BR9807278A - Composição farmacêutica para a liberação programada de dexfenfluramina - Google Patents
Composição farmacêutica para a liberação programada de dexfenfluraminaInfo
- Publication number
- BR9807278A BR9807278A BR9807278-1A BR9807278A BR9807278A BR 9807278 A BR9807278 A BR 9807278A BR 9807278 A BR9807278 A BR 9807278A BR 9807278 A BR9807278 A BR 9807278A
- Authority
- BR
- Brazil
- Prior art keywords
- dexfenfluramine
- pharmaceutical composition
- scheduled release
- release
- programmed release
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Emergency Medicine (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Patente de Invenção: <B>''COMPOSIçãO FARMACêUTICA PARA A LIBERAçãO PROGRAMADA DE DEXFENFLURAMINA''<D>. A invenção se refere a uma nova composição farmacêutica que permite a liberação programda de dexfenfluramina, caracterizada pelo fato de ela conter uma mistura de minigrânulos tais como definidos na descrição. Medicamentos.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9702446A FR2760190B1 (fr) | 1997-02-28 | 1997-02-28 | Composition pharmaceutique pour la liberation programmee de dexfenfluramine |
| PCT/FR1998/000377 WO1998037876A1 (fr) | 1997-02-28 | 1998-02-26 | Composition pharmaceutique pour la liberation programmee de dexfenfluramine |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR9807278A true BR9807278A (pt) | 2000-05-23 |
Family
ID=9504315
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR9807278-1A BR9807278A (pt) | 1997-02-28 | 1998-02-26 | Composição farmacêutica para a liberação programada de dexfenfluramina |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US5980952A (pt) |
| EP (1) | EP0975339A1 (pt) |
| JP (1) | JP2001513100A (pt) |
| CN (1) | CN1248913A (pt) |
| AU (1) | AU727614B2 (pt) |
| BR (1) | BR9807278A (pt) |
| CA (1) | CA2280980A1 (pt) |
| FR (1) | FR2760190B1 (pt) |
| HU (1) | HUP0001234A3 (pt) |
| NO (1) | NO994140L (pt) |
| NZ (1) | NZ337208A (pt) |
| PL (1) | PL335374A1 (pt) |
| WO (1) | WO1998037876A1 (pt) |
| ZA (1) | ZA981679B (pt) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2760190B1 (fr) * | 1997-02-28 | 1999-04-09 | Adir | Composition pharmaceutique pour la liberation programmee de dexfenfluramine |
| US7244765B2 (en) * | 2004-06-25 | 2007-07-17 | Cytokine Pharmasciences, Inc | Guanylhydrazone salts, compositions, processes of making and methods of using |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2738303A (en) * | 1952-07-18 | 1956-03-13 | Smith Kline French Lab | Sympathomimetic preparation |
| US3520975A (en) * | 1967-11-27 | 1970-07-21 | Robins Co Inc A H | Anorexigenic compositions comprising fenfluramine and scopolamine |
| FR2183546B1 (pt) * | 1972-05-10 | 1975-06-20 | Servier Lab | |
| US4309445A (en) * | 1980-06-16 | 1982-01-05 | Massachusetts Institute Of Technology | d-Fenfluramine for modifying feeding behavior |
| US4452815A (en) * | 1980-06-16 | 1984-06-05 | Massachusetts Institute Of Technology | Method of utilizing d,l-fenfluramine for modifying feeding behavior |
| US4728512A (en) * | 1985-05-06 | 1988-03-01 | American Home Products Corporation | Formulations providing three distinct releases |
| GB8519310D0 (en) * | 1985-07-31 | 1985-09-04 | Zyma Sa | Granular active substances |
| US4649161A (en) * | 1986-06-16 | 1987-03-10 | Massachusetts Institute Of Technology | Method for treating depression with d-fenfluramine |
| EP0308317A1 (fr) * | 1987-09-14 | 1989-03-22 | Sanofi | Composition anorexigène à mâcher et son procédé de préparation |
| US5258186A (en) * | 1989-03-10 | 1993-11-02 | Yamanouchi Pharmaceutical Co., Ltd. | Drug release controlling coating material for long acting formulations |
| US5133974A (en) * | 1989-05-05 | 1992-07-28 | Kv Pharmaceutical Company | Extended release pharmaceutical formulations |
| US5084287A (en) * | 1990-03-15 | 1992-01-28 | Warner-Lambert Company | Pharmaceutically useful micropellets with a drug-coated core and controlled-release polymeric coat |
| FR2663539B1 (fr) * | 1990-06-22 | 1994-10-07 | Adir | Utilisation de la d-fenfluramine pour l'obtention de medicaments destines au traitement des deficiences immunitaires chez le sujet age. |
| FR2677886B1 (fr) * | 1991-06-18 | 1995-03-31 | Adir | Comprime matriciel permettant la liberation prolongee d'indapamide apres administration par voie orale. |
| US5213811A (en) * | 1991-09-13 | 1993-05-25 | Sterling Drug Inc. | Oral sustained-release drug compositions |
| WO1994008709A1 (fr) * | 1992-10-09 | 1994-04-28 | Kanegafuchi Kagaku Kogyo Kabushiki Kaisha | Procede de production de granules fins |
| CA2158173C (en) * | 1993-03-17 | 2001-12-04 | Pietr Hitzig | Method of treating addictive behaviors |
| US5502080A (en) * | 1994-11-01 | 1996-03-26 | Hitzig; Pietr | Combined use of dopamine and serotonin agonists in the treatment of allergic disorders |
| FR2760190B1 (fr) * | 1997-02-28 | 1999-04-09 | Adir | Composition pharmaceutique pour la liberation programmee de dexfenfluramine |
-
1997
- 1997-02-28 FR FR9702446A patent/FR2760190B1/fr not_active Expired - Fee Related
-
1998
- 1998-02-17 US US09/024,364 patent/US5980952A/en not_active Expired - Fee Related
- 1998-02-26 CA CA002280980A patent/CA2280980A1/fr not_active Abandoned
- 1998-02-26 CN CN98802919A patent/CN1248913A/zh active Pending
- 1998-02-26 BR BR9807278-1A patent/BR9807278A/pt not_active IP Right Cessation
- 1998-02-26 HU HU0001234A patent/HUP0001234A3/hu unknown
- 1998-02-26 AU AU67346/98A patent/AU727614B2/en not_active Ceased
- 1998-02-26 NZ NZ337208A patent/NZ337208A/xx unknown
- 1998-02-26 EP EP98912553A patent/EP0975339A1/fr not_active Withdrawn
- 1998-02-26 JP JP53738198A patent/JP2001513100A/ja active Pending
- 1998-02-26 WO PCT/FR1998/000377 patent/WO1998037876A1/fr not_active Ceased
- 1998-02-26 PL PL98335374A patent/PL335374A1/xx unknown
- 1998-02-27 ZA ZA981679A patent/ZA981679B/xx unknown
-
1999
- 1999-08-26 NO NO994140A patent/NO994140L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| EP0975339A1 (fr) | 2000-02-02 |
| WO1998037876A1 (fr) | 1998-09-03 |
| AU6734698A (en) | 1998-09-18 |
| HUP0001234A2 (hu) | 2001-06-28 |
| NO994140D0 (no) | 1999-08-26 |
| NZ337208A (en) | 2000-08-25 |
| ZA981679B (en) | 1998-08-24 |
| NO994140L (no) | 1999-10-28 |
| FR2760190A1 (fr) | 1998-09-04 |
| AU727614B2 (en) | 2000-12-14 |
| US5980952A (en) | 1999-11-09 |
| HUP0001234A3 (en) | 2001-07-30 |
| PL335374A1 (en) | 2000-04-25 |
| CN1248913A (zh) | 2000-03-29 |
| JP2001513100A (ja) | 2001-08-28 |
| CA2280980A1 (fr) | 1998-09-03 |
| FR2760190B1 (fr) | 1999-04-09 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PC | Transfer |
Free format text: LES LABORATOIRES SERVIER (FR) |
|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 7A,8A E 9A ANUIDADES. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1887 DE 06/03/2007. |