AU2011345414A1 - Substituted methyl amines, serotonin 5-HT6 receptor antagonists, methods for the production and use thereof - Google Patents
Substituted methyl amines, serotonin 5-HT6 receptor antagonists, methods for the production and use thereofInfo
- Publication number
- AU2011345414A1 AU2011345414A1 AU2011345414A AU2011345414A AU2011345414A1 AU 2011345414 A1 AU2011345414 A1 AU 2011345414A1 AU 2011345414 A AU2011345414 A AU 2011345414A AU 2011345414 A AU2011345414 A AU 2011345414A AU 2011345414 A1 AU2011345414 A1 AU 2011345414A1
- Authority
- AU
- Australia
- Prior art keywords
- serotonin
- production
- methods
- receptor antagonists
- substituted methyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- QZAYGJVTTNCVMB-UHFFFAOYSA-N serotonin Chemical class C1=C(O)C=C2C(CCN)=CNC2=C1 QZAYGJVTTNCVMB-UHFFFAOYSA-N 0.000 title 2
- 108091005435 5-HT6 receptors Proteins 0.000 title 1
- 150000003956 methylamines Chemical class 0.000 title 1
- 239000002464 receptor antagonist Substances 0.000 title 1
- 229940044551 receptor antagonist Drugs 0.000 title 1
- 229940076279 serotonin Drugs 0.000 title 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| RU2010152052 | 2010-12-21 | ||
| RU2010152052/04A RU2443697C1 (en) | 2010-12-21 | 2010-12-21 | Substituted methyl-amines, serotonin 5-ht6 receptor antagonists, methods of production and use |
| PCT/RU2011/000981 WO2012087182A2 (en) | 2010-12-21 | 2011-12-13 | Substituted methyl amines, serotonin 5-ht6 receptor antagonists, methods for the production and use thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU2011345414A1 true AU2011345414A1 (en) | 2013-08-08 |
| AU2011345414B2 AU2011345414B2 (en) | 2016-12-01 |
Family
ID=45852279
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2011345414A Expired - Fee Related AU2011345414B2 (en) | 2010-12-21 | 2011-12-13 | Substituted methyl amines, serotonin 5-HT6 receptor antagonists, methods for the production and use thereof |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US8829002B2 (en) |
| EP (2) | EP3072882A1 (en) |
| JP (1) | JP6033788B2 (en) |
| KR (1) | KR20140023269A (en) |
| AU (1) | AU2011345414B2 (en) |
| CA (1) | CA2845524A1 (en) |
| EA (1) | EA201300663A1 (en) |
| RU (1) | RU2443697C1 (en) |
| WO (1) | WO2012087182A2 (en) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2500672C1 (en) * | 2012-10-25 | 2013-12-10 | Андрей Александрович Иващенко | (3-arylsulphonyl quinolin-8-yl-dialkyl-amines - selective serotonin 5-ht6 receptor antagonists, methods for production and use thereof |
| AR106515A1 (en) | 2015-10-29 | 2018-01-24 | Bayer Cropscience Ag | SILISPHENOXYHETEROCICLES, TRISUSTITUTED AND ANALOG |
| CN109134354B (en) * | 2018-09-19 | 2022-03-25 | 天津科技大学 | The synthetic method of 2-pyridyl methyl sulfide and the synthetic technique of related medicine |
| EP4045485A1 (en) | 2019-10-18 | 2022-08-24 | The Regents Of The University Of California | 3-phenylsulphonyl-quinoline derivatives as agents for treating pathogenic blood vessels disorders |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2538833B2 (en) | 1982-04-27 | 1986-04-25 | Roux Paul | UNDERGROUND LOCAL, SUCH AS A CELLAR, METHOD FOR FURNISHING SAME AND REMOVABLE ARMORING DEVICE USED FOR IMPLEMENTING SAID METHOD |
| DE69906397T2 (en) | 1998-01-16 | 2004-02-19 | F. Hoffmann-La Roche Ag | Benzosulfonderivate |
| US6194410B1 (en) | 1998-03-11 | 2001-02-27 | Hoffman-La Roche Inc. | Pyrazolopyrimidine and pyrazolines and process for preparation thereof |
| DE19858593A1 (en) | 1998-12-18 | 2000-06-21 | Merck Patent Gmbh | (2-Phenyl-4-(phenylsulfonyl)-oxazol-5-yl)-amine therapeutic agents having 5-HT6 receptor affinity, useful for treating CNS disorders such as psychosis, schizophrenia, depression or Alzheimer's disease |
| DE19956791A1 (en) * | 1999-11-25 | 2001-05-31 | Merck Patent Gmbh | New 2-heterocyclyl-4-arylsulfonyl-5-amino-oxazole derivatives useful in treatment of central nervous system disorders and as pesticides |
| US20040014966A1 (en) | 2000-06-20 | 2004-01-22 | Jacobsen Eric Jon | Bis-arylsulfones |
| US6586592B2 (en) * | 2000-06-20 | 2003-07-01 | Pharmacia & Upjohn Company | Bis-arylsulfones |
| PE20020063A1 (en) * | 2000-06-20 | 2002-01-30 | Upjohn Co | BIS-ARYLSULFONES AS LIGANDS OF THE 5-HT RECEPTOR |
| DE10129940A1 (en) * | 2001-06-13 | 2002-12-19 | Merck Patent Gmbh | Medicament used for treating central nervous system disorders e.g. psychosis, depression or neurological disorders, comprises new or known 4-phenylsulfonyl-oxazole-5-amine derivative which are serotonin 5-HT6 receptor ligands |
| EP1465872A1 (en) | 2001-12-28 | 2004-10-13 | Bayer Pharmaceuticals Corporation | 4-sulfide/sulfoxide/sulfonyl-1h-pyrazolyl derivative compounds, for use in diseases associated with the 5-ht2c receptor |
| BRPI0308696B8 (en) * | 2002-03-27 | 2021-05-25 | Axovant Sciences Gmbh | quinoline-derived compound, its preparation process, its pharmaceutical composition and its uses |
| GB0419192D0 (en) * | 2004-08-27 | 2004-09-29 | Merck Sharp & Dohme | Therapeutic agents |
| AU2008345225A1 (en) * | 2007-12-21 | 2009-07-09 | University Of Rochester | Method for altering the lifespan of eukaryotic organisms |
| EA017968B1 (en) * | 2008-01-24 | 2013-04-30 | Андрей Александрович ИВАЩЕНКО | SUBSTITUTED 2-AMINO-3-SULFONYLPYRAZOLO[1,5-a]PYRIMIDINES/ANTAGONISTS OF SEROTONIN 5-HTRECEPTORS, METHODS FOR THE PRODUCTION AND THE USE THEREOF |
| RU2393157C1 (en) * | 2008-10-06 | 2010-06-27 | Андрей Александрович Иващенко | 2-ALKYLAMINO-3-ARYLSULFONYL-PYRAZOLO[1,5-a]PYRIMIDINES, SEROTONIN 5-HT6 RECEPTOR ANTAGONISTS, METHODS OF PRODUCING AND USING SAID COMPOUNDS |
-
2010
- 2010-12-21 RU RU2010152052/04A patent/RU2443697C1/en not_active IP Right Cessation
-
2011
- 2011-12-13 EA EA201300663A patent/EA201300663A1/en unknown
- 2011-12-13 EP EP16000808.2A patent/EP3072882A1/en not_active Withdrawn
- 2011-12-13 WO PCT/RU2011/000981 patent/WO2012087182A2/en not_active Ceased
- 2011-12-13 EP EP11851231.8A patent/EP2657225A4/en not_active Withdrawn
- 2011-12-13 US US13/993,131 patent/US8829002B2/en not_active Expired - Fee Related
- 2011-12-13 KR KR1020137018965A patent/KR20140023269A/en not_active Withdrawn
- 2011-12-13 JP JP2013546064A patent/JP6033788B2/en not_active Expired - Fee Related
- 2011-12-13 CA CA2845524A patent/CA2845524A1/en not_active Abandoned
- 2011-12-13 AU AU2011345414A patent/AU2011345414B2/en not_active Expired - Fee Related
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