AU2003290400A1 - A novel synthesis of 2-azabicyclic-3-carboxylic acids, useful as important drug intermediates - Google Patents
A novel synthesis of 2-azabicyclic-3-carboxylic acids, useful as important drug intermediatesInfo
- Publication number
- AU2003290400A1 AU2003290400A1 AU2003290400A AU2003290400A AU2003290400A1 AU 2003290400 A1 AU2003290400 A1 AU 2003290400A1 AU 2003290400 A AU2003290400 A AU 2003290400A AU 2003290400 A AU2003290400 A AU 2003290400A AU 2003290400 A1 AU2003290400 A1 AU 2003290400A1
- Authority
- AU
- Australia
- Prior art keywords
- azabicyclic
- useful
- carboxylic acids
- novel synthesis
- important drug
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- 230000015572 biosynthetic process Effects 0.000 title 1
- 239000003814 drug Substances 0.000 title 1
- 229940079593 drug Drugs 0.000 title 1
- 239000000543 intermediate Substances 0.000 title 1
- 238000003786 synthesis reaction Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/IN2003/000367 WO2005049567A1 (en) | 2003-11-24 | 2003-11-24 | A novel synthesis of 2-azabicyclic-3-carboxylic acids, useful as important drug intermediates |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2003290400A1 true AU2003290400A1 (en) | 2005-06-08 |
Family
ID=34611186
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2003290400A Abandoned AU2003290400A1 (en) | 2003-11-24 | 2003-11-24 | A novel synthesis of 2-azabicyclic-3-carboxylic acids, useful as important drug intermediates |
Country Status (3)
| Country | Link |
|---|---|
| EP (1) | EP1692106A1 (en) |
| AU (1) | AU2003290400A1 (en) |
| WO (1) | WO2005049567A1 (en) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN100376556C (en) * | 2005-10-14 | 2008-03-26 | 浙江工业大学 | Preparation method of 2-azabicyclo[3,3,0]octane-3-carboxylate hydrochloride |
| DE102005061756B4 (en) | 2005-12-21 | 2008-01-03 | Sanofi-Aventis Deutschland Gmbh | Improved process for the preparation of ramipril |
| EP2267144A3 (en) * | 2006-12-04 | 2011-05-25 | DSM IP Assets B.V. | Whole-cell catalytic system comprising a hydantoinase, a racemase and a carbamoylase |
| CN101827814B (en) | 2007-10-17 | 2012-11-28 | 中化帝斯曼制药有限公司荷兰公司 | Novel carbamoylglycine derivatives |
| WO2010049401A1 (en) * | 2008-10-30 | 2010-05-06 | Dsm Ip Assets B.V. | Method for the synthesis of a ramipril intermediate |
| CN106536541B (en) * | 2014-06-11 | 2021-01-08 | 赛诺菲-安万特德国有限公司 | Process for the preparation of ramipril |
| CN104817486B (en) * | 2015-03-31 | 2018-05-22 | 浙江工业大学 | A kind of synthetic method of ramipril intermediate |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3431541A1 (en) * | 1984-08-28 | 1986-03-06 | Hoechst Ag, 6230 Frankfurt | CIS, ENDO-2-AZABICYCLOALKAN-3-CARBONIC ACID DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, THEIR USE AND INTERMEDIATE PRODUCTS IN THEIR PRODUCTION |
-
2003
- 2003-11-24 EP EP03782763A patent/EP1692106A1/en not_active Withdrawn
- 2003-11-24 AU AU2003290400A patent/AU2003290400A1/en not_active Abandoned
- 2003-11-24 WO PCT/IN2003/000367 patent/WO2005049567A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO2005049567A1 (en) | 2005-06-02 |
| EP1692106A1 (en) | 2006-08-23 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK6 | Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase |