepteur y2 neuropeptidiques selectifs
US20090105122A1 (en)	2009-04-23	Selective neuropeptide y2 receptor agonists
US20090280106A1 (en)	2009-11-12	Pituitary adenylate cyclase acivating peptide (pacap) receptor (vpac2) agonists and their pharmacological methods of use
US20090143283A1 (en)	2009-06-04	Pituitary Adenylate Cyclase Activating Peptide (PACAP) Receptor (VPAC2) Agonists and Their Pharmacological Methods of Use
WO2006091506A2 (fr)	2006-08-31	Agonistes du recepteur y4 de neuropeptide
WO2006091505A2 (fr)	2006-08-31	Agonistes du recepteur y de neuropeptide
CN1913914A (zh)	2007-02-14	垂体腺苷酸环化酶激活肽(pacap)受体(vpac2)激动剂及其药理学使用方法
HK1131161A (en)	2010-01-15	Pituitary adenylate cyclase activating peptide (pacap) receptor (vpac2) agonists and their pharmacological methods of use
KR20050018988A (ko)	2005-02-28	뇌하수체 아데닐레이트 사이클라제 활성화펩타이드(ｐａｃａｐ) 수용체(ｖｐａｃ２) 효능제 및 그의약물학적 사용방법
MXPA06008404A (en)	2006-12-13	Pituitary adenylate cyclase activating peptide (pacap) receptor (vpac2) agonists and their pharmacological methods of use
HK1109855A (en)	2008-06-27	Pegylation of vasoactive intestinal peptide (vip)/pituitary adenylate cyclase activating peptide (pacap) receptor 2 (vpac2) agonists and methods of use

Legal Events

Date	Code	Title	Description
2012-05-07	FZDE	Dead