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AU6923998A - Quinoline-2(1h)-one and dihydroquinoline-2(1h)-one derivatives as ligands of 5-ht, 5-ht2 and 5-ht1-like receptors - Google Patents

Quinoline-2(1h)-one and dihydroquinoline-2(1h)-one derivatives as ligands of 5-ht, 5-ht2 and 5-ht1-like receptors

Info

Publication number
AU6923998A
AU6923998A AU69239/98A AU6923998A AU6923998A AU 6923998 A AU6923998 A AU 6923998A AU 69239/98 A AU69239/98 A AU 69239/98A AU 6923998 A AU6923998 A AU 6923998A AU 6923998 A AU6923998 A AU 6923998A
Authority
AU
Australia
Prior art keywords
dihydroquinoline
quinoline
ligands
receptors
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU69239/98A
Other languages
English (en)
Inventor
Caroline Cadilhac
Olivier Duclos
Eric Guilpain
Christian Hoornaert
Gary Mccort
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Synthelabo SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo SA filed Critical Synthelabo SA
Publication of AU6923998A publication Critical patent/AU6923998A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AU69239/98A 1997-03-20 1998-03-17 Quinoline-2(1h)-one and dihydroquinoline-2(1h)-one derivatives as ligands of 5-ht, 5-ht2 and 5-ht1-like receptors Abandoned AU6923998A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR9703387A FR2761071B1 (fr) 1997-03-20 1997-03-20 Derives de quinolein-2(1h)-one et de dihydroquinolein-2(1h)- one, leur preparation et leur application en therapeutique
FR9703387 1997-03-20
PCT/FR1998/000528 WO1998042712A1 (fr) 1997-03-20 1998-03-17 Derives de quinolein-2(1h)-one et de dihydroquinolein-2(1h)-one en tant que lingands des recepteurs 5-ht, 5-ht2 et 5-ht1-like

Publications (1)

Publication Number Publication Date
AU6923998A true AU6923998A (en) 1998-10-20

Family

ID=9504998

Family Applications (1)

Application Number Title Priority Date Filing Date
AU69239/98A Abandoned AU6923998A (en) 1997-03-20 1998-03-17 Quinoline-2(1h)-one and dihydroquinoline-2(1h)-one derivatives as ligands of 5-ht, 5-ht2 and 5-ht1-like receptors

Country Status (6)

Country Link
EP (1) EP0971928A1 (fr)
AR (1) AR012094A1 (fr)
AU (1) AU6923998A (fr)
FR (1) FR2761071B1 (fr)
WO (1) WO1998042712A1 (fr)
ZA (1) ZA982362B (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU748050B2 (en) * 1998-07-28 2002-05-30 3M Innovative Properties Company Oxazolo, thiazolo and selenazolo (4,5-C)-quinolin-4-amines and analogs thereof

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2797874B1 (fr) * 1999-08-27 2002-03-29 Adir Nouveaux derives de la pyridine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
MY127093A (en) † 2000-05-17 2006-11-30 Lucite Int Uk Ltd Bidentate ligands useful in catalyst systems
SE0004245D0 (sv) 2000-11-20 2000-11-20 Pharmacia Ab Novel compounds and their use
PL361690A1 (en) * 2000-11-20 2004-10-04 Biovitrum Ab Piperazinylpyrazine compounds as agonist or antagonist of serotonin 5ht-2 receptor
US7160888B2 (en) 2003-08-22 2007-01-09 Warner Lambert Company Llc [1,8]naphthyridin-2-ones and related compounds for the treatment of schizophrenia
JP4596792B2 (ja) * 2004-02-24 2010-12-15 あすか製薬株式会社 ５−ｈｔ１ａ作動作用と５−ｈｔ３拮抗作用を併有する薬剤
EP2094686A1 (fr) * 2006-09-26 2009-09-02 Glaxo Group Limited Derives de quinolinone 5-{2-[4-(2-methyl-5-quinolinyl)-l-piperidinyl]ethyl} utilises comme modulateurs du recepteur 5ht1a pour traiter les disfonctionnements sexuels, les anomalies cognitives, les troubles psychotiques, l'anxiete, la depression
ES2829973T3 (es) 2010-11-22 2021-06-02 Univ California Cromóforos semiconductores de moléculas pequeñas orgánicas para su uso en dispositivos electrónicos orgánicos
MA41168A (fr) * 2014-12-17 2017-10-24 Acraf Nouveaux composés antibactériens

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1278792C (fr) * 1985-05-06 1991-01-08 Joseph P. Yevich Derives antipsychotiques de pyridinylpiperazine a anneaux condenses
FR2637591B1 (fr) * 1988-10-11 1992-10-23 Synthelabo Derives de quinoleinone, leur preparation et leur application en therapeutique
FR2738823B1 (fr) * 1995-09-15 1997-10-31 Synthelabo Derives de 3-(omega-(4-(thieno(3,2-c)pyridin-4-yl)piperazin- 1-yl)alkyl)-3,4-dihydroquinolein-2(1h)-one,leur preparation et leur application en therapeutique
CO4750663A1 (es) * 1995-09-15 1999-03-31 Sanofi Synthelabo Derivados de quinolein-2 (1h)-ona, su preparacion y su aplicacion en terapeutica

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU748050B2 (en) * 1998-07-28 2002-05-30 3M Innovative Properties Company Oxazolo, thiazolo and selenazolo (4,5-C)-quinolin-4-amines and analogs thereof

Also Published As

Publication number Publication date
EP0971928A1 (fr) 2000-01-19
FR2761071A1 (fr) 1998-09-25
ZA982362B (en) 1998-09-23
WO1998042712A1 (fr) 1998-10-01
AR012094A1 (es) 2000-09-27
FR2761071B1 (fr) 1999-12-03

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