BRPI0813903A2 - Processos para a prepração de pirazóis - Google Patents

Processos para a prepração de pirazóis

Info

Publication number: BRPI0813903A2
Authority: BR; Brazil
Prior art keywords: pirazois; preparing; processes; preparing pirazois
Prior art date: 2007-06-27

Application number

BRPI0813903-2A2A

Other languages

English (en)

Inventor

Martin Charles Bowden

Brian David Gott

David Anthony Jackson

Original Assignee

Syngenta Participations Ag

Syngenta Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2007-06-27

Filing date

2008-06-16

Publication date

2014-12-30

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38812166&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0813903(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2008-06-16 Application filed by Syngenta Participations Ag, Syngenta Ltd filed Critical Syngenta Participations Ag

2014-12-30 Publication of BRPI0813903A2 publication Critical patent/BRPI0813903A2/pt

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/16—Halogen atoms or nitro radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
- C07C251/72—Hydrazones
- C07C251/74—Hydrazones having doubly-bound carbon atoms of hydrazone groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C251/76—Hydrazones having doubly-bound carbon atoms of hydrazone groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of a saturated carbon skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Plural Heterocyclic Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

BRPI0813903-2A2A 2007-06-27 2008-06-16 Processos para a prepração de pirazóis BRPI0813903A2 (pt)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP07012546A EP2008996A1 (en)	2007-06-27	2007-06-27	Process for the production of pyrazoles
PCT/EP2008/004830 WO2009000442A2 (en)	2007-06-27	2008-06-16	Processes for the preparation of pyrazoles

Publications (1)

Publication Number	Publication Date
BRPI0813903A2 true BRPI0813903A2 (pt)	2014-12-30

Family

ID=38812166

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
BRPI0813903-2A2A BRPI0813903A2 (pt)	2007-06-27	2008-06-16	Processos para a prepração de pirazóis
BRPI0813284-4A BRPI0813284B1 (pt)	2007-06-27	2008-06-16	Process for the preparation of a compound of the formula (I) and compound

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
BRPI0813284-4A BRPI0813284B1 (pt)	2007-06-27	2008-06-16	Process for the preparation of a compound of the formula (I) and compound

Country Status (18)

Country	Link
US (3)	US20100256390A1 (pt)
EP (3)	EP2008996A1 (pt)
JP (2)	JP2010531315A (pt)
KR (2)	KR20100025533A (pt)
CN (3)	CN102516175A (pt)
AR (2)	AR067355A1 (pt)
AU (2)	AU2008267472A1 (pt)
BR (2)	BRPI0813903A2 (pt)
CA (2)	CA2690246A1 (pt)
CL (2)	CL2008001897A1 (pt)
CO (2)	CO6251313A2 (pt)
CR (2)	CR11161A (pt)
EC (2)	ECSP099817A (pt)
IL (2)	IL202419A0 (pt)
MX (2)	MX2009013592A (pt)
RU (2)	RU2010102137A (pt)
TW (2)	TW200916445A (pt)
WO (2)	WO2009000441A1 (pt)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP2008996A1 (en) *	2007-06-27	2008-12-31	Syngeta Participations AG	Process for the production of pyrazoles
EP2133341A1 (de) *	2008-02-25	2009-12-16	Bayer CropScience AG	Verfahren zur regioselektiven Synthese von 1-Alkyl-3-haloalkyl-pyrazol-4-carbonsäure-Derivaten
KR20160131129A (ko)	2008-09-30	2016-11-15	솔베이(소시에떼아노님)	할로겐화 환형 화합물의 합성 방법
GB0908435D0 (en) *	2009-05-15	2009-06-24	Syngenta Ltd	Processes
WO2012025469A1 (en) *	2010-08-24	2012-03-01	Solvay Sa	Improved process for the preparation of esters of 1-h-pyrazole-4-carboxylic acids
FR2975992B1 (fr) *	2011-06-01	2013-11-08	Rhodia Operations	Procede de preparation d'un compose fluoromethylpyrazole sous forme acide carboxylique ou derivee
FR2975990B1 (fr) *	2011-06-01	2013-05-24	Rhodia Operations	Procede de preparation d'un compose organique fluore
JP6101345B2 (ja) *	2012-05-14	2017-03-22	バイエル・クロップサイエンス・アクチェンゲゼルシャフト	１−アルキル−３−フルオロアルキル−１ｈ−ピラゾール−４−カルボニルクロライド類の製造方法
US8871947B2 (en)	2013-02-04	2014-10-28	KingChem LLC	Preparation of alkyl 3-difluoromethyl-1-methyl-1H-pyrazole-4-carboxylic acid ester
WO2015059067A1 (de)	2013-10-23	2015-04-30	Bayer Cropscience Ag	Verfahren zur herstellung von halogenketonen
CN103570623B (zh) *	2013-11-12	2015-05-20	湖南化工研究院	一种3-(二氟甲基)-1-甲基-1h-吡唑-4-羧酸的制备方法
WO2015085464A1 (en)	2013-12-09	2015-06-18	King Chem, Llc	Process for preparing alkyl 3-difluoromethyl-1-methyl-1h-pyrazole-4-carboxylate and its analogs
CN103787977B (zh)	2014-01-21	2016-05-25	南通雅本化学有限公司	一种空气氧化制备3-氟代烷基-1-取代吡唑-4-羧酸的方法
CN105541716B (zh)	2015-03-26	2024-02-23	Ａｇｃ株式会社	吡唑衍生物的制造方法
CN104945325B (zh) *	2015-06-19	2017-04-05	浙江永太科技股份有限公司	一种吡唑甲酸衍生物的制备方法
ES2844530T3 (es)	2015-06-19	2021-07-22	Zhejiang Yongtai Technology Co Ltd	Método para preparar un derivado del ácido pirazolcarboxílico e intermedio del mismo
WO2017054112A1 (zh)	2015-09-28	2017-04-06	常州市卜弋科研化工有限公司	3-氟代烷基-1-甲基吡唑-4-羧酸的制备方法
CN106554311B (zh) *	2015-09-28	2019-03-01	常州市卜弋科研化工有限公司	3-氟代烷基-1-甲基吡唑-4-羧酸的制备方法
CN112041303A (zh)	2018-05-21	2020-12-04	Pi工业有限公司	制备取代的杂环化合物的方法
CN109232425A (zh) *	2018-10-16	2019-01-18	山东省农药科学研究院	一种苯丙烯氟菌唑中间体3-(二氟甲基)-1-甲基-1h-吡唑-4-羧酸的合成方法
CN110577503A (zh)	2019-08-02	2019-12-17	宿迁市科莱博生物化学有限公司	一种卤素取代化合物及其制备方法和应用
CN111303035A (zh) *	2020-03-18	2020-06-19	徐州圣元化工有限公司	一种3-(二氟甲基)-1-甲基-1h-吡唑-4-羧酸的制备方法
CN111233768B (zh) *	2020-03-18	2021-08-03	徐州圣元化工有限公司	一种3-(二氟甲基)-1-甲基-1h-吡唑-4-羧酸乙酯的制备方法
WO2022233129A1 (en)	2021-05-05	2022-11-10	Fujian Yongjing Technology Co., Ltd	New process for the synthesis of 5-fluoro-3- (difuoromethyl) -5-fluoro-1-methyl-1h-pyrazole-4-carboxylic acid derivatives and the free acid thereof
CN114195715B (zh) *	2021-12-31	2024-05-10	福建永晶科技股份有限公司	1-甲基-3-二氟甲基-4-吡唑酸和1-甲基-3-三氟甲基-4-吡唑酸的制备方法
CN117384096A (zh) *	2023-12-13	2024-01-12	山东国邦药业有限公司	一种二氟吡唑酸的制备方法
CN117447401B (zh) *	2023-12-26	2024-04-19	山东国邦药业有限公司	一种二氟吡唑酸的合成方法
CN119241439B (zh) *	2024-12-05	2025-03-07	湖南斯派克科技股份有限公司	一种农药中间体二氟吡唑酸的合成方法

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPH0759557B2 (ja) *	1987-12-25	1995-06-28	三井東圧化学株式会社	１，３−ジアルキルピラゾール−４−アルデヒド誘導体の製造方法
JPH0759558B2 (ja) *	1987-12-25	1995-06-28	三井東圧化学株式会社	１，３−ジアルキルピラゾール−４−アルデヒド類の製造法
JPH089599B2 (ja) *	1988-08-02	1996-01-31	三井東圧化学株式会社	ピラゾールカルボン酸類の製造方法
EP1565150A1 (fr) *	2002-11-20	2005-08-24	L'oreal	Utilisation d'un compose pyrazolcarboxamide pour stimuler la pousse des fibres keratiniques et/ou freiner leur chute
DE10349500A1 (de) *	2003-10-23	2005-06-02	Bayer Cropscience Ag	Verfahren zum Herstellen von 2-Dihalogenacyl-3-amino-acrylsäureestern und 3-Dihalogenmethyl-pyrazol-4-carbonsäureestern
ES2345261T3 (es) *	2004-02-27	2010-09-20	Eli Lilly And Company	Derivados de 4-amino-piperidina como inhibidores de la captacion de monoamina.
PE20060096A1 (es) *	2004-06-18	2006-03-16	Basf Ag	(orto-fenil)-anilidas de acido 1-metil-3-difluorometil-pirazol-4-carboxilico como agentes fungicidas
CA2577525C (en) *	2004-08-18	2010-03-30	Pfizer Inc.	Inhibitors of hepatitis c virus rna-dependent rna polymerase, and compositions and treatments using the same
CN101133031B (zh) *	2005-02-25	2010-07-21	财团法人相模中央化学研究所	1-取代-3-氟代烷基吡唑-4-羧酸酯的制造方法
EP2253623B1 (en) *	2005-09-16	2013-10-23	Syngenta Participations AG.	New crystal form of a pyrazole fungicide
CA2686659A1 (en) *	2007-06-01	2008-12-04	Basf Se	Method for the production of n-substituted (3-dihalomethyl-1-methylpyrazol-4-yl)carboxamides
EP2008996A1 (en) *	2007-06-27	2008-12-31	Syngeta Participations AG	Process for the production of pyrazoles

2007
- 2007-06-27 EP EP07012546A patent/EP2008996A1/en not_active Ceased
2008
- 2008-06-16 EP EP08773461A patent/EP2167461B1/en active Active
- 2008-06-16 US US12/665,738 patent/US20100256390A1/en not_active Abandoned
- 2008-06-16 BR BRPI0813903-2A2A patent/BRPI0813903A2/pt not_active Application Discontinuation
- 2008-06-16 CN CN2011103836384A patent/CN102516175A/zh active Pending
- 2008-06-16 KR KR1020097026870A patent/KR20100025533A/ko not_active Withdrawn
- 2008-06-16 RU RU2010102137/04A patent/RU2010102137A/ru not_active Application Discontinuation
- 2008-06-16 JP JP2010513718A patent/JP2010531315A/ja active Pending
- 2008-06-16 CN CN200880021857A patent/CN101796021A/zh active Pending
- 2008-06-16 MX MX2009013592A patent/MX2009013592A/es not_active Application Discontinuation
- 2008-06-16 CA CA2690246A patent/CA2690246A1/en not_active Abandoned
- 2008-06-16 AU AU2008267472A patent/AU2008267472A1/en not_active Abandoned
- 2008-06-16 RU RU2010102135/04A patent/RU2010102135A/ru not_active Application Discontinuation
- 2008-06-16 JP JP2010513717A patent/JP5563449B2/ja active Active
- 2008-06-16 EP EP08773462A patent/EP2170832A2/en not_active Withdrawn
- 2008-06-16 BR BRPI0813284-4A patent/BRPI0813284B1/pt active IP Right Grant
- 2008-06-16 WO PCT/EP2008/004829 patent/WO2009000441A1/en not_active Ceased
- 2008-06-16 MX MX2009013591A patent/MX2009013591A/es active IP Right Grant
- 2008-06-16 CA CA002689218A patent/CA2689218A1/en not_active Abandoned
- 2008-06-16 WO PCT/EP2008/004830 patent/WO2009000442A2/en not_active Ceased
- 2008-06-16 US US12/666,179 patent/US8269020B2/en active Active
- 2008-06-16 KR KR1020097026780A patent/KR20100025531A/ko not_active Withdrawn
- 2008-06-16 CN CN200880022057A patent/CN101687806A/zh active Pending
- 2008-06-16 AU AU2008267473A patent/AU2008267473A1/en not_active Abandoned
- 2008-06-23 TW TW097123281A patent/TW200916445A/zh unknown
- 2008-06-23 TW TW097123280A patent/TW200914428A/zh unknown
- 2008-06-26 CL CL2008001897A patent/CL2008001897A1/es unknown
- 2008-06-26 CL CL2008001896A patent/CL2008001896A1/es unknown
- 2008-06-27 AR ARP080102804A patent/AR067355A1/es not_active Application Discontinuation
- 2008-06-27 AR ARP080102805A patent/AR067356A1/es not_active Application Discontinuation
2009
- 2009-11-30 IL IL202419A patent/IL202419A0/en unknown
- 2009-12-10 IL IL202664A patent/IL202664A/en active IP Right Grant
- 2009-12-14 CO CO09142558A patent/CO6251313A2/es not_active Application Discontinuation
- 2009-12-14 CR CR11161A patent/CR11161A/es not_active Application Discontinuation
- 2009-12-14 CR CR11162A patent/CR11162A/es not_active Application Discontinuation
- 2009-12-14 CO CO09142556A patent/CO6251314A2/es not_active Application Discontinuation
- 2009-12-18 EC EC2009009817A patent/ECSP099817A/es unknown
- 2009-12-18 EC EC2009009818A patent/ECSP099818A/es unknown
2012
- 2012-09-17 US US13/621,686 patent/US8785657B2/en active Active

Also Published As

Publication number	Publication date
CN101687806A (zh)	2010-03-31
CL2008001896A1 (es)	2009-03-06
AR067355A1 (es)	2009-10-07
EP2167461B1 (en)	2012-08-08
CA2690246A1 (en)	2008-12-31
JP2010531314A (ja)	2010-09-24
EP2170832A2 (en)	2010-04-07
AR067356A1 (es)	2009-10-07
CN102516175A (zh)	2012-06-27
WO2009000442A2 (en)	2008-12-31
KR20100025531A (ko)	2010-03-09
MX2009013591A (es)	2010-01-20
US20130023668A1 (en)	2013-01-24
WO2009000441A8 (en)	2010-01-14
US20100240907A1 (en)	2010-09-23
EP2167461A1 (en)	2010-03-31
US8785657B2 (en)	2014-07-22
EP2008996A1 (en)	2008-12-31
CO6251314A2 (es)	2011-02-21
CN101796021A (zh)	2010-08-04
US8269020B2 (en)	2012-09-18
WO2009000442A8 (en)	2010-01-21
CO6251313A2 (es)	2011-02-21
WO2009000441A1 (en)	2008-12-31
AU2008267472A1 (en)	2008-12-31
IL202419A0 (en)	2010-06-30
RU2010102137A (ru)	2011-08-10
BRPI0813284B1 (pt)	2017-10-31
CR11162A (es)	2010-04-21
JP5563449B2 (ja)	2014-07-30
TW200914428A (en)	2009-04-01
JP2010531315A (ja)	2010-09-24
CL2008001897A1 (es)	2009-01-02
IL202664A0 (en)	2010-06-30
ECSP099818A (es)	2010-01-29
CR11161A (es)	2010-05-19
CA2689218A1 (en)	2008-12-31
KR20100025533A (ko)	2010-03-09
WO2009000442A3 (en)	2009-07-23
BRPI0813284A8 (pt)	2017-04-04
MX2009013592A (es)	2010-01-20
ECSP099817A (es)	2010-01-29
RU2010102135A (ru)	2011-08-10
US20100256390A1 (en)	2010-10-07
TW200916445A (en)	2009-04-16
BRPI0813284A2 (pt)	2014-12-30
AU2008267473A1 (en)	2008-12-31
IL202664A (en)	2014-07-31

Publication	Publication Date	Title
BRPI0813284A2 (pt)	2014-12-30	Processos para a preparação de pirazóis
BRPI0819568A2 (pt)	2017-07-04	métodos para a preparação de um composto
BRPI0819238A2 (pt)	2014-10-07	Métodos para a produção de caseína
BRPI0820733A2 (pt)	2015-06-16	Processo para a preparação de macrociclo
BRPI0919050A2 (pt)	2015-12-08	dispositivo para o preparo de uma bebida
BRPI0812999A2 (pt)	2014-12-23	Método para preparar um composto
BRPI0817978A2 (pt)	2015-04-07	Métodos para preparar um catalisador de polimerização
BRPI0817836A2 (pt)	2015-03-31	Método para a produção de cerveja
BRPI0810139A2 (pt)	2014-10-29	Catalisador para a preparação de metil mercaptano
BRPI0816911A2 (pt)	2015-03-17	Processo para preparação de 4-aminobut-2-enolidas
BRPI0821129A2 (pt)	2015-06-16	Métodos para a inibição de cicatrização
BRPI0812422A2 (pt)	2014-12-02	Processo de preparação de um aldeído hidroxiaromático
BRPI0809652A2 (pt)	2014-10-07	Processo melhorado para a síntese de solifenacina
BRPI0914674A2 (pt)	2015-10-20	processo para preparação de um pó
BRPI0807870A2 (pt)	2014-06-17	Método para a produção de um revestimento
BRPI0820548A8 (pt)	2015-09-29	métodos para a formação de artigos microsporosos e microbicidas
BRPI0923297A2 (pt)	2015-07-28	Processos para a fabricação de um composto, e para a preparação de um composto imdiazolinona herbicida
BRPI0808031A2 (pt)	2014-06-17	Processo para a preparação de di-n-butil tereftalato
BRPI0811315A2 (pt)	2015-01-27	Processo para a preparação de um composto
BRPI0915242A2 (pt)	2016-02-16	método para a preparação de um polímero
BRPI0814011A2 (pt)	2016-03-22	método para preparação de biobutanol
BRPI0813482A2 (pt)	2015-02-03	Processo para preparar dimetacrilatos de butanodiol
BRPI0811510A2 (pt)	2014-11-18	Método para a produção de moldes
BRPI0922087A2 (pt)	2015-08-11	Processos para fabricar um composto e para preparar um composto
BRPI0813319A2 (pt)	2014-12-23	Método para preparar um composto, e, composto

Legal Events

Date	Code	Title
2015-01-20	B06F	Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
2015-04-07	B11E	Dismissal acc. art. 34 of ipl - requirements for examination incomplete
2020-09-24	B11T	Dismissal of application maintained [chapter 11.20 patent gazette]