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AU9102991A - 2,6-methano-2h-1-benzoxocincarboxamides as 5-ht3-antagonists - Google Patents

2,6-methano-2h-1-benzoxocincarboxamides as 5-ht3-antagonists

Info

Publication number
AU9102991A
AU9102991A AU91029/91A AU9102991A AU9102991A AU 9102991 A AU9102991 A AU 9102991A AU 91029/91 A AU91029/91 A AU 91029/91A AU 9102991 A AU9102991 A AU 9102991A AU 9102991 A AU9102991 A AU 9102991A
Authority
AU
Australia
Prior art keywords
benzoxocincarboxamides
methano
antagonists
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU91029/91A
Inventor
John E. Airey
Matthew R Powers
Walter Rodriguez
Raymond D. Youssefyeh
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Rhone Poulenc Rorer International Holdings Inc
Original Assignee
Rhone Poulenc Rorer International Holdings Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Rorer International Holdings Inc filed Critical Rhone Poulenc Rorer International Holdings Inc
Publication of AU9102991A publication Critical patent/AU9102991A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D313/00—Heterocyclic compounds containing rings of more than six members having one oxygen atom as the only ring hetero atom
    • C07D313/16—Eight-membered rings
    • C07D313/20—Eight-membered rings condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU91029/91A 1990-11-29 1991-11-22 2,6-methano-2h-1-benzoxocincarboxamides as 5-ht3-antagonists Abandoned AU9102991A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US62024190A 1990-11-29 1990-11-29
US620241 1996-03-22

Publications (1)

Publication Number Publication Date
AU9102991A true AU9102991A (en) 1992-06-25

Family

ID=24485149

Family Applications (1)

Application Number Title Priority Date Filing Date
AU91029/91A Abandoned AU9102991A (en) 1990-11-29 1991-11-22 2,6-methano-2h-1-benzoxocincarboxamides as 5-ht3-antagonists

Country Status (2)

Country Link
AU (1) AU9102991A (en)
WO (1) WO1992009284A1 (en)

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3869475A (en) * 1973-04-05 1975-03-04 Yissum Res Dev Co 2,6-methano-benzoxacin compounds
GB1579137A (en) * 1976-07-06 1980-11-12 Lilly Co Eli 5-isopropylidene-2,6-methano-3,4,5,6-tetrahydro-2h-1-benzoxocins
US4054583A (en) * 1976-07-06 1977-10-18 Eli Lilly And Company Process for converting 2,7-dihydroxy-5-isopropylidene-9-substituted-2,6-methano-3,4,5,6-tetrahydro-2H-1-benzoxocin to trans-1-hydroxy-3-substituted-6,6-dimethyl-6,6a,7,8,10,10a-hexahydro-9H-dibenzo(b,d)pyran-9-one
ES494130A0 (en) * 1979-08-09 1981-10-01 Glaxo Group Ltd A PROCEDURE FOR THE PREPARATION OF NEW BENZOXOCINE DERIVATIVES.
FR2531083B1 (en) * 1982-06-29 1986-11-28 Sandoz Sa NOVEL PIPERIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICINES
US4888353A (en) * 1986-02-28 1989-12-19 Erbamont, Inc. Carboxamides useful as antiemetic or antipsychotic agents
US4910193A (en) * 1985-12-16 1990-03-20 Sandoz Ltd. Treatment of gastrointestinal disorders
US4921982A (en) * 1988-07-21 1990-05-01 Eli Lilly And Company 5-halo-2,3-dihydro-2,2-dimethylbenzofuran-7-carboxylic acids useful as intermediates for 5-HT3 antagonists
JPH01168686A (en) * 1987-12-24 1989-07-04 Yoshitomi Pharmaceut Ind Ltd Benzofuran and benzopyran compounds
US4857517A (en) * 1988-02-04 1989-08-15 Rorer Pharmaceutical Corporation Quinuclidyl benzoxepins as 5-HT3 antagonists
US4924010A (en) * 1988-02-04 1990-05-08 Rorer Pharmaceutical Corporation Benzoxepins as intermediates to 5HT3 antagonists
US4859683A (en) * 1988-02-04 1989-08-22 Rorer Pharmaceutical Corporation Certain benzoxepins and their pharmaceutical compositions and methods
NZ227841A (en) * 1988-02-12 1991-08-27 Merck Sharp & Dohme Heterocyclic compounds with at least two non-condensed five membered rings and pharmaceutical compositions
US4863921A (en) * 1988-04-27 1989-09-05 Rorer Pharmaceutical Corporation Dibenzofurancarboxamides and their pharmaceutical compositions and methods
US4920227A (en) * 1988-11-29 1990-04-24 Rorer Pharmaceutical Corp. Benzobicyclic carboxamide 5-HT3 antagonists
US4920219A (en) * 1988-11-29 1990-04-24 Rorer Pharmaceutical Corp. Substituted saturated and unsaturated indole quinoline and benzazepine carboxamides and their use as pharmacological agents

Also Published As

Publication number Publication date
WO1992009284A1 (en) 1992-06-11

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