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BRPI0514125A - piridinas condensadas como inibidores de cinase - Google Patents

piridinas condensadas como inibidores de cinase

Info

Publication number
BRPI0514125A
BRPI0514125A BRPI0514125-7A BRPI0514125A BRPI0514125A BR PI0514125 A BRPI0514125 A BR PI0514125A BR PI0514125 A BRPI0514125 A BR PI0514125A BR PI0514125 A BRPI0514125 A BR PI0514125A
Authority
BR
Brazil
Prior art keywords
kinase inhibitors
condensed
condensed pyridines
pyridines
compounds
Prior art date
Application number
BRPI0514125-7A
Other languages
English (en)
Inventor
Carmen Almansa Rosales
Marina Virgili Bernado
Pedro Manuel Grima Poveda
Original Assignee
Palau Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Palau Pharma Sa filed Critical Palau Pharma Sa
Publication of BRPI0514125A publication Critical patent/BRPI0514125A/pt

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
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Abstract

PIRIDINAS CONDENSADAS COMO INIBIDORES DE CINASE. Novos compostos de fórmula I, em que os significados para os vários substituintes são como descritas na descrição. Estes compostos são úteis como inibidores de p38 cinase.
BRPI0514125-7A 2004-08-03 2005-08-02 piridinas condensadas como inibidores de cinase BRPI0514125A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ES200401971 2004-08-03
PCT/EP2005/008371 WO2006013095A2 (en) 2004-08-03 2005-08-02 Condensed pyridines as kinase inhibitors

Publications (1)

Publication Number Publication Date
BRPI0514125A true BRPI0514125A (pt) 2008-05-27

Family

ID=35741197

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0514125-7A BRPI0514125A (pt) 2004-08-03 2005-08-02 piridinas condensadas como inibidores de cinase

Country Status (15)

Country Link
US (1) US20090264446A9 (pt)
EP (1) EP1833828A2 (pt)
JP (1) JP2008508341A (pt)
KR (1) KR20070045227A (pt)
CN (1) CN1993360A (pt)
AR (1) AR050188A1 (pt)
AU (1) AU2005268845A1 (pt)
BR (1) BRPI0514125A (pt)
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