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CA2643747A1 - Autoimmune conditions and nadph oxidase defects - Google Patents

Autoimmune conditions and nadph oxidase defects Download PDF

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Publication number
CA2643747A1
CA2643747A1 CA002643747A CA2643747A CA2643747A1 CA 2643747 A1 CA2643747 A1 CA 2643747A1 CA 002643747 A CA002643747 A CA 002643747A CA 2643747 A CA2643747 A CA 2643747A CA 2643747 A1 CA2643747 A1 CA 2643747A1
Authority
CA
Canada
Prior art keywords
compound
alkyl
integer
alkynyl
cycloalkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002643747A
Other languages
French (fr)
Inventor
Marcel Linschoten
Anders Bergman
Tolmachev Andrey Alekseevich
Peter Olofsson
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Swedish Orphan Biovitrum AB
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2643747A1 publication Critical patent/CA2643747A1/en
Abandoned legal-status Critical Current

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/045Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Transplantation (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pain & Pain Management (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Dermatology (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

The invention relates to methods and materials involved in treating autoimmune conditions. In particular, the invention relates to methods and compounds (and compositions including the compounds) involved in treating, preventing, or delaying the onset of autoimmune conditions. The compounds can include one or more isoprenoid units. The compounds can enhance NADPH oxidase activity.

Claims (25)

1. Use of a compound wherein the compound has the following general formula:

m + n = an integer from 0-9;
X is selected from wherein represents a single or double bond between C2 and C3;
Y is -O-C(==O)R';

R' is H, alkyl, alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl, on heteroaryl, each of which is optionally substituted; and R'' is H, alkyl, alkenyl, alkynyl or cycloalkyl, each of which is optionally substituted;

in the manufacture of a medicament for the treatment of an autoimmune condition.
2. The use according to claim 1, wherein the compound has the general formula:

wherein:
m + n = an integer from 0-9;

represents a single or double bond between C2 and C3; and Y is -O-C(=O)R', wherein R' is H, alkyl, alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl; or heteroaryl, each of which is optionally substituted.
3. The use of claim 2, wherein R' is C1-C~ alkyl.
4, The use of claim 3, wherein R' is CH3.
5. The use of claim 2, wherein ~ + n = an integer from 0-5.
6. The use of claim 1, wherein one of m and n is 0, and the other is an integer from 1-5.
7. The use of claim 1, wherein m + n = 3.
8. The use of claim 7, wherein one of m and n is 0.
9. The use of claim 8, wherein n is 0.
10. The use of claim 2, wherein m + n = 2.
11. The use of claim 2, wherein represents a double bond between C2 and C3.
12. The use of claim 2, wherein the compound is selected from the group consisting of:

Farnesyl acetate (Acetic acid 3,7,11-trimethyl-dodeca-2,6,10-trienyl ester);
Phytyl acetate (Acetic acid 3,7,11,15-tetra-methyl-hexadec-2-enyl-ester);
Di-hydro-phytol (3,7,11,25-Tetramethyl-hexadecan-1-ol); and Di-hydro-phytyl acetate (Acetic acid 3,7,11,15-tetramethyl-hexadecyl ester);
13. The use according to claim 1, wherein the compound has the general formula:
wherein n+m= an integer from 0 to 9; and R' is H, alkyl, alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl, or heteroaryl, each of which is optionally substituted.
14. The use of claim 13, wherein m + n = 3
15. The use of claim 14, wherein n is 0.
16. The use of claim 13, wherein R' is hydrogen.
17. The use of claim 13, wherein the compound is 3,7,11,15-tetramethyl-1-hexadecen-3-ol.
18 . The use according to claim 1, wherein the compound has the general formula:
wherein n+m= an integer from 0 to 9, and R'' is H, alkyl, alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl, or heteroaryl, each of which is optionally substituted.
19. The use of claim 18, wherein m + n = 3.
20. The use of claim 19, wherein n is 0.
21. The use of claim 18, wherein R" is C1-C3 alkyl substituted with from 1-3 halogens.
22. The use of claim 18, wherein the compound is 6-difluoromethoxy-2,5,7,8-tetramethyl-2-(4,8,12-trimethyl-tridecyl)-chroman.
23. The use of any one of claims 1 to 22, wherein said autoimmune condition is arthritis.
24. The use of any one of claims 1 to 22, wherein said autoimmune condition is multiple sclerosis.
25. The use of any one of claims 1 to 22, wherein said autoimmune condition is inflammatory bowel disease.
CA002643747A 2006-03-15 2007-03-15 Autoimmune conditions and nadph oxidase defects Abandoned CA2643747A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US78238106P 2006-03-15 2006-03-15
US60/782,381 2006-03-15
PCT/EP2007/052457 WO2007104790A1 (en) 2006-03-15 2007-03-15 Autoimmune conditions and nadph oxidase defects

Publications (1)

Publication Number Publication Date
CA2643747A1 true CA2643747A1 (en) 2007-09-20

Family

ID=38236360

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002643747A Abandoned CA2643747A1 (en) 2006-03-15 2007-03-15 Autoimmune conditions and nadph oxidase defects

Country Status (8)

Country Link
EP (1) EP2004159A1 (en)
JP (1) JP2010521412A (en)
KR (1) KR20090008233A (en)
CN (1) CN101404985A (en)
AU (1) AU2007224438B2 (en)
CA (1) CA2643747A1 (en)
NZ (1) NZ570803A (en)
WO (1) WO2007104790A1 (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB201104600D0 (en) 2011-03-18 2011-05-04 Pronoxis Ab New compounds and medical uses
US10780061B2 (en) 2014-09-26 2020-09-22 Daegu Gyeongbuk Institute Of Science And Technology Composition comprising farnesol and use thereof
RU2631887C2 (en) * 2015-09-07 2017-09-28 Вагиф Султанович Султанов Active drug ingredient, drug, pharmaceutical composition and method for treatment of demyelinating diseases of living organism, including disease prevention
FR3110427B1 (en) * 2020-05-20 2023-07-14 Laboratoires Eriger Coupling terpene conjugate
JP2024501949A (en) * 2020-12-23 2024-01-17 アクセス ツー アドバンスト ヘルス インスティチュート Solanesol vaccine adjuvant and its preparation method

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS61257944A (en) * 1986-03-20 1986-11-15 Nisshin Flour Milling Co Ltd Remedy for ulcer
US4983637A (en) * 1988-06-24 1991-01-08 Stephen Herman Method for treating viral infection of HIV
US5475029A (en) * 1993-07-08 1995-12-12 The Board Of Trustees Of The Leland Stanford Junior University Farnesyl compounds as cholesterol lowering agents
JPH10168090A (en) * 1996-12-11 1998-06-23 Eisai Co Ltd Apoptotic inducer
US6703384B2 (en) * 1998-09-23 2004-03-09 Research Development Foundation Tocopherols, tocotrienols, other chroman and side chain derivatives and uses thereof
JP2001172171A (en) * 1999-10-06 2001-06-26 Kazuhito Rokutan Revulsive for heat shock protein
GB0019290D0 (en) * 2000-08-04 2000-09-27 Symphar Sa Methods for inducing apolipoprotein E secretion
JP4578235B2 (en) * 2002-05-13 2010-11-10 アレクシス・アクチボラゲット Autoimmune status and NADPH oxidase deficiency
KR20070044805A (en) * 2004-04-15 2007-04-30 키아스마, 인코포레이티드 Compositions That Can Promote Biological Barrier Permeation
FR2869230B1 (en) * 2004-04-23 2006-07-28 Alessio Patrizia D COMPOSITION FOR PREVENTING OR TREATING CELL DEGENERATION WITH AT LEAST ONE MOLECULE CAPABLE OF MAINTAINING THE REVERSIBILITY OF ADHESION MOLECULE EXPRESSION AND POLYMERIZATION OF ACTIN FIBERS

Also Published As

Publication number Publication date
JP2010521412A (en) 2010-06-24
WO2007104790A1 (en) 2007-09-20
CN101404985A (en) 2009-04-08
KR20090008233A (en) 2009-01-21
AU2007224438A1 (en) 2007-09-20
AU2007224438B2 (en) 2012-07-26
NZ570803A (en) 2011-06-30
EP2004159A1 (en) 2008-12-24

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FZDE Discontinued

Effective date: 20140317