AU2018227575A1 - Processes for the preparation of fungicidal compounds - Google Patents
Processes for the preparation of fungicidal compounds Download PDFInfo
- Publication number
- AU2018227575A1 AU2018227575A1 AU2018227575A AU2018227575A AU2018227575A1 AU 2018227575 A1 AU2018227575 A1 AU 2018227575A1 AU 2018227575 A AU2018227575 A AU 2018227575A AU 2018227575 A AU2018227575 A AU 2018227575A AU 2018227575 A1 AU2018227575 A1 AU 2018227575A1
- Authority
- AU
- Australia
- Prior art keywords
- formula
- salt
- compound
- stereomerically enriched
- providing
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- 0 CC(C)*C(C(C)(C)N(C(c1c(N2C[C@@](c(cc(cc3)F)c3OC)OC*(C)C#N)[s]c(-[n]3nccn3)c1C)=O)C2=O)=O Chemical compound CC(C)*C(C(C)(C)N(C(c1c(N2C[C@@](c(cc(cc3)F)c3OC)OC*(C)C#N)[s]c(-[n]3nccn3)c1C)=O)C2=O)=O 0.000 description 19
- LFFZHZYJVDCJRT-UHFFFAOYSA-N CC(C(C)=O)N(C(c1c(N2CC(c3cc(F)ccc3OC)=O)[s]c(-[n]3nccn3)c1C)=O)C2=O Chemical compound CC(C(C)=O)N(C(c1c(N2CC(c3cc(F)ccc3OC)=O)[s]c(-[n]3nccn3)c1C)=O)C2=O LFFZHZYJVDCJRT-UHFFFAOYSA-N 0.000 description 1
- AZIQWVPYKCFWBQ-UHFFFAOYSA-N CC(C(O)=O)N(C(c1c(N2)[s]c(-[n]3nccn3)c1C)=O)C2=O Chemical compound CC(C(O)=O)N(C(c1c(N2)[s]c(-[n]3nccn3)c1C)=O)C2=O AZIQWVPYKCFWBQ-UHFFFAOYSA-N 0.000 description 1
- NDNHVVQZOQKDJS-UHFFFAOYSA-N CC(C)(C(NC(C=[IH])C=[IH])=O)N(C(c1c(N2CC(c3cc(F)ccc3OC)OCCC#N)[s]c(-[n]3nccn3)c1C)=O)C2=O Chemical compound CC(C)(C(NC(C=[IH])C=[IH])=O)N(C(c1c(N2CC(c3cc(F)ccc3OC)OCCC#N)[s]c(-[n]3nccn3)c1C)=O)C2=O NDNHVVQZOQKDJS-UHFFFAOYSA-N 0.000 description 1
- FACJOGDUGZPCCJ-UHFFFAOYSA-N CC(C)(C(O)=O)N(C(c1c(N2)[s]c(I)c1C)=O)C2=O Chemical compound CC(C)(C(O)=O)N(C(c1c(N2)[s]c(I)c1C)=O)C2=O FACJOGDUGZPCCJ-UHFFFAOYSA-N 0.000 description 1
- XRYQEFNDQSMPGO-UHFFFAOYSA-N CC(C)(C(O)=O)N(C(c1c(N2)[s]c(N3N=CCN3)c1C)=O)C2=O Chemical compound CC(C)(C(O)=O)N(C(c1c(N2)[s]c(N3N=CCN3)c1C)=O)C2=O XRYQEFNDQSMPGO-UHFFFAOYSA-N 0.000 description 1
- NLPQICGJPGCSQQ-UHFFFAOYSA-N CC(C)N(C)C(C(C)N(C(c1c(N2)[s]c(I)c1C)=O)C2=O)=O Chemical compound CC(C)N(C)C(C(C)N(C(c1c(N2)[s]c(I)c1C)=O)C2=O)=O NLPQICGJPGCSQQ-UHFFFAOYSA-N 0.000 description 1
- MKFLWZUFONEKCB-LYGOMILNSA-N CC(C)N(C)C(C(C)N(C(c1c(N2C[C@](C)(c3cc(F)ccc3OC)[O]=C)[s]c(C(O)=O)c1C)=O)C2=O)=O Chemical compound CC(C)N(C)C(C(C)N(C(c1c(N2C[C@](C)(c3cc(F)ccc3OC)[O]=C)[s]c(C(O)=O)c1C)=O)C2=O)=O MKFLWZUFONEKCB-LYGOMILNSA-N 0.000 description 1
- CLHYQNBLTGFTPS-UHFFFAOYSA-N CC(C)NC(C(C)(C)N(C(c1c(N2)[s]c(I)c1C)=O)C2=O)=O Chemical compound CC(C)NC(C(C)(C)N(C(c1c(N2)[s]c(I)c1C)=O)C2=O)=O CLHYQNBLTGFTPS-UHFFFAOYSA-N 0.000 description 1
- ZJKNEHOUUFJRPM-UHFFFAOYSA-N CC(C)NC(C(C)N(C(c1c(N2CC(c3cc(F)ccc3OC)=O)[s]c(I)c1C)=O)C2=O)=O Chemical compound CC(C)NC(C(C)N(C(c1c(N2CC(c3cc(F)ccc3OC)=O)[s]c(I)c1C)=O)C2=O)=O ZJKNEHOUUFJRPM-UHFFFAOYSA-N 0.000 description 1
- AZYULZZHGQAGMD-UHFFFAOYSA-O CC(C)[N](C)(C12[O](C)=C(c3c(N4)[s]c([NH2+]N=CC=N)c3C)N1C4=O)C2=O Chemical compound CC(C)[N](C)(C12[O](C)=C(c3c(N4)[s]c([NH2+]N=CC=N)c3C)N1C4=O)C2=O AZYULZZHGQAGMD-UHFFFAOYSA-O 0.000 description 1
- DFDOHEPVFHYOOE-UHFFFAOYSA-N CCNC(C(C)(C)N(C(c1c(N2CC(c3cc(F)ccc3OC)C#[O]CCC#N)[s]c(C(OCC)=O)c1C)=O)C2=O)=O Chemical compound CCNC(C(C)(C)N(C(c1c(N2CC(c3cc(F)ccc3OC)C#[O]CCC#N)[s]c(C(OCC)=O)c1C)=O)C2=O)=O DFDOHEPVFHYOOE-UHFFFAOYSA-N 0.000 description 1
- DZKUAHPABWCZEZ-LLVKDONJSA-N CCNC([C@@H](C)N(C(c1c(N2CC(c3cc(F)ccc3OC)=O)[s]c(I)c1C)=O)C2=O)=O Chemical compound CCNC([C@@H](C)N(C(c1c(N2CC(c3cc(F)ccc3OC)=O)[s]c(I)c1C)=O)C2=O)=O DZKUAHPABWCZEZ-LLVKDONJSA-N 0.000 description 1
- SMJNNMUTOGTWKC-JTSKRJEESA-N CCOC(c1c(C)c(C(N(C(C)(C)C(NC(C)C)=O)C(N2C[C@@H](c(cc(cc3)F)c3OC)OC[C@@H](C)C#N)=O)=O)c2[s]1)=O Chemical compound CCOC(c1c(C)c(C(N(C(C)(C)C(NC(C)C)=O)C(N2C[C@@H](c(cc(cc3)F)c3OC)OC[C@@H](C)C#N)=O)=O)c2[s]1)=O SMJNNMUTOGTWKC-JTSKRJEESA-N 0.000 description 1
- SMJNNMUTOGTWKC-UGNFMNBCSA-N CCOC(c1c(C)c(C(N(C(C)(C)C(NC(C)C)=O)C(N2C[C@@H](c3cc(F)ccc3OC)OCC(C)C#N)=O)=O)c2[s]1)=O Chemical compound CCOC(c1c(C)c(C(N(C(C)(C)C(NC(C)C)=O)C(N2C[C@@H](c3cc(F)ccc3OC)OCC(C)C#N)=O)=O)c2[s]1)=O SMJNNMUTOGTWKC-UGNFMNBCSA-N 0.000 description 1
- WELKXBYUTQSLCV-SFHVURJKSA-N CCOC(c1c(C)c(C(N(C(C)(C)C(OCC(C)C)=O)C(N2C[C@@H](c(cc(cc3)F)c3OC)O)=O)=O)c2[s]1)=O Chemical compound CCOC(c1c(C)c(C(N(C(C)(C)C(OCC(C)C)=O)C(N2C[C@@H](c(cc(cc3)F)c3OC)O)=O)=O)c2[s]1)=O WELKXBYUTQSLCV-SFHVURJKSA-N 0.000 description 1
- GTCLCPJNZBSUQB-UHFFFAOYSA-N CCOC(c1c(C)c(C(N(C(C)C(N(C)C(C)C)=O)C(N2CC(c3cc(F)ccc3OC)=O)=O)=O)c2[s]1)=O Chemical compound CCOC(c1c(C)c(C(N(C(C)C(N(C)C(C)C)=O)C(N2CC(c3cc(F)ccc3OC)=O)=O)=O)c2[s]1)=O GTCLCPJNZBSUQB-UHFFFAOYSA-N 0.000 description 1
- SCZHYCWCRLTUKZ-LBPRGKRZSA-N CC[C@@H](c(cc(cc1)F)c1OC)OCCC#N Chemical compound CC[C@@H](c(cc(cc1)F)c1OC)OCCC#N SCZHYCWCRLTUKZ-LBPRGKRZSA-N 0.000 description 1
- SBOAFGXPOKSPEE-UHFFFAOYSA-N CC[O](C)(C)C(c1c(N)[s]c(-[n]2nccc2)c1C)=O Chemical compound CC[O](C)(C)C(c1c(N)[s]c(-[n]2nccc2)c1C)=O SBOAFGXPOKSPEE-UHFFFAOYSA-N 0.000 description 1
- FVJHQFACCDCTEJ-UHFFFAOYSA-N CC[O](C)(C)C(c1c(NC(NC(C)(C)C(OC(C)(C)C)=O)=O)[s]c(-[n]2nccc2)c1C)=O Chemical compound CC[O](C)(C)C(c1c(NC(NC(C)(C)C(OC(C)(C)C)=O)=O)[s]c(-[n]2nccc2)c1C)=O FVJHQFACCDCTEJ-UHFFFAOYSA-N 0.000 description 1
- XFBIFOHVBKQIHN-UHFFFAOYSA-N CCc1c(-[n]2nccn2)[s]c(NC(N2C(C)C(NC(C)C)=O)=O)c1C2=O Chemical compound CCc1c(-[n]2nccn2)[s]c(NC(N2C(C)C(NC(C)C)=O)=O)c1C2=O XFBIFOHVBKQIHN-UHFFFAOYSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- G—PHYSICS
- G02—OPTICS
- G02B—OPTICAL ELEMENTS, SYSTEMS OR APPARATUS
- G02B6/00—Light guides; Structural details of arrangements comprising light guides and other optical elements, e.g. couplings
- G02B6/24—Coupling light guides
- G02B6/36—Mechanical coupling means
- G02B6/38—Mechanical coupling means having fibre to fibre mating means
- G02B6/3807—Dismountable connectors, i.e. comprising plugs
- G02B6/389—Dismountable connectors, i.e. comprising plugs characterised by the method of fastening connecting plugs and sockets, e.g. screw- or nut-lock, snap-in, bayonet type
- G02B6/3893—Push-pull type, e.g. snap-in, push-on
-
- G—PHYSICS
- G02—OPTICS
- G02B—OPTICAL ELEMENTS, SYSTEMS OR APPARATUS
- G02B6/00—Light guides; Structural details of arrangements comprising light guides and other optical elements, e.g. couplings
- G02B6/44—Mechanical structures for providing tensile strength and external protection for fibres, e.g. optical transmission cables
- G02B6/4439—Auxiliary devices
- G02B6/444—Systems or boxes with surplus lengths
- G02B6/4453—Cassettes
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Physics & Mathematics (AREA)
- General Physics & Mathematics (AREA)
- Optics & Photonics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Wood Science & Technology (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201762466944P | 2017-03-03 | 2017-03-03 | |
| US62/466,944 | 2017-03-03 | ||
| PCT/US2018/020728 WO2018161008A1 (fr) | 2017-03-03 | 2018-03-02 | Procédés de préparation de composés fongicides |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2018227575A1 true AU2018227575A1 (en) | 2019-09-19 |
Family
ID=61683933
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2018227575A Abandoned AU2018227575A1 (en) | 2017-03-03 | 2018-03-02 | Processes for the preparation of fungicidal compounds |
Country Status (11)
| Country | Link |
|---|---|
| EP (1) | EP3589635A1 (fr) |
| JP (1) | JP2020509038A (fr) |
| KR (1) | KR20190125359A (fr) |
| CN (1) | CN110382504A (fr) |
| AR (1) | AR111224A1 (fr) |
| AU (1) | AU2018227575A1 (fr) |
| BR (1) | BR112019017915A2 (fr) |
| CA (1) | CA3054810A1 (fr) |
| CO (1) | CO2019009579A2 (fr) |
| EA (1) | EA201991880A1 (fr) |
| WO (1) | WO2018161008A1 (fr) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2020509047A (ja) | 2017-03-03 | 2020-03-26 | ギリアード サイエンシーズ， インコーポレイテッド | Ａｃｃ阻害剤およびその固体形態を調製するためのプロセス |
| WO2020092239A1 (fr) * | 2018-10-29 | 2020-05-07 | Gilead Apollo, Llc | Procédés de préparation de composés fongicides |
| EP3669652A1 (fr) | 2018-12-21 | 2020-06-24 | Bayer AG | Combinaison de composés actifs |
| AR119594A1 (es) | 2019-08-09 | 2021-12-29 | Gilead Sciences Inc | Derivados de tienopirimidina como inhibidores acc y usos de los mismos |
| WO2021149771A1 (fr) * | 2020-01-22 | 2021-07-29 | 日産化学株式会社 | Composé thiénouracile et et agent de lutte contre les parasites |
| CN114539042A (zh) * | 2022-02-23 | 2022-05-27 | 河南旭瑞新材料科技有限公司 | 一种5-氟-2-羟基苯乙酮的合成新工艺 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2776038B1 (fr) * | 2011-11-11 | 2018-01-10 | Gilead Apollo, LLC | Inhibiteurs de l'acc et utilisations associées |
| AR106472A1 (es) * | 2015-10-26 | 2018-01-17 | Gilead Apollo Llc | Inhibidores de acc y usos de los mismos |
| WO2017091602A1 (fr) * | 2015-11-25 | 2017-06-01 | Gilead Apollo, Llc | Inhibiteurs de l'acc à base d'esters et utilisations associées |
| WO2017091627A1 (fr) | 2015-11-25 | 2017-06-01 | Gilead Apollo, Llc | Compositions fongicides contenant des dérivés de 2,4-dioxo-1,4-dihydrothiéno[2,3-d] pyrimidine |
| BR112018010113B1 (pt) * | 2015-11-25 | 2022-06-14 | Gilead Apollo, Llc | Composto de pirazol útil como inibidor da acetil-coa carboxilase (acc) |
| AU2016361428A1 (en) * | 2015-11-25 | 2018-05-24 | Gilead Apollo, Llc | Triazole ACC inhibitors and uses thereof |
-
2018
- 2018-03-02 CA CA3054810A patent/CA3054810A1/fr not_active Abandoned
- 2018-03-02 EA EA201991880A patent/EA201991880A1/ru unknown
- 2018-03-02 EP EP18711772.6A patent/EP3589635A1/fr not_active Withdrawn
- 2018-03-02 CN CN201880015391.0A patent/CN110382504A/zh active Pending
- 2018-03-02 BR BR112019017915-1A patent/BR112019017915A2/pt not_active IP Right Cessation
- 2018-03-02 WO PCT/US2018/020728 patent/WO2018161008A1/fr not_active Ceased
- 2018-03-02 KR KR1020197027893A patent/KR20190125359A/ko not_active Withdrawn
- 2018-03-02 AR ARP180100490A patent/AR111224A1/es unknown
- 2018-03-02 AU AU2018227575A patent/AU2018227575A1/en not_active Abandoned
- 2018-03-02 JP JP2019547390A patent/JP2020509038A/ja active Pending
-
2019
- 2019-09-03 CO CONC2019/0009579A patent/CO2019009579A2/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA3054810A1 (fr) | 2018-09-07 |
| EP3589635A1 (fr) | 2020-01-08 |
| AR111224A1 (es) | 2019-06-19 |
| BR112019017915A2 (pt) | 2020-05-12 |
| KR20190125359A (ko) | 2019-11-06 |
| CN110382504A (zh) | 2019-10-25 |
| CO2019009579A2 (es) | 2020-01-17 |
| WO2018161008A1 (fr) | 2018-09-07 |
| EA201991880A1 (ru) | 2020-02-25 |
| JP2020509038A (ja) | 2020-03-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK1 | Application lapsed section 142(2)(a) - no request for examination in relevant period |