AU2003205747A1 - Thiazole derivatives and their use d2- and 5-ht1a-receptor ligands - Google Patents

Thiazole derivatives and their use d2- and 5-ht1a-receptor ligands

Info

Publication number: AU2003205747A1
Authority: AU; Australia
Prior art keywords: ht1a; receptor ligands; thiazole derivatives; thiazole; derivatives
Prior art date: 2002-03-06
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

AU2003205747A

Inventor

Gerd Bartoszyk

Henning Bottcher

Volker Eiermann

Joachim Marz

Christoph Seyfried

Christoph Van Amsterdam

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Merck Patent GmbH

Original Assignee

Merck Patent GmbH

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-03-06

Filing date

2003-02-07

Publication date

2003-09-16

2003-02-07 Application filed by Merck Patent GmbH filed Critical Merck Patent GmbH

2003-09-16 Publication of AU2003205747A1 publication Critical patent/AU2003205747A1/en

Status Abandoned legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Health & Medical Sciences (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Psychology (AREA)
Pain & Pain Management (AREA)
Psychiatry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

AU2003205747A 2002-03-06 2003-02-07 Thiazole derivatives and their use d2- and 5-ht1a-receptor ligands Abandoned AU2003205747A1 (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
EP02005013		2002-03-06
EP02005013.4		2002-03-06
PCT/EP2003/001247 WO2003074518A1 (en)	2002-03-06	2003-02-07	Thiazole derivatives and their use d2- and 5-ht1a-receptor ligands

Publications (1)

Publication Number	Publication Date
AU2003205747A1 true AU2003205747A1 (en)	2003-09-16

Family

ID=27771842

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AU2003205747A Abandoned AU2003205747A1 (en)	2002-03-06	2003-02-07	Thiazole derivatives and their use d2- and 5-ht1a-receptor ligands

Country Status (3)

Country	Link
AR (1)	AR038870A1 (en)
AU (1)	AU2003205747A1 (en)
WO (1)	WO2003074518A1 (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DK1408976T5 (en)	2001-07-20	2011-01-10	Psychogenics Inc	Treatment of Attention Deficit Hyperactivity Disorder (ADHD)
WO2023144764A1 (en)	2022-01-29	2023-08-03	Suven Life Sciences Limited	Benzoisothiazole and benzoisoxazole compounds for the treatment of mental disorders

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ZA954688B (en) *	1994-06-08	1996-01-29	Lundbeck & Co As H	Serotonin 5-HT1A and dopamin D2 receptor ligands
DE4425145A1 (en) *	1994-07-15	1996-01-18	Basf Ag	Use of thiazole and thiadiazole compounds
US6242448B1 (en) *	1998-12-17	2001-06-05	American Home Products Corporation	Trisubstituted-oxazole derivatives as serotonin ligands

2003
- 2003-02-07 WO PCT/EP2003/001247 patent/WO2003074518A1/en not_active Ceased
- 2003-02-07 AU AU2003205747A patent/AU2003205747A1/en not_active Abandoned
- 2003-03-05 AR ARP030100725A patent/AR038870A1/en not_active Application Discontinuation

Also Published As

Publication number	Publication date
WO2003074518A1 (en)	2003-09-12
AR038870A1 (en)	2005-02-02

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Legal Events

Date	Code	Title	Description
2004-11-25	MK6	Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase