BR9909796B1 - "derivados de piperidinopirimidina para aplicação tópica" - Google Patents

"derivados de piperidinopirimidina para aplicação tópica"

Info

Publication number: BR9909796B1
Authority: BR; Brazil
Prior art keywords: weight; piperidinopyrimidine; topical application; solvent; acceptable salt
Prior art date: 1998-04-22

Application number

BRPI9909796-6B1A

Other languages

English (en)

Other versions

BR9909796A (pt

Inventor

Tony Wai-Chiu So

Peter Paul Deo

Russell John Tait

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-04-22

Filing date

1999-04-20

Publication date

2013-10-29

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=3807366&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR9909796(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1999-04-20 Application filed filed Critical

2000-12-26 Publication of BR9909796A publication Critical patent/BR9909796A/pt

2013-10-29 Publication of BR9909796B1 publication Critical patent/BR9909796B1/pt

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/12—Carboxylic acids; Salts or anhydrides thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
- A61K8/494—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with more than one nitrogen as the only hetero atom
- A61K8/4953—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with more than one nitrogen as the only hetero atom containing pyrimidine ring derivatives, e.g. minoxidil
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0014—Skin, i.e. galenical aspects of topical compositions
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/04—Antipruritics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/14—Drugs for dermatological disorders for baldness or alopecia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q7/00—Preparations for affecting hair growth

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Chemical & Material Sciences (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Medicinal Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Dermatology (AREA)
Chemical Kinetics & Catalysis (AREA)
Oil, Petroleum & Natural Gas (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Birds (AREA)
Organic Chemistry (AREA)
Medicinal Preparation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Cosmetics (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Plural Heterocyclic Compounds (AREA)
Compositions Of Macromolecular Compounds (AREA)

BRPI9909796-6B1A 1998-04-22 1999-04-20 "derivados de piperidinopirimidina para aplicação tópica" BR9909796B1 (pt)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
AUPP3107A AUPP310798A0 (en)	1998-04-22	1998-04-22	Vehicle system for a composition comprising a piperidinopyrimidine derivative
PCT/AU1999/000294 WO1999053923A1 (en)	1998-04-22	1999-04-20	Pharmaceutical composition

Publications (2)

Publication Number	Publication Date
BR9909796A BR9909796A (pt)	2000-12-26
BR9909796B1 true BR9909796B1 (pt)	2013-10-29

Family

ID=3807366

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BRPI9909796-6B1A BR9909796B1 (pt)	1998-04-22	1999-04-20	"derivados de piperidinopirimidina para aplicação tópica"

Country Status (13)

Country	Link
US (2)	US6946120B2 (pt)
EP (2)	EP1695708B1 (pt)
JP (3)	JP3710380B2 (pt)
AT (1)	ATE331517T1 (pt)
AU (1)	AUPP310798A0 (pt)
BR (1)	BR9909796B1 (pt)
CA (1)	CA2328950C (pt)
CY (1)	CY1120513T1 (pt)
DE (1)	DE69932158T2 (pt)
DK (2)	DK1073439T3 (pt)
ES (2)	ES2665271T3 (pt)
PT (2)	PT1073439E (pt)
WO (1)	WO1999053923A1 (pt)

Families Citing this family (107)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9504265D0 (en)	1995-03-03	1995-04-19	Medeva Plc	Corticosteroid-containing pharmaceutical composition
AUPO983897A0 (en)	1997-10-17	1997-11-06	Soltec Research Pty Ltd	Topical antifungal composition
AUPP310798A0 (en) *	1998-04-22	1998-05-14	Soltec Research Pty Ltd	Vehicle system for a composition comprising a piperidinopyrimidine derivative
JPH11349451A (ja) *	1998-06-08	1999-12-21	Taisho Pharmaceut Co Ltd	育毛剤
US8263580B2 (en)	1998-09-11	2012-09-11	Stiefel Research Australia Pty Ltd	Vitamin formulation
US6342496B1 (en) *	1999-03-01	2002-01-29	Sepracor Inc.	Bupropion metabolites and methods of use
US20030108500A1 (en) *	2000-04-07	2003-06-12	Koji Imamura	Hair growth stimulant compositions
DE60114168T2 (de) *	2000-04-07	2006-07-13	Taisho Pharmaceutical Co., Ltd.	Haarwachstumstimulierende mittel mit verlängerter wirkung
JP4892786B2 (ja) *	2000-04-07	2012-03-07	大正製薬株式会社	持続性育毛製剤
US8512718B2 (en)	2000-07-03	2013-08-20	Foamix Ltd.	Pharmaceutical composition for topical application
US7442369B1 (en) *	2000-08-09	2008-10-28	Mcneil Ab	Compositions of minoxidil
AUPR048600A0 (en) *	2000-10-02	2000-10-26	Soltec Research Pty Ltd	Pharmaceutical vehicle
MXPA03010458A (es) *	2001-05-15	2004-03-09	Taisho Pharmaceuticals Co Ltd	Composicion liquida que contiene minoxidilo.
SE0104421D0 (sv) *	2001-12-21	2001-12-21	Ponsus Pharma Ab	New composition
IL152486A0 (en)	2002-10-25	2003-05-29	Meir Eini	Alcohol-free cosmetic and pharmaceutical foam carrier
US7704518B2 (en)	2003-08-04	2010-04-27	Foamix, Ltd.	Foamable vehicle and pharmaceutical compositions thereof
US10117812B2 (en)	2002-10-25	2018-11-06	Foamix Pharmaceuticals Ltd.	Foamable composition combining a polar solvent and a hydrophobic carrier
US8900554B2 (en)	2002-10-25	2014-12-02	Foamix Pharmaceuticals Ltd.	Foamable composition and uses thereof
US20080138296A1 (en)	2002-10-25	2008-06-12	Foamix Ltd.	Foam prepared from nanoemulsions and uses
US8119109B2 (en)	2002-10-25	2012-02-21	Foamix Ltd.	Foamable compositions, kits and methods for hyperhidrosis
US9265725B2 (en)	2002-10-25	2016-02-23	Foamix Pharmaceuticals Ltd.	Dicarboxylic acid foamable vehicle and pharmaceutical compositions thereof
US7700076B2 (en)	2002-10-25	2010-04-20	Foamix, Ltd.	Penetrating pharmaceutical foam
US8119150B2 (en)	2002-10-25	2012-02-21	Foamix Ltd.	Non-flammable insecticide composition and uses thereof
US9668972B2 (en)	2002-10-25	2017-06-06	Foamix Pharmaceuticals Ltd.	Nonsteroidal immunomodulating kit and composition and uses thereof
US7820145B2 (en)	2003-08-04	2010-10-26	Foamix Ltd.	Oleaginous pharmaceutical and cosmetic foam
US8486376B2 (en)	2002-10-25	2013-07-16	Foamix Ltd.	Moisturizing foam containing lanolin
US9211259B2 (en)	2002-11-29	2015-12-15	Foamix Pharmaceuticals Ltd.	Antibiotic kit and composition and uses thereof
JP2006505583A (ja)	2002-10-25	2006-02-16	フォーミックスエルティーディー．	化粧剤および医薬用フォーム
RS20050557A (sr)	2003-01-24	2007-09-21	Connetics Australia Pty Ltd.,	Klindamicin fosfat u obliku pene
US7575739B2 (en)	2003-04-28	2009-08-18	Foamix Ltd.	Foamable iodine composition
US7186416B2 (en)	2003-05-28	2007-03-06	Stiefel Laboratories, Inc.	Foamable pharmaceutical compositions and methods for treating a disorder
US8795693B2 (en)	2003-08-04	2014-08-05	Foamix Ltd.	Compositions with modulating agents
US8486374B2 (en)	2003-08-04	2013-07-16	Foamix Ltd.	Hydrophilic, non-aqueous pharmaceutical carriers and compositions and uses
BRPI0414883A (pt) *	2003-09-29	2006-12-12	Ethena Healthcare Inc	composição, concentrado de composição, e, composições alcoólicas desinfetante e semelhante a gel
GB0323908D0 (en) *	2003-10-11	2003-11-12	Nupharm Lab Ltd	Pharmaceutical foam formulation
WO2005067873A1 (en) *	2003-12-22	2005-07-28	Regrowth, Llc	Topical solutions comprising high concentrations of piperidinopyrimidine derivatives and methods of use thereof
US20050163811A1 (en) *	2004-01-23	2005-07-28	Richard Lee	Topical solutions comprising high concentrations of piperidinopyrimidine derivatives and methods of use thereof
US20060057075A1 (en) *	2004-08-02	2006-03-16	Moshe Arkin	Pharmaceutical and cosmeceutical wash-off mousse shampoo compositions, processes for preparing the same and uses thereof
US20060034779A1 (en) *	2004-08-02	2006-02-16	Agis Industries (1983) Ltd.	Foamable compositions containing vitamin D3 analogues, processes for preparing same and methods of treatment utilizng same
DE102004062775A1 (de)	2004-12-21	2006-06-29	Stockhausen Gmbh	Alkoholischer Pumpschaum
MX2007010893A (es)	2005-03-07	2008-02-25	Deb Worldwide Healthcare Inc	Composiciones espumantes de alto contenido de alcohol con agentes tensioactivos basados en silicon.
CA2609953A1 (en)	2005-05-09	2007-04-12	Foamix Ltd.	Saccharide foamable compositions
NZ563560A (en)	2005-06-01	2009-11-27	Stiefel Res Australia Pty Ltd	Vitamin formulation for treating a dermatological skin disorder
US8147815B2 (en) *	2005-12-16	2012-04-03	Celmatrix Corporation	Topical administration carrier composition and therapeutic formulations comprising same
CA2647127C (en)	2006-03-31	2015-10-06	Stiefel Research Australia Pty Ltd	Foamable suspension gel
US20080260655A1 (en)	2006-11-14	2008-10-23	Dov Tamarkin	Substantially non-aqueous foamable petrolatum based pharmaceutical and cosmetic compositions and their uses
KR100893469B1 (ko) *	2006-12-22	2009-04-17	씨제이제일제당 (주)	피부 투과성이 우수한 미녹시딜 함유 발모용 외용액제조성물
US8580860B2 (en) *	2007-02-23	2013-11-12	Gojo Industries, Inc.	Foamable alcoholic composition
US8021649B2 (en)	2007-02-22	2011-09-20	Cronk Peter J	Continuous spray scalp therapy and dispensing systems for same
US8636982B2 (en)	2007-08-07	2014-01-28	Foamix Ltd.	Wax foamable vehicle and pharmaceutical compositions thereof
WO2009069006A2 (en)	2007-11-30	2009-06-04	Foamix Ltd.	Foam containing benzoyl peroxide
WO2010041141A2 (en)	2008-10-07	2010-04-15	Foamix Ltd.	Oil-based foamable carriers and formulations
WO2009090495A2 (en)	2007-12-07	2009-07-23	Foamix Ltd.	Oil and liquid silicone foamable carriers and formulations
AU2009205314A1 (en)	2008-01-14	2009-07-23	Foamix Ltd.	Poloxamer foamable pharmaceutical compositions with active agents and/or therapeutic cells and uses
JP5420946B2 (ja) *	2009-03-23	2014-02-19	富士フイルム株式会社	胆汁酸を含むミノキシジル水性組成物
JP2010222317A (ja) *	2009-03-25	2010-10-07	Shiseido Co Ltd	水中油型乳化化粧料
WO2010125470A2 (en)	2009-04-28	2010-11-04	Foamix Ltd.	Foamable vehicle and pharmaceutical compositions comprising aprotic polar solvents and uses thereof
CA2769625C (en)	2009-07-29	2017-04-11	Foamix Ltd.	Non surfactant hydro-alcoholic foamable compositions, breakable foams and their uses
WO2011013008A2 (en)	2009-07-29	2011-02-03	Foamix Ltd.	Non surface active agent non polymeric agent hydro-alcoholic foamable compositions, breakable foams and their uses
JP5833007B2 (ja)	2009-08-31	2015-12-16	ドクター・レディーズ・ラボラトリーズ・リミテッド	ステロイドを含む局所製剤
US8945516B2 (en)	2009-10-02	2015-02-03	Foamix Pharmaceuticals Ltd.	Surfactant-free water-free foamable compositions, breakable foams and gels and their uses
US9849142B2 (en)	2009-10-02	2017-12-26	Foamix Pharmaceuticals Ltd.	Methods for accelerated return of skin integrity and for the treatment of impetigo
US20110189114A1 (en) *	2010-01-29	2011-08-04	Nyangenya Maniga	minoxidil composition and non-aerosol, non-spray foam method of delivery therefor
US9271917B2 (en)	2010-01-29	2016-03-01	Nyangenya Maniga	Method and apparatus for delivery of a measured dosage of a non-aerosol, non-spray foam composition of minoxidil
US20130324567A1 (en) *	2010-09-21	2013-12-05	Conrex Pharmaceutical Corporation	Restoration of hair
JP2014500275A (ja)	2010-12-06	2014-01-09	フォリカ，インコーポレイテッド	禿頭症を治療するため、および毛髪の成長を促進するための方法
US9717741B2 (en)	2012-10-11	2017-08-01	Anaplasi Pharmaceuticals Llc	Method and compositions for treating psoriasis
ES2924084T3 (es)	2012-10-11	2022-10-04	Chem Cure Ass Llc	Composición tópica para su uso en el tratamiento de la psoriasis
WO2014122436A1 (en)	2013-02-07	2014-08-14	Cipla House	Topical pharmaceutical compositions comprising minoxidil
US8642097B1 (en)	2013-03-19	2014-02-04	Nyangenya Maniga	Natural product energy drink and method of use thereof
WO2014184173A1 (en)	2013-05-14	2014-11-20	Montero Gida Sanayi Ve Ticaret A.S.	Hair care formulations
US20160184431A1 (en)	2014-03-11	2016-06-30	Promius Pharma Llc	Topical compositions comprising a corticosteroid
US9468606B2 (en)	2014-03-31	2016-10-18	Johnson & Johnson Consumer Inc.	Compostions and methods for enhancing the topical application of an acidic benefit agent
US9474699B2 (en)	2014-03-31	2016-10-25	Johnson & Johnson Consumer Inc.	Compostions and methods for enhancing the topical application of a basic benefit agent
CN106456467A (zh)	2014-06-16	2017-02-22	强生消费者公司	用于增强有色化妆品的局部施用的组合物和方法
US20150359742A1 (en)	2014-06-17	2015-12-17	Johnson & Johnson Consumer Inc.	Compositions and methods for enhancing the topical application of a benefit agent including powder to liquid particles and a second powder
US9675537B2 (en) *	2014-06-30	2017-06-13	Johnson & Johnson Consumer Inc.	Hair growth composition and method
JP7072346B2 (ja) *	2015-03-27	2022-05-20	大正製薬株式会社	ローション剤
WO2016159916A1 (en) *	2015-03-31	2016-10-06	Ogi̇g Sağlik Ürünleri̇ Ve Hi̇zmetleri̇ Sanayi̇ Ti̇caret Li̇mi̇ted Şi̇rketi̇	A foamy pharmaceutical formulation used in dermatological diseases
WO2016186896A1 (en) *	2015-05-18	2016-11-24	Thrower Angelo Perry	Hair regrowth treatment and growth stimulant
AU2016326143B2 (en)	2015-09-27	2021-05-27	Follica, Inc.	Needling device and drug applicator
EP3359198B1 (en)	2015-10-06	2020-05-13	Assos Ilaç Kimya Gida Ürünleri Üretim Ve Tic. A.S.	Topical minoxidil composition
US10561593B2 (en) *	2015-12-28	2020-02-18	Johnson & Johnson Consumer Inc.	Hair growth composition and method
CN105434352A (zh) *	2015-12-31	2016-03-30	浙江万晟药业有限公司	一种米诺地尔泡沫剂及其制备方法与应用
JP2018048104A (ja) *	2016-01-22	2018-03-29	大正製薬株式会社	外用組成物
JP2018048105A (ja) *	2016-01-22	2018-03-29	大正製薬株式会社	外用組成物
JP6848565B2 (ja) *	2016-03-30	2021-03-24	大正製薬株式会社	エアゾール剤
MX377365B (es)	2016-09-08	2025-03-10	Journey Medical Corp	Composiciones y métodos para tratar rosácea y acné.
US10736905B1 (en)	2016-09-09	2020-08-11	Shahin Fatholahi	Nefopam dosage forms and methods of treatment
JP7366515B2 (ja) *	2016-09-15	2023-10-23	大正製薬株式会社	外用組成物
US9962444B2 (en)	2016-09-27	2018-05-08	Shane Malek	Pharmacokinetically extended action topical hair growth formulation, and administration method
US10702495B2 (en)	2017-02-20	2020-07-07	Nexien Biopharma, Inc.	Method and compositions for treating dystrophies and myotonia
US10736874B1 (en)	2017-09-08	2020-08-11	Shahin Fatholahi	Methods for treating pain associated with sickle cell disease
US11446311B2 (en)	2017-09-08	2022-09-20	Shahin Fatholahi	Methods for treating pain associated with sickle cell disease
JP2019210268A (ja) *	2018-05-30	2019-12-12	ダイヤ製薬株式会社	外用剤及び外用剤の製造方法
WO2019232242A1 (en)	2018-05-30	2019-12-05	Follica, Inc.	Methods for promoting hair growth
WO2020206623A1 (en) *	2019-04-10	2020-10-15	Goldfinch Bio, Inc.	Crystal forms
US12409121B2 (en)	2019-05-06	2025-09-09	Spinart, LLC	Formulations and methods for preparing stable cosmetic compositions
EP3750528A1 (en)	2019-06-11	2020-12-16	Nexien Biopharma, Inc.	Compositions for treating dystrophies and myotonia
CN114025768B (zh)	2019-06-28	2023-12-22	古鲁生物制药有限公司	促进毛发生长的药品
EP3886799B1 (en)	2019-08-07	2023-11-15	Aneira Pharma, Inc.	Compositions for the treatment of hair loss
BR102021003531A2 (pt) *	2021-02-24	2022-08-30	Eurofarma Laboratorios S.A.	Composição farmacêutica tópica espumável
JP2025536556A (ja)	2022-10-25	2025-11-07	ヴェラダーミクスインコーポレイテッド	放出調節ミノキシジル用組成物および使用方法
TW202444338A (zh)	2023-04-07	2024-11-16	義大利商卡斯歐皮亞股份公司	克拉司酮與米諾地爾之組合療法
CN116919892B (zh) *	2023-08-03	2024-08-16	济南中海医药科技有限公司	一种米诺地尔外用溶液的制备方法
WO2025172818A1 (en) *	2024-02-14	2025-08-21	Cassiopea S.P.A.	Pyrilutamide combination therapy
CN118908900B (zh) *	2024-10-10	2025-01-28	山东则正医药技术有限公司	一种米诺地尔乳酸盐晶型及其制备方法和应用

Family Cites Families (69)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US515836A (en) *		1894-03-06		Basin-clamp
US4596812A (en) *	1976-05-24	1986-06-24	The Upjohn Company	Methods and solutions for treating male pattern alopecia
US4139619A (en) *	1976-05-24	1979-02-13	The Upjohn Company	6-Amino-4-(substituted amino)-1,2-dihydro-1-hydroxy-2-iminopyrimidine, topical compositions and process for hair growth
IT1066697B (it) *	1976-11-08	1985-03-12	Manetti & Roberts Italo Brit	Attivatore per composizioni cosmetiche e composizioni cosmetiche che lo contengono
US5183817A (en) *	1981-02-17	1993-02-02	Bazzano Gail S	Combinations of retinoids and minoxidil-type compounds for hair growth
EP0093770B1 (en) *	1981-11-09	1991-06-19	BAZZANO, Gail S	The use of retinoids and minoxidil (2,4-diamino-6-piperidino-pyrimidine-3-oxide) to increase the rate of growth of human scalp hair and to treat certain types of alopecias
WO1985001876A1 (en)	1983-10-24	1985-05-09	Lockley Services Pty. Ltd.	Foamable biocide composition
EP0190158A1 (en)	1984-06-21	1986-08-13	Soltec Research Pty. Ltd.	Aerosol product
JPS61197161A (ja)	1985-02-25	1986-09-01	Amada Co Ltd	ドレツシング装置
IT1201436B (it) *	1985-07-19	1989-02-02	Vincenzo Zappia	Formulazioni topiche a lento rilascio
US5041439A (en) *	1986-06-13	1991-08-20	The Procter & Gamble Company	Penetrating topical pharmaceutical compositions
DE3781034T2 (de) *	1986-06-13	1993-02-18	Procter & Gamble	Topische pharmazeutische zubereitung mit besserer durchdringungsfaehigkeit.
LU86548A1 (fr) *	1986-08-07	1988-03-02	Oreal	Composition sous forme de gel pour induire et stimuler la croissance des cheveux et diminuer leur chute a base de derives de piperidino-pyrimidine
AU7875487A (en) *	1986-08-08	1988-02-24	Upjohn Company, The	Methods, compositions and solutions for treating alopecia
AU8025787A (en)	1986-09-12	1988-04-07	Upjohn Company, The	Foams for delivery of minoxidil
JPS63150211A (ja)	1986-12-15	1988-06-22	Taisho Pharmaceut Co Ltd	ミノキシジル配合外用剤
AU618517B2 (en)	1986-12-23	1992-01-02	Eugene J. Van Scott	Additives enhancing topical actions of therapeutic agents
US5389677B1 (en)	1986-12-23	1997-07-15	Tristrata Inc	Method of treating wrinkles using glycalic acid
US4882182A (en)	1987-01-08	1989-11-21	Soltec Research Pty. Ltd.	Aerosol product
US4828837A (en) *	1987-03-30	1989-05-09	Liposome Technology, Inc.	Non-crystalline minoxidil composition, its production and application
US5030442A (en) *	1987-03-30	1991-07-09	Liposome Technology, Inc.	Non-crystalline minoxidil composition
JPH0745387B2 (ja)	1987-09-09	1995-05-17	株式会社資生堂	発毛、養毛促進剤
JP2810041B2 (ja)	1987-09-09	1998-10-15	株式会社資生堂	頭皮・頭髪用養毛料
JP2810040B2 (ja) *	1987-09-09	1998-10-15	株式会社資生堂	頭皮・頭髪用養毛料
KR910010018B1 (ko) *	1987-10-02	1991-12-10	가부시기가이샤 시세이도	양모제
US4866067A (en) *	1987-12-07	1989-09-12	Ricerche De Schiena s.n.c del Dr. Michele Giuseppe Di Schiena & C.	6-piperidino-2,4-diaminopyrimidine-3-oxide salt of 3-carboxypyridine n-oxide and topical, related compositions
US4888354A (en)	1987-12-21	1989-12-19	Theratech, Inc.	Skin penetration enhancement using free base and acid addition salt combinations of active agents
EP0417075B1 (en)	1988-02-18	1993-06-09	The Upjohn Company	Minoxidil gel
US5225189A (en) *	1988-02-18	1993-07-06	The Upjohn Company	Minoxidil gel
AU619256B2 (en)	1988-03-03	1992-01-23	Connetics Australia Pty Ltd	Acne treatment
LU87249A1 (fr) *	1988-06-17	1990-02-28	Oreal	Composition pour induire et stimuler la croissance des cheveux et/ou freiner leur chute,a base d'un agent tensio-actif amphotere et d'un derive de pyrimidine
US4938953A (en) *	1988-08-09	1990-07-03	The Upjohn Company	Self-preserving conditioning shampoo formulation
US5104646A (en) *	1989-08-07	1992-04-14	The Procter & Gamble Company	Vehicle systems for use in cosmetic compositions
AU646069B2 (en)	1990-08-10	1994-02-03	Pharmacia & Upjohn Company Llc	Stimulation of hair growth with potassium channel openers and 5alpha-reductase inhibitors
WO1992004419A1 (en)	1990-09-03	1992-03-19	Soltec Research Pty. Ltd.	A concentrated aerosol space spray
US5935554A (en)	1990-09-03	1999-08-10	Soltec Research Pty. Ltd.	Concentrated aerosol space spray that is not an emulsion
HUT66183A (en) *	1991-03-19	1994-10-28	Procter & Gamble	Multicomponent hair care compositions having -among others- plasticizing effect
ZA94170B (en)	1993-01-20	1995-03-15	Soltec Res Pty Ltd	Ectoparasiticidal formulation
JPH0748230A (ja) *	1993-07-31	1995-02-21	Hideo Horiuchi	育毛剤の製造法
FR2717683B1 (fr)	1994-03-22	1996-06-28	Fabre Pierre Cosmetique	Composition capillaire à base de minoxidil.
GB9504265D0 (en)	1995-03-03	1995-04-19	Medeva Plc	Corticosteroid-containing pharmaceutical composition
US5783202A (en)	1995-03-14	1998-07-21	Soltec Research Pty. Ltd.	Pediculicidal mousse composition for killing head lice
FR2736824B1 (fr) *	1995-07-18	1997-10-10	Fabre Pierre Dermo Cosmetique	Composition capillaire a base de minoxidil a faible teneur en solvant gras
JPH0971513A (ja)	1995-09-07	1997-03-18	Taisho Pharmaceut Co Ltd	育毛剤
JP3518096B2 (ja)	1995-09-29	2004-04-12	松下電器産業株式会社	映像記録再生機器の製造方法
US5834014A (en) *	1995-10-06	1998-11-10	The Regents Of The University Of Michigan	Stimulation of hair follicles
JP4467085B2 (ja) *	1996-01-05	2010-05-26	大正製薬株式会社	ヒノキチオール含有組成物
JPH09188629A (ja)	1996-01-06	1997-07-22	Pola Chem Ind Inc	抗体産生細胞抑制剤及びそれを含有する組成物
US5788155A (en)	1996-06-28	1998-08-04	S. C. Johnson & Son, Inc.	Air freshener dispenser device with dual cartridge capacity
US5838669A (en)	1996-08-28	1998-11-17	At&T Corp.	Method of synchronizing satellite switched CDMA communication system
JP3061575B2 (ja)	1996-10-17	2000-07-10	日立建機株式会社	孔掘削装置
AUPO379596A0 (en)	1996-11-22	1996-12-19	Soltec Research Pty Ltd	Percutaneous delivery system
JPH10158782A (ja)	1996-12-05	1998-06-16	Nkk Corp	フォトエッチング時の穿孔性とプレス成形性に優れたシャドウマスク用鋼板及びその製造方法
JPH10265343A (ja)	1997-01-23	1998-10-06	Taisho Pharmaceut Co Ltd	持効性育毛剤
US6255313B1 (en)	1997-01-23	2001-07-03	Taisho Pharmaceutical Co., Ltd.	Sustained release hair growth composition
JPH10279437A (ja) *	1997-03-31	1998-10-20	Shiseido Co Ltd	頭髪用化粧料
AUPO688997A0 (en)	1997-05-20	1997-06-12	Soltec Research Pty Ltd	Sunscreen composition
AUPO983897A0 (en)	1997-10-17	1997-11-06	Soltec Research Pty Ltd	Topical antifungal composition
US6231875B1 (en)	1998-03-31	2001-05-15	Johnson & Johnson Consumer Companies, Inc.	Acidified composition for topical treatment of nail and skin conditions
JPH11302131A (ja) *	1998-04-15	1999-11-02	Shiseido Co Ltd	頭皮頭髪用化粧料
AUPP310798A0 (en) *	1998-04-22	1998-05-14	Soltec Research Pty Ltd	Vehicle system for a composition comprising a piperidinopyrimidine derivative
JPH11349451A (ja)	1998-06-08	1999-12-21	Taisho Pharmaceut Co Ltd	育毛剤
US6284234B1 (en)	1998-08-04	2001-09-04	Johnson & Johnson Consumer Companies, Inc.	Topical delivery systems for active agents
AUPP583198A0 (en)	1998-09-11	1998-10-01	Soltec Research Pty Ltd	Mousse composition
US6383471B1 (en)	1999-04-06	2002-05-07	Lipocine, Inc.	Compositions and methods for improved delivery of ionizable hydrophobic therapeutic agents
AUPQ002999A0 (en)	1999-04-29	1999-05-20	Soltec Research Pty Ltd	Non-aqueous shampoo composition
US20030157046A1 (en) *	2000-04-07	2003-08-21	Koji Imamura	Minoxidil-containing preparations
JP4780429B2 (ja)	2000-04-07	2011-09-28	大正製薬株式会社	ミノキシジル含有製剤
US20030108500A1 (en)	2000-04-07	2003-06-12	Koji Imamura	Hair growth stimulant compositions

1998
- 1998-04-22 AU AUPP3107A patent/AUPP310798A0/en not_active Abandoned
1999
- 1999-04-20 DK DK99914373T patent/DK1073439T3/da active
- 1999-04-20 WO PCT/AU1999/000294 patent/WO1999053923A1/en not_active Ceased
- 1999-04-20 EP EP06012033.4A patent/EP1695708B1/en not_active Expired - Lifetime
- 1999-04-20 PT PT99914373T patent/PT1073439E/pt unknown
- 1999-04-20 CA CA002328950A patent/CA2328950C/en not_active Expired - Lifetime
- 1999-04-20 AT AT99914373T patent/ATE331517T1/de active
- 1999-04-20 JP JP2000544327A patent/JP3710380B2/ja not_active Expired - Lifetime
- 1999-04-20 BR BRPI9909796-6B1A patent/BR9909796B1/pt not_active IP Right Cessation
- 1999-04-20 DE DE69932158T patent/DE69932158T2/de not_active Expired - Lifetime
- 1999-04-20 DK DK06012033.4T patent/DK1695708T3/en active
- 1999-04-20 PT PT60120334T patent/PT1695708T/pt unknown
- 1999-04-20 EP EP99914373A patent/EP1073439B1/en not_active Expired - Lifetime
- 1999-04-20 ES ES06012033.4T patent/ES2665271T3/es not_active Expired - Lifetime
- 1999-04-20 ES ES99914373T patent/ES2268856T3/es not_active Expired - Lifetime
2002
- 2002-04-16 US US10/124,197 patent/US6946120B2/en not_active Expired - Lifetime
2003
- 2003-06-24 JP JP2003178898A patent/JP4338455B2/ja not_active Expired - Lifetime
2004
- 2004-09-10 US US10/949,116 patent/US20050037060A1/en not_active Abandoned
2007
- 2007-03-01 JP JP2007050885A patent/JP2007137899A/ja active Pending
2018
- 2018-05-18 CY CY20181100524T patent/CY1120513T1/el unknown

Also Published As

Publication number	Publication date
PT1695708T (pt)	2018-05-18
ATE331517T1 (de)	2006-07-15
EP1695708A3 (en)	2012-07-18
JP3710380B2 (ja)	2005-10-26
US20050037060A1 (en)	2005-02-17
ES2665271T3 (es)	2018-04-25
WO1999053923A1 (en)	1999-10-28
EP1695708A2 (en)	2006-08-30
DK1695708T3 (en)	2018-04-23
CA2328950A1 (en)	1999-10-28
DE69932158T2 (de)	2007-05-10
EP1073439A1 (en)	2001-02-07
CY1120513T1 (el)	2019-07-10
DE69932158D1 (de)	2006-08-10
JP4338455B2 (ja)	2009-10-07
ES2268856T3 (es)	2007-03-16
US6946120B2 (en)	2005-09-20
JP2004059587A (ja)	2004-02-26
JP2007137899A (ja)	2007-06-07
PT1073439E (pt)	2006-11-30
AUPP310798A0 (en)	1998-05-14
EP1073439B1 (en)	2006-06-28
US20020172649A1 (en)	2002-11-21
JP2002512192A (ja)	2002-04-23
CA2328950C (en)	2008-07-29
EP1073439A4 (en)	2003-07-02
EP1695708B1 (en)	2018-02-28
BR9909796A (pt)	2000-12-26
DK1073439T3 (da)	2006-10-23

Publication	Publication Date	Title
BR9909796B1 (pt)	2013-10-29	"derivados de piperidinopirimidina para aplicação tópica"
US5976566A (en)	1999-11-02	Non-steroidal antiinflammtory drug formulations for topical application to the skin
AU601423B2 (en)	1990-09-13	Dual phase solvent carrier system
DE60027463D1 (de)	2006-05-24	Pharmazeutische zusammensetzungen enthaltend resveratrol und verwendungen davon
CA2382886A1 (en)	2001-03-08	Benzamide formulation with histone deacetylase inhibitor activity
US4670254A (en)	1987-06-02	Gel preparations for topical application of diclofenac sodium
WO1999015210A3 (en)	1999-06-17	Bioadhesive compositions and methods for topical administration of active agents
AU2002361265A1 (en)	2003-07-09	Pharmaceutical composition for the treatment of psoriasis and other skin diseases
IE831611L (en)	1984-01-13	Topical anti-inflammatory compositions
NO863636L (no)	1987-03-13	Fremgangsmaate for fremstilling av transdermalt resorberbare preparater av arylpropionsyrederivater.
ATE321543T1 (de)	2006-04-15	Pharmazeutische zusammensetzungen mit hydroximsäurederivaten
MY101536A (en)	1991-11-30	Anti-inflammatory and analgesic tape for external use
CA2223918A1 (en)	1996-12-19	Pyrrole derivatives and medicinal composition
CA2360300A1 (en)	2000-08-17	A transdermal composition of an antivomiting agent and a preparation containing the same
AU3851399A (en)	1999-12-13	Minoxidil compositions for external use
KR880002524A (ko)	1988-05-09	니코란딜 외용제
CA2264693A1 (en)	1999-01-14	Azelastine hydrochloride-containing percutaneous preparation having good percutaneous absorbability and reduced skin irritation
GB1593097A (en)	1981-07-15	Pharmaceutical compositions containing a bischromone
AU714913B2 (en)	2000-01-13	Intranasal formulations for promoting sleep and method of using the same
JPS5750914A (en)	1982-03-25	Betamethasone external pharmaceutical
DE69720496D1 (en)	2003-05-08	Benzimidazolderivate
KR950703338A (ko)	1995-09-20	3-치환된 2-옥스인돌-1-카복스아미드 약학 조성물(3-substituted 2-oxindole-1-carboxamide pharmaceutical compositions)
IT1215340B (it)	1990-02-08	Derivati di esteri dell'acido immidazol-1-il-carbossilico, procedimenti per la loro preparazione e composizioni fungicide che contengono il derivato come componente attivo.
DK0452809T3 (da)	1994-09-05	Terapautisk middel til pollakisuri, urgeinkontinens eller urininkontinens omfattende alfa-phenyl-alfa-pyridylalkansyrederivater
EP1466909A4 (en)	2005-12-07	HALOGENBENZYLAMINOPROPIONSÄUREDERIVATE

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