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BR0011767A - ésteres de (-) -(1s,4r) n protegido 4-amino-2-ciclopenteno-1-carboxilato e respectivos processos de preparação - Google Patents

ésteres de (-) -(1s,4r) n protegido 4-amino-2-ciclopenteno-1-carboxilato e respectivos processos de preparação

Info

Publication number
BR0011767A
BR0011767A BR0011767-6A BR0011767A BR0011767A BR 0011767 A BR0011767 A BR 0011767A BR 0011767 A BR0011767 A BR 0011767A BR 0011767 A BR0011767 A BR 0011767A
Authority
BR
Brazil
Prior art keywords
cyclopentene
protected
amino
preparation processes
carboxylate esters
Prior art date
Application number
BR0011767-6A
Other languages
English (en)
Inventor
Max Rey
Gregor Welti
Cynthia Maryanoff
Original Assignee
Biocryst Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biocryst Pharm Inc filed Critical Biocryst Pharm Inc
Publication of BR0011767A publication Critical patent/BR0011767A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C269/04—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups from amines with formation of carbamate groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/46—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
    • C07C229/48—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups and carboxyl groups bound to carbon atoms of the same non-condensed ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/10—Systems containing only non-condensed rings with a five-membered ring the ring being unsaturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

"éSTERES DE (-)-(1S, 4R) N PROTEGIDO 4-AMINO-2-CICLOPENTENO-1-CARBOXILATO E RESPECTIVOS PROCESSOS DE PREPARAçãO". Resumo A invenção refere-se a um processo de preparação de ésteres de (-)-(1S, 4R) N protegido 4-amino-2-ciclopenteno-1-carboxilato representados pela fórmula (I) em que R^ 1^ e R^ 2^ são conforme descritos no Relatório Descritivo.
BR0011767-6A 1999-06-28 2000-06-09 ésteres de (-) -(1s,4r) n protegido 4-amino-2-ciclopenteno-1-carboxilato e respectivos processos de preparação BR0011767A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US14129299P 1999-06-28 1999-06-28
PCT/US2000/015969 WO2001001569A2 (en) 1999-06-28 2000-06-09 Process for preparing (-)-(1s,4r) n-protected 4-amino-2-cyclopentene-1-carboxylate esters

Publications (1)

Publication Number Publication Date
BR0011767A true BR0011767A (pt) 2002-04-23

Family

ID=22495050

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0011767-6A BR0011767A (pt) 1999-06-28 2000-06-09 ésteres de (-) -(1s,4r) n protegido 4-amino-2-ciclopenteno-1-carboxilato e respectivos processos de preparação

Country Status (16)

Country Link
US (1) US6495711B2 (pt)
EP (1) EP1206443A2 (pt)
JP (1) JP4532801B2 (pt)
KR (1) KR20020013937A (pt)
CN (1) CN1358170A (pt)
AR (1) AR024493A1 (pt)
AU (1) AU5479700A (pt)
BR (1) BR0011767A (pt)
CA (1) CA2377801A1 (pt)
CZ (1) CZ20014656A3 (pt)
HU (1) HUP0201873A3 (pt)
IL (1) IL147243A0 (pt)
NO (1) NO20016390L (pt)
PL (1) PL352675A1 (pt)
SK (1) SK19062001A3 (pt)
WO (1) WO2001001569A2 (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101538228B (zh) * 2008-03-21 2012-05-30 北京普世康医药技术有限公司 抗流感和禽流感病毒药物化合物帕拉米韦的合成方法
CN102863359B (zh) * 2012-05-16 2014-05-07 常州制药厂有限公司 一种抗流感药物的合成方法
US10385006B2 (en) * 2014-10-27 2019-08-20 Granules India Limited Process for the preparation of amino alcohol derivatives or salts thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8815265D0 (en) 1988-06-27 1988-08-03 Wellcome Found Therapeutic nucleosides
ATE118208T1 (de) 1989-10-16 1995-02-15 Chiroscience Ltd Chirale azabicycloheptanone und verfahren zu ihrer herstellung.
JPH06116217A (ja) * 1992-10-02 1994-04-26 Kuraray Co Ltd （±）−シス−４−アミノシクロペント−２−エンカルボン酸誘導体の光学分割法
US5399580A (en) * 1993-03-08 1995-03-21 Burroughs Wellcome Co. Therapeutic nucleosides-uses
CN1227466A (zh) 1996-06-14 1999-09-01 生物晶体药品股份有限公司 用作神经氨酸酶抑制剂的取代环戊烷化合物
GB9625455D0 (en) * 1996-12-07 1997-01-22 Glaxo Group Ltd Process for resolving mixtures of carbocyclic steroisomers
BR9813480A (pt) * 1997-12-17 2000-10-10 Biocryst Pharm Inc Compostos inibidores de neuraminidase de ciclopentano substituìdo, composição e métodos de inibição da neuraminidase do vìrus da influenza- e de tratamento de infecção por vìrus da influenza-

Also Published As

Publication number Publication date
AU5479700A (en) 2001-01-31
WO2001001569A2 (en) 2001-01-04
NO20016390D0 (no) 2001-12-27
JP2003503368A (ja) 2003-01-28
AR024493A1 (es) 2002-10-02
HUP0201873A3 (en) 2003-03-28
US20020052524A1 (en) 2002-05-02
IL147243A0 (en) 2002-08-14
WO2001001569A3 (en) 2001-05-03
SK19062001A3 (sk) 2003-03-04
PL352675A1 (en) 2003-09-08
KR20020013937A (ko) 2002-02-21
CN1358170A (zh) 2002-07-10
CA2377801A1 (en) 2001-01-04
EP1206443A2 (en) 2002-05-22
US6495711B2 (en) 2002-12-17
CZ20014656A3 (cs) 2002-11-13
HUP0201873A2 (en) 2002-10-28
NO20016390L (no) 2002-02-19
JP4532801B2 (ja) 2010-08-25

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Legal Events

Date Code Title Description
FA10 Dismissal: dismissal - article 33 of industrial property law
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]