AU2002356369A1 - Xanthine derivatives as muscarinic receptor antagonists - Google Patents
Xanthine derivatives as muscarinic receptor antagonistsInfo
- Publication number
- AU2002356369A1 AU2002356369A1 AU2002356369A AU2002356369A AU2002356369A1 AU 2002356369 A1 AU2002356369 A1 AU 2002356369A1 AU 2002356369 A AU2002356369 A AU 2002356369A AU 2002356369 A AU2002356369 A AU 2002356369A AU 2002356369 A1 AU2002356369 A1 AU 2002356369A1
- Authority
- AU
- Australia
- Prior art keywords
- receptor antagonists
- muscarinic receptor
- xanthine derivatives
- xanthine
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- LRFVTYWOQMYALW-UHFFFAOYSA-N 9H-xanthine Chemical class O=C1NC(=O)NC2=C1NC=N2 LRFVTYWOQMYALW-UHFFFAOYSA-N 0.000 title 1
- 229940121948 Muscarinic receptor antagonist Drugs 0.000 title 1
- 229940083747 low-ceiling diuretics xanthine derivative Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pulmonology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/IB2002/005589 WO2004056810A1 (fr) | 2002-12-23 | 2002-12-23 | Derives de xanthine utilise en tant qu'antagonistes des recepteurs muscariniques |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2002356369A1 true AU2002356369A1 (en) | 2004-07-14 |
Family
ID=32676694
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2002356369A Abandoned AU2002356369A1 (en) | 2002-12-23 | 2002-12-23 | Xanthine derivatives as muscarinic receptor antagonists |
Country Status (4)
| Country | Link |
|---|---|
| EP (1) | EP1590345A1 (fr) |
| AU (1) | AU2002356369A1 (fr) |
| CA (1) | CA2511726A1 (fr) |
| WO (1) | WO2004056810A1 (fr) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE419236T1 (de) | 2002-07-08 | 2009-01-15 | Ranbaxy Lab Ltd | 3,6-disubstituierte azabicyclo-3.1.0 hexan- derivate als muscarinische rezeptorantagonisten |
| EP1618091A1 (fr) | 2003-04-09 | 2006-01-25 | Ranbaxy Laboratories, Ltd. | Derives d'azabicyclo hexane substitues en tant qu'antagonistes de recepteurs muscariniques |
| EP1626957A1 (fr) | 2003-04-11 | 2006-02-22 | Ranbaxy Laboratories Limited | Derives azabicyclo utiles comme antagonistes du recepteur muscarinique |
| DE602004018844D1 (de) * | 2004-06-16 | 2009-02-12 | Ranbaxy Lab Ltd | Als antagonisten des muscarinrezeptors geeignete xanthinderivate |
| EP1934184A1 (fr) | 2005-10-05 | 2008-06-25 | Ranbaxy Laboratories, Ltd. | Dérivés de 3 -azabicyclooctane en tant qu antagonistes de récepteurs muscariniques |
| WO2007110782A1 (fr) | 2005-12-30 | 2007-10-04 | Ranbaxy Laboratories Limited | Antagonistes des récepteurs muscariniques |
| BRPI0620844A2 (pt) | 2005-12-30 | 2011-11-29 | Ranbaxy Lab Ltd | compostos antagonistas dos receptores muscarìnicos, seus métodos de preparação, composições farmacêuticas compreendendo os mesmos, usos dos referidos compostos na preparação de medicamentos |
| US8202891B2 (en) | 2007-04-24 | 2012-06-19 | Theravance, Inc. | Quaternary ammonium compounds useful as muscarinic receptor antagonists |
| US20090326004A1 (en) | 2008-06-03 | 2009-12-31 | Ranbaxy Laboratories Limited | Muscarinic receptor antagonists |
| US9133116B2 (en) | 2010-09-28 | 2015-09-15 | Panacea Biotec Ltd. | Bicyclic compounds |
| WO2020243423A1 (fr) | 2019-05-31 | 2020-12-03 | Ikena Oncology, Inc. | Inhibiteurs de tead et leurs utilisations |
| CA3142351A1 (fr) | 2019-05-31 | 2020-12-03 | Ikena Oncology, Inc. | Inhibiteurs de tead et leurs utilisations |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT8721978A0 (it) * | 1987-09-21 | 1987-09-21 | Angeli Inst Spa | Nuovi derivati ammidinici triciclici. |
| US5889006A (en) * | 1995-02-23 | 1999-03-30 | Schering Corporation | Muscarinic antagonists |
| ES2165768B1 (es) * | 1999-07-14 | 2003-04-01 | Almirall Prodesfarma Sa | Nuevos derivados de quinuclidina y composiciones farmaceuticas que los contienen. |
-
2002
- 2002-12-23 WO PCT/IB2002/005589 patent/WO2004056810A1/fr not_active Ceased
- 2002-12-23 CA CA002511726A patent/CA2511726A1/fr not_active Abandoned
- 2002-12-23 EP EP02808274A patent/EP1590345A1/fr not_active Withdrawn
- 2002-12-23 AU AU2002356369A patent/AU2002356369A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CA2511726A1 (fr) | 2004-07-08 |
| EP1590345A1 (fr) | 2005-11-02 |
| WO2004056810A1 (fr) | 2004-07-08 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK6 | Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase |