AU2003275093A1 - Process of making phenylpyrazoles useful as selective 5ht2a modulators and intermediates thereof - Google Patents
Process of making phenylpyrazoles useful as selective 5ht2a modulators and intermediates thereofInfo
- Publication number
- AU2003275093A1 AU2003275093A1 AU2003275093A AU2003275093A AU2003275093A1 AU 2003275093 A1 AU2003275093 A1 AU 2003275093A1 AU 2003275093 A AU2003275093 A AU 2003275093A AU 2003275093 A AU2003275093 A AU 2003275093A AU 2003275093 A1 AU2003275093 A1 AU 2003275093A1
- Authority
- AU
- Australia
- Prior art keywords
- phenylpyrazoles
- modulators
- intermediates
- useful
- making
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- 239000000543 intermediate Substances 0.000 title 1
- 150000008048 phenylpyrazoles Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/16—Halogen atoms or nitro radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US41329902P | 2002-09-24 | 2002-09-24 | |
| US60/413,299 | 2002-09-24 | ||
| PCT/US2003/029736 WO2004028450A2 (en) | 2002-09-24 | 2003-09-22 | Process of making phenylpyrazoles useful as selective 5ht2a modulators and intermediates thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU2003275093A1 true AU2003275093A1 (en) | 2004-04-19 |
| AU2003275093A8 AU2003275093A8 (en) | 2004-04-19 |
Family
ID=32043230
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2003275093A Abandoned AU2003275093A1 (en) | 2002-09-24 | 2003-09-22 | Process of making phenylpyrazoles useful as selective 5ht2a modulators and intermediates thereof |
Country Status (2)
| Country | Link |
|---|---|
| AU (1) | AU2003275093A1 (en) |
| WO (1) | WO2004028450A2 (en) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MXPA06000795A (en) | 2003-07-22 | 2006-08-23 | Arena Pharm Inc | Diaryl and arylheteroaryl urea derivatives as modulators of the 5-ht2a serotonin receptor useful for the prophylaxis and treatment of disorders related therto. |
| EP1727803B3 (en) | 2004-03-23 | 2014-04-23 | Arena Pharmaceuticals, Inc. | Processes for preparing substituted n-aryl-n'-[3-(1h-pyrazol-5-yl)phenyl] ureas and intermediates thereof |
| PE20061130A1 (en) | 2004-11-19 | 2007-01-05 | Arena Pharm Inc | 3-PHENYL-PIRAZOLE DERIVATIVES AS MODULATORS OF THE SEROTONIN 5-HT2A RECEPTOR |
| AR052886A1 (en) * | 2005-01-26 | 2007-04-11 | Arena Pharm Inc | PROCEDURES TO PREPARE PHENYLPIRAZOL REPLACED UREAS AND TO OBTAIN YOUR SYNTHESIS INTERMEDIARIES |
| JP5389642B2 (en) | 2006-05-18 | 2014-01-15 | アリーナ ファーマシューティカルズ， インコーポレイテッド | 3-pyrazolyl-benzamido-4-ethers, secondary amines and derivatives thereof as modulators of 5-HT2A serotonin receptors useful for the treatment of disorders associated with 5-HT2A serotonin receptors |
| ES2543718T3 (en) | 2006-05-18 | 2015-08-21 | Arena Pharmaceuticals, Inc. | Crystalline forms and processes for the preparation of phenyl-pyrazoles useful as modulators of the serotonin 5-HT2A receptor |
| ES2536762T3 (en) | 2006-05-18 | 2015-05-28 | Arena Pharmaceuticals, Inc. | Primary amines and their derivatives as 5-HT2A serotonin receptor modulators useful for the treatment of disorders related to this |
| TWI415845B (en) | 2006-10-03 | 2013-11-21 | Arena Pharm Inc | Pyrazole derivatives as modulators of the 5-ht2a serotonin receptor useful for the treatment of disorders related thereto |
| ES2421237T7 (en) | 2007-08-15 | 2013-09-30 | Arena Pharmaceuticals, Inc. | Imidazo [1,2-a] pyridine derivatives as modulators of the serotonergic 5ht2a receptor in the treatment of disorders related thereto |
| US20110021538A1 (en) | 2008-04-02 | 2011-01-27 | Arena Pharmaceuticals, Inc. | Processes for the preparation of pyrazole derivatives useful as modulators of the 5-ht2a serotonin receptor |
| WO2010062321A1 (en) | 2008-10-28 | 2010-06-03 | Arena Pharmaceuticals, Inc. | Processes useful for the preparation of 1-[3-(4-bromo-2-methyl-2h-pyrazol-3-yl)-4-methoxy-phenyl]-3-(2,4-difluoro-phenyl)-urea and crystalline forms related thereto |
| PT2364142T (en) | 2008-10-28 | 2018-04-23 | Arena Pharm Inc | Compositions of a 5-ht2a serotonin receptor modulator useful for the treatment of disorders related thereto |
| US8980891B2 (en) | 2009-12-18 | 2015-03-17 | Arena Pharmaceuticals, Inc. | Crystalline forms of certain 3-phenyl-pyrazole derivatives as modulators of the 5-HT2A serotonin receptor useful for the treatment of disorders related thereto |
| MX388281B (en) | 2015-06-12 | 2025-03-11 | Axovant Sciences Gmbh | Diaryl and arylheteroaryl urea derivatives useful for the prophylaxis and treatment of rem sleep behavior disorder |
| HK1247555A1 (en) | 2015-07-15 | 2018-09-28 | Axovant Sciences Gmbh | Diaryl and arylheteroaryl urea derivatives as modulators of the 5-ht2a serotonin receptor useful for the prophylaxis and treatment of hallucinations associated with a neurodegenerative disease |
| EP4631938A1 (en) | 2022-12-08 | 2025-10-15 | Shionogi & Co., Ltd | Nitrogen-containing heterocycle with serotonin receptor-binding activity and carbocyclic derivative |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2682379B1 (en) * | 1991-10-09 | 1994-02-11 | Rhone Poulenc Agrochimie | NEW FUNGICIDAL PHENYLPYRAZOLES. |
-
2003
- 2003-09-22 AU AU2003275093A patent/AU2003275093A1/en not_active Abandoned
- 2003-09-22 WO PCT/US2003/029736 patent/WO2004028450A2/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO2004028450A3 (en) | 2004-10-07 |
| WO2004028450A2 (en) | 2004-04-08 |
| AU2003275093A8 (en) | 2004-04-19 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK6 | Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase |