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BR9608804A - Processos para sintetizar (1s,2r) indandiol para sintetizar (1s) amino (2r) indanol substancialmente isento de qualquer estereoisômero de bio-resolução para remover cis (1s,2r) indandiol de uma mistura de cis (1s,2r) indandiol e cis (1r,2s) indandiol e cultura pura - Google Patents

Processos para sintetizar (1s,2r) indandiol para sintetizar (1s) amino (2r) indanol substancialmente isento de qualquer estereoisômero de bio-resolução para remover cis (1s,2r) indandiol de uma mistura de cis (1s,2r) indandiol e cis (1r,2s) indandiol e cultura pura

Info

Publication number
BR9608804A
BR9608804A BR9608804A BR9608804A BR9608804A BR 9608804 A BR9608804 A BR 9608804A BR 9608804 A BR9608804 A BR 9608804A BR 9608804 A BR9608804 A BR 9608804A BR 9608804 A BR9608804 A BR 9608804A
Authority
BR
Brazil
Prior art keywords
indandiol
cis
stereoisomer
synthesize
bio
Prior art date
Application number
BR9608804A
Other languages
English (en)
Portuguese (pt)
Inventor
Neal C Connors
Francis P Gailliot
Barry C Buckland
Randolph L Greasham
Chris H Senanayake
Chanyong Lee
Rober C Olewinski Jr
F Edward Roberts
Paul J Reider
Michel M Chartrain
Thomas R Verhoeven
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9602938.4A external-priority patent/GB9602938D0/en
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of BR9608804A publication Critical patent/BR9608804A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C35/00Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C07C35/22Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring polycyclic, at least one hydroxy group bound to a condensed ring system
    • C07C35/23Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring polycyclic, at least one hydroxy group bound to a condensed ring system with hydroxy on a condensed ring system having two rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C215/00Compounds containing amino and hydroxy groups bound to the same carbon skeleton
    • C07C215/02Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C215/22Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated
    • C07C215/28Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings
    • C07C215/38Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings with rings other than six-membered aromatic rings being part of the carbon skeleton
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P41/00Processes using enzymes or microorganisms to separate optical isomers from a racemic mixture
    • C12P41/002Processes using enzymes or microorganisms to separate optical isomers from a racemic mixture by oxidation/reduction reactions
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P7/00Preparation of oxygen-containing organic compounds
    • C12P7/02Preparation of oxygen-containing organic compounds containing a hydroxy group
    • C12P7/22Preparation of oxygen-containing organic compounds containing a hydroxy group aromatic
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P7/00Preparation of oxygen-containing organic compounds
    • C12P7/24Preparation of oxygen-containing organic compounds containing a carbonyl group
    • C12P7/26Ketones

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Wood Science & Technology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Biotechnology (AREA)
  • Microbiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Analytical Chemistry (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
BR9608804A 1995-06-20 1996-06-14 Processos para sintetizar (1s,2r) indandiol para sintetizar (1s) amino (2r) indanol substancialmente isento de qualquer estereoisômero de bio-resolução para remover cis (1s,2r) indandiol de uma mistura de cis (1s,2r) indandiol e cis (1r,2s) indandiol e cultura pura BR9608804A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US36095P 1995-06-20 1995-06-20
GBGB9602938.4A GB9602938D0 (en) 1996-02-13 1996-02-13 Conversion of indene
PCT/US1996/010445 WO1997000966A1 (fr) 1995-06-20 1996-06-14 Conversion d'indene en (1s)-amino-(2r)-indanol depourvu de tout stereo-isomere, par combinaison de bioconversion de dioxygenase et d'etapes chimiques

Publications (1)

Publication Number Publication Date
BR9608804A true BR9608804A (pt) 1999-02-17

Family

ID=26308684

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9608804A BR9608804A (pt) 1995-06-20 1996-06-14 Processos para sintetizar (1s,2r) indandiol para sintetizar (1s) amino (2r) indanol substancialmente isento de qualquer estereoisômero de bio-resolução para remover cis (1s,2r) indandiol de uma mistura de cis (1s,2r) indandiol e cis (1r,2s) indandiol e cultura pura

Country Status (5)

Country Link
CN (1) CN1194006A (fr)
AR (1) AR002536A1 (fr)
AU (1) AU6180096A (fr)
BR (1) BR9608804A (fr)
WO (1) WO1997000966A1 (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9420067D0 (en) * 1994-10-05 1994-11-16 Zeneca Ltd Process
US5858737A (en) * 1995-06-20 1999-01-12 Merck & Co., Inc. Conversion of indene to (1S)-amino-(2R)-indanol free of any stereoisomer, by combination of dioxygenase bioconversion and chemical steps
US5824540A (en) * 1995-06-20 1998-10-20 Merck & Co., Inc. Pseudomonas putida strain with dioxygenase activity
EP0874059A4 (fr) * 1996-01-12 1999-10-27 Nippon Steel Chemical Co Procede de production de derives de l'indane
NL1005832C2 (nl) * 1997-04-17 1998-10-20 Dsm Nv Werkwijze voor de bereiding van CIS-(1S,2R)-aminoindanol.
GB2336841A (en) 1998-04-28 1999-11-03 Merck & Co Inc Preparation of cis-(is,2r)-indanediol by the microbial reduction of 1,2-indanedione
WO2000009659A1 (fr) * 1998-08-13 2000-02-24 Lonza Ag Procede pour la production de derives d'indane
NL1010354C2 (nl) * 1998-10-20 2000-04-25 Dsm Biotech Gmbh Bereiding van aminoalcoholen.
HRP20180282T1 (hr) * 2008-04-17 2018-03-23 Io Biotech Aps Imunoterapija na bazi indoleamin 2, 3-dioksigenaze

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5599985A (en) * 1993-09-14 1997-02-04 Sepracor, Inc. Optically pure 1-amido-2-indanols
US5420353A (en) * 1994-03-11 1995-05-30 Merck & Co., Inc. Regiospecific process to make cis-1-amino-2-alkanol from epoxide
GB9420067D0 (en) * 1994-10-05 1994-11-16 Zeneca Ltd Process

Also Published As

Publication number Publication date
AU6180096A (en) 1997-01-22
AR002536A1 (es) 1998-03-25
WO1997000966A1 (fr) 1997-01-09
CN1194006A (zh) 1998-09-23

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Legal Events

Date Code Title Description
EG Technical examination (opinion): publication of technical examination (opinion)
B09B Decision: refusal