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AU2001289675A1 - Novel Heteroaryl Derivatives and the Use Thereof as Pharmaceuticals - Google Patents

Novel Heteroaryl Derivatives and the Use Thereof as Pharmaceuticals

Info

Publication number
AU2001289675A1
AU2001289675A1 AU2001289675A AU2001289675A AU2001289675A1 AU 2001289675 A1 AU2001289675 A1 AU 2001289675A1 AU 2001289675 A AU2001289675 A AU 2001289675A AU 2001289675 A AU2001289675 A AU 2001289675A AU 2001289675 A1 AU2001289675 A1 AU 2001289675A1
Authority
AU
Australia
Prior art keywords
pharmaceuticals
heteroaryl derivatives
novel heteroaryl
novel
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU2001289675A
Other versions
AU2001289675B2 (en
Inventor
Beate Aue
Silke Baasner
Gerald Bacher
Thomas Beckers
Peter Emig
Eckhard Gunther
Bernd Nickel
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aeterna Zentaris GmbH
Original Assignee
Zentaris AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE10035927A external-priority patent/DE10035927A1/en
Application filed by Zentaris AG filed Critical Zentaris AG
Publication of AU2001289675A1 publication Critical patent/AU2001289675A1/en
Assigned to ZENTARIS GMBH reassignment ZENTARIS GMBH Request for Assignment Assignors: ZENTARIS AG
Application granted granted Critical
Publication of AU2001289675B2 publication Critical patent/AU2001289675B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

AU2001289675A 2000-07-21 2001-07-18 Novel heteroaryl derivatives and the use thereof as pharmaceuticals Ceased AU2001289675B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10035927A DE10035927A1 (en) 2000-07-21 2000-07-21 New heteroaryl derivatives and their use as medicines
DE10035927.2 2000-07-21
PCT/EP2001/008263 WO2002008194A1 (en) 2000-07-21 2001-07-18 Novel heteroaryl derivatives and the use thereof as pharmaceuticals

Publications (2)

Publication Number Publication Date
AU2001289675A1 true AU2001289675A1 (en) 2002-05-02
AU2001289675B2 AU2001289675B2 (en) 2005-04-07

Family

ID=7649979

Family Applications (2)

Application Number Title Priority Date Filing Date
AU2001289675A Ceased AU2001289675B2 (en) 2000-07-21 2001-07-18 Novel heteroaryl derivatives and the use thereof as pharmaceuticals
AU8967501A Pending AU8967501A (en) 2000-07-21 2001-07-18 Novel heteroaryl derivatives and the use thereof as pharmaceuticals

Family Applications After (1)

Application Number Title Priority Date Filing Date
AU8967501A Pending AU8967501A (en) 2000-07-21 2001-07-18 Novel heteroaryl derivatives and the use thereof as pharmaceuticals

Country Status (28)

Country Link
US (1) US6706722B2 (en)
EP (1) EP1301485B1 (en)
JP (1) JP2004504382A (en)
KR (1) KR20030022296A (en)
CN (1) CN1296359C (en)
AR (1) AR033383A1 (en)
AT (1) ATE365717T1 (en)
AU (2) AU2001289675B2 (en)
BG (1) BG107507A (en)
BR (1) BR0112591A (en)
CA (1) CA2353360A1 (en)
CY (1) CY1106890T1 (en)
CZ (1) CZ2003427A3 (en)
DE (2) DE10035927A1 (en)
DK (1) DK1301485T3 (en)
ES (1) ES2291349T3 (en)
HU (1) HUP0303729A3 (en)
IL (1) IL153476A0 (en)
MX (1) MXPA02012564A (en)
NO (1) NO324939B1 (en)
NZ (1) NZ524155A (en)
PL (1) PL358808A1 (en)
PT (1) PT1301485E (en)
RU (1) RU2267488C2 (en)
SK (1) SK1932003A3 (en)
UA (1) UA75085C2 (en)
WO (1) WO2002008194A1 (en)
ZA (1) ZA200210411B (en)

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DE10035928A1 (en) * 2000-07-21 2002-03-07 Asta Medica Ag New heteroaryl derivatives and their use as medicines
DE10037310A1 (en) * 2000-07-28 2002-02-07 Asta Medica Ag New indole derivatives and their use as medicines
EP1517898A1 (en) * 2002-06-29 2005-03-30 Zentaris GmbH Arylcarbonylpiperazines and heteroarylcarbonylpiperazines and the use thereof for treating benign and malignant tumour diseases
MXPA05000487A (en) * 2002-07-17 2005-03-23 Zentaris Gmbh Novel anthracene derivatives and the use thereof as a medicament.
US7125461B2 (en) * 2003-05-07 2006-10-24 L & L Products, Inc. Activatable material for sealing, baffling or reinforcing and method of forming same
FR2855825B1 (en) * 2003-06-04 2008-08-22 Aventis Pharma Sa ARYL-HETEROAROMATIC PRODUCTS, COMPOSITIONS CONTAINING SAME AND USE THEREOF
AR044586A1 (en) * 2003-06-04 2005-09-21 Aventis Pharma Sa ARIL PRODUCTS - HETEROAROMATICOS, COMPOSITIONS THAT CONTAIN THEM AND THEIR USE
US7249415B2 (en) * 2003-06-26 2007-07-31 Zephyros, Inc. Method of forming members for sealing or baffling
DE10331500A1 (en) * 2003-07-11 2005-02-24 Zentaris Gmbh Novel acridine derivatives and their use as pharmaceuticals
EP1853594A2 (en) * 2005-01-27 2007-11-14 Alma Mater Studiorum -Universita' di Bologna Organic compounds useful for the treatment of alzheimer's disease, their use and method of preparation
US20070299093A1 (en) * 2005-01-27 2007-12-27 Alma Mater Studiorum-Universitá Di Bologna Organic Compounds Useful for the Treatment of Alzheimer's Disease, Their Use and Method of Preparation
WO2008106128A2 (en) * 2007-02-26 2008-09-04 Vitae Pharmaceuticals, Inc. CYCLIC UREA AND CARBAMATE INHIBITORS OF 11β -HYDROXYSTEROID DEHYDROGENASE 1
ATE554078T1 (en) * 2007-07-26 2012-05-15 Vitae Pharmaceuticals Inc SYNTHESIS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE-1 INHIBITORS
AR069207A1 (en) * 2007-11-07 2010-01-06 Vitae Pharmaceuticals Inc CYCLIC UREAS AS INHIBITORS OF THE 11 BETA - HIDROXI-ESTEROIDE DESHIDROGENASA 1
EP2229368A1 (en) 2007-12-11 2010-09-22 Vitae Pharmaceuticals, Inc. Cyclic urea inhibitors of 11beta-hydroxysteroid dehydrogenase 1
TW200934490A (en) * 2008-01-07 2009-08-16 Vitae Pharmaceuticals Inc Lactam inhibitors of 11 &abgr;-hydroxysteroid dehydrogenase 1
EP2252601B1 (en) * 2008-01-24 2012-12-19 Vitae Pharmaceuticals, Inc. Cyclic carbazate and semicarbazide inhibitors of 11beta-hydroxysteroid dehydrogenase 1
CA2714532A1 (en) * 2008-02-11 2009-08-20 Vitae Pharmaceuticals, Inc. 1,3-oxazepan-2-one and 1,3-diazepan-2-one inhibitors of 11.beta.-hydroxysteroid dehydrogenase 1
JP5730021B2 (en) * 2008-02-15 2015-06-03 ヴァイティー ファーマシューティカルズ，インコーポレイテッド Cycloalkyllactam derivatives as inhibitors of 11β-hydroxysteroid dehydrogenase 1
WO2009117109A1 (en) * 2008-03-18 2009-09-24 Vitae Pharmaceuticals, Inc. Inhibitors of 11beta-hydroxysteroid dehydrogenase type 1
WO2009134387A1 (en) 2008-05-01 2009-11-05 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
JP5451752B2 (en) * 2008-05-01 2014-03-26 ヴァイティー ファーマシューティカルズ，インコーポレイテッド Cyclic inhibitor of 11β-hydroxysteroid dehydrogenase 1
WO2009134392A1 (en) 2008-05-01 2009-11-05 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
NZ588954A (en) 2008-05-01 2012-08-31 Vitae Pharmaceuticals Inc Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
PL2324018T3 (en) 2008-07-25 2014-02-28 Boehringer Ingelheim Int Cyclic inhibitors of 11 beta-hydroxysteroid dehydrogenase 1
CA2729998A1 (en) 2008-07-25 2010-01-28 Boehringer Ingelheim International Gmbh Inhibitors of 11beta-hydroxysteroid dehydrogenase 1
EP2393807B1 (en) 2009-02-04 2013-08-14 Boehringer Ingelheim International GmbH Cyclic inhibitors of 11 -hydroxysteroid dehydrogenase 1
TW201039034A (en) * 2009-04-27 2010-11-01 Chunghwa Picture Tubes Ltd Pixel structure and the method of forming the same
KR20120061771A (en) * 2009-04-30 2012-06-13 비타이 파마슈티컬즈, 인코포레이티드 Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
UA109255C2 (en) 2009-04-30 2015-08-10 Берінгер Інгельхайм Інтернешнл Гмбх Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
WO2011011123A1 (en) 2009-06-11 2011-01-27 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1 based on the 1,3 -oxazinan- 2 -one structure
JP5749263B2 (en) 2009-07-01 2015-07-15 ヴァイティー ファーマシューティカルズ，インコーポレイテッド Cyclic inhibitor of 11β-hydroxysteroid dehydrogenase 1
EP2582698B1 (en) 2010-06-16 2016-09-14 Vitae Pharmaceuticals, Inc. Substituted 5-,6- and 7-membered heterocycles, medicaments containing such compounds, and their use
WO2011161128A1 (en) 2010-06-25 2011-12-29 Boehringer Ingelheim International Gmbh Azaspirohexanones as inhibitors of 11-beta-hsd1 for the treatment of metabolic disorders
KR20130137628A (en) 2010-11-02 2013-12-17 베링거 인겔하임 인터내셔날 게엠베하 Pharmaceutical combinations for the treatment of metabolic disorders

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US4937246A (en) * 1987-11-25 1990-06-26 Takeda Chemical Industries, Ltd. PAF antagonist, 1,4-disubstituted piperazine compounds and production thereof
US5030631A (en) * 1989-11-27 1991-07-09 Schering Corporation Tricylclic arylsulfonamides
RU2126001C1 (en) * 1995-01-10 1999-02-10 Самдзин Фармасьютикал Ко., Лтд Piperazine derivatives and pharmaceutical composition on their basis
CZ59398A3 (en) * 1996-06-29 1998-07-15 Samjin Pharmaceutical Co., Ltd. Piperazine Derivatives and Process for their Preparation
US5861395A (en) 1996-09-13 1999-01-19 Schering Corporation Compounds useful for inhibition of farnesyl proteins transferase
FR2753706B1 (en) 1996-09-20 1998-10-30 NOVEL N-SUBSTITUTED CYCLIC AMINES, THEIR PREPARATION PROCESS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
DE19743435A1 (en) 1997-10-01 1999-04-08 Merck Patent Gmbh Benzamidine derivatives
BR9913654A (en) 1998-08-28 2001-11-27 Scios Inc P-38alpha kinase inhibitors
JP2002538121A (en) 1999-03-03 2002-11-12 メルク エンド カムパニー インコーポレーテッド Inhibitors of prenyl protein transferase

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