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CA2157037A1 - Derives de la benzylimidazopyridine, antagonistes du recepteur de l'angiotensine ii - Google Patents

Derives de la benzylimidazopyridine, antagonistes du recepteur de l'angiotensine ii

Info

Publication number
CA2157037A1
CA2157037A1 CA002157037A CA2157037A CA2157037A1 CA 2157037 A1 CA2157037 A1 CA 2157037A1 CA 002157037 A CA002157037 A CA 002157037A CA 2157037 A CA2157037 A CA 2157037A CA 2157037 A1 CA2157037 A1 CA 2157037A1
Authority
CA
Canada
Prior art keywords
compound according
ethyl
alkyl
pyridin
methylphenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002157037A
Other languages
English (en)
Inventor
Paul A. Da Silva Jardine
Ronald T. Wester
Philip A. Carpino
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Corp SRL
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2157037A1 publication Critical patent/CA2157037A1/fr
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CA002157037A 1993-03-10 1994-02-14 Derives de la benzylimidazopyridine, antagonistes du recepteur de l'angiotensine ii Abandoned CA2157037A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US4395893A 1993-03-10 1993-03-10
US08/043,958 1993-03-10

Publications (1)

Publication Number Publication Date
CA2157037A1 true CA2157037A1 (fr) 1994-09-15

Family

ID=21929806

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002157037A Abandoned CA2157037A1 (fr) 1993-03-10 1994-02-14 Derives de la benzylimidazopyridine, antagonistes du recepteur de l'angiotensine ii

Country Status (7)

Country Link
EP (1) EP0690859A1 (fr)
JP (1) JPH08502757A (fr)
AU (1) AU6297494A (fr)
CA (1) CA2157037A1 (fr)
FI (1) FI941117L (fr)
IL (1) IL108842A0 (fr)
WO (1) WO1994020499A1 (fr)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4200954A1 (de) * 1991-04-26 1992-10-29 Bayer Ag Heterocyclisch substituierte phenylessigsaeurederivate

Also Published As

Publication number Publication date
FI941117A7 (fi) 1994-09-11
AU6297494A (en) 1994-09-26
WO1994020499A1 (fr) 1994-09-15
EP0690859A1 (fr) 1996-01-10
FI941117L (fi) 1994-09-11
JPH08502757A (ja) 1996-03-26
IL108842A0 (en) 1994-06-24
FI941117A0 (fi) 1994-03-09

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Legal Events

Date Code Title Description
EEER Examination request
FZDE Discontinued