BRPI0509305A - uso de um sensibilizador insulìnico, composição farmecêutica, e , kit - Google Patents
uso de um sensibilizador insulìnico, composição farmecêutica, e , kitInfo
- Publication number
- BRPI0509305A BRPI0509305A BRPI0509305-8A BRPI0509305A BRPI0509305A BR PI0509305 A BRPI0509305 A BR PI0509305A BR PI0509305 A BRPI0509305 A BR PI0509305A BR PI0509305 A BRPI0509305 A BR PI0509305A
- Authority
- BR
- Brazil
- Prior art keywords
- insulin sensitizer
- pharmaceutical composition
- kit
- suppressed
- effects
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/192—Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/421—1,3-Oxazoles, e.g. pemoline, trimethadione
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Diabetes (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
"USO DE UM SENSIBILIZADOR INSULìNICO, COMPOSIçãO FARMACêUTICA, E, KIT" Um objeto da presente invenção é prover um método altamente seguro para tratar uma doença, em que os efeitos colaterais (por exemplo, edema) sejam suprimidos ao mesmo tempo em que se mantenha excelentes efeitos farmacêuticos. E fornecida uma composição farmacêutica que inclui um sensibilizador insulínico como um ingrediente ativo, caracterizada em um ciclo de administração do sensibilizador insulínico em que a sua dosagem seja reduzida ou suprimida durante o período de administração, é repetido uma vez ou mais.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2004094598 | 2004-03-29 | ||
| PCT/JP2005/005526 WO2005092382A1 (ja) | 2004-03-29 | 2005-03-25 | インスリン抵抗性改善剤を含有する糖尿病治療剤 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0509305A true BRPI0509305A (pt) | 2007-09-04 |
Family
ID=35055995
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0509305-8A BRPI0509305A (pt) | 2004-03-29 | 2005-03-25 | uso de um sensibilizador insulìnico, composição farmecêutica, e , kit |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20070049515A1 (pt) |
| EP (1) | EP1731170A1 (pt) |
| KR (1) | KR20070011329A (pt) |
| CN (1) | CN1972715A (pt) |
| BR (1) | BRPI0509305A (pt) |
| CA (1) | CA2560928A1 (pt) |
| TW (1) | TW200536515A (pt) |
| WO (1) | WO2005092382A1 (pt) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2007058504A1 (en) * | 2005-11-21 | 2007-05-24 | Lg Life Sciences, Ltd. | Novel compounds as agonist for ppar gamma and ppar alpha, method for preparation of the same, and pharmaceutical composition containing the same |
| TW200730173A (en) * | 2005-12-16 | 2007-08-16 | Sankyo Co | Pharmaceutical composition enhancing production of adiponectin |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR240698A1 (es) * | 1985-01-19 | 1990-09-28 | Takeda Chemical Industries Ltd | Procedimiento para preparar compuestos de 5-(4-(2-(5-etil-2-piridil)-etoxi)benzil)-2,4-tiazolidindiona y sus sales |
| EP0306228B1 (en) * | 1987-09-04 | 1999-11-17 | Beecham Group Plc | Substituted thiazolidinedione derivatives |
| US5594016A (en) * | 1992-12-28 | 1997-01-14 | Mitsubishi Chemical Corporation | Naphthalene derivatives |
| CZ293016B6 (cs) * | 1995-06-01 | 2004-01-14 | Sankyo Company Limited | Benzimidazolové deriváty a farmaceutické prostředky s jejich obsahem |
| EA002357B1 (ru) * | 1995-12-28 | 2002-04-25 | Фудзисава Фармасьютикал Ко., Лтд. | Производные бензимидазола |
| AR029876A1 (es) * | 1998-05-11 | 2003-07-23 | Takeda Pharmaceutical | Compuesto de acido oxiiminoalcanoilo, composicion farmaceutica y agente para controlar receptores relacionados con retinoide que lo comprenden y su uso |
| TWI284533B (en) * | 1999-05-24 | 2007-08-01 | Sankyo Co | Pharmaceutical composition for treating hyperglycemia, impaired glucose tolerance, diabetes complications and for improving insulin resistant |
| JP2002220336A (ja) * | 2000-11-22 | 2002-08-09 | Sankyo Co Ltd | 縮合複素環化合物の塩酸塩を含有する糖尿病の予防薬、治療薬 |
| WO2002051441A1 (en) * | 2000-12-26 | 2002-07-04 | Sankyo Company, Limited | Medicinal compositions containing diuretic and insulin resistance-improving agent |
| IL159320A0 (en) * | 2001-06-12 | 2004-06-01 | Wellstat Therapeutics Corp | Compounds for the treatment of metabolic disorders |
| US20050119314A1 (en) * | 2002-04-05 | 2005-06-02 | Sankyo Company, Limited | Pharmaceutical composition comprising an ACAT inhibitor and an insulin resistance reducing agent |
| KR20040099394A (ko) * | 2002-04-05 | 2004-11-26 | 상꾜 가부시키가이샤 | Acat 저해제 및 인슐린 저항성 개선제를 함유하는의약 조성물 |
-
2005
- 2005-03-25 KR KR1020067019743A patent/KR20070011329A/ko not_active Withdrawn
- 2005-03-25 BR BRPI0509305-8A patent/BRPI0509305A/pt not_active Application Discontinuation
- 2005-03-25 WO PCT/JP2005/005526 patent/WO2005092382A1/ja not_active Ceased
- 2005-03-25 EP EP05726976A patent/EP1731170A1/en not_active Withdrawn
- 2005-03-25 CA CA002560928A patent/CA2560928A1/en not_active Abandoned
- 2005-03-25 CN CNA2005800165817A patent/CN1972715A/zh active Pending
- 2005-03-28 TW TW094109508A patent/TW200536515A/zh unknown
-
2006
- 2006-09-22 US US11/525,481 patent/US20070049515A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| TW200536515A (en) | 2005-11-16 |
| CN1972715A (zh) | 2007-05-30 |
| US20070049515A1 (en) | 2007-03-01 |
| KR20070011329A (ko) | 2007-01-24 |
| EP1731170A1 (en) | 2006-12-13 |
| WO2005092382A1 (ja) | 2005-10-06 |
| CA2560928A1 (en) | 2005-10-06 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B11A | Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing | ||
| B11Y | Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette] |