AU2001289063A1 - Novel thio derivatives of sordarin as antifungal agents - Google Patents
Novel thio derivatives of sordarin as antifungal agentsInfo
- Publication number
- AU2001289063A1 AU2001289063A1 AU2001289063A AU8906301A AU2001289063A1 AU 2001289063 A1 AU2001289063 A1 AU 2001289063A1 AU 2001289063 A AU2001289063 A AU 2001289063A AU 8906301 A AU8906301 A AU 8906301A AU 2001289063 A1 AU2001289063 A1 AU 2001289063A1
- Authority
- AU
- Australia
- Prior art keywords
- sordarin
- antifungal agents
- thio derivatives
- novel thio
- novel
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- 229940121375 antifungal agent Drugs 0.000 title 1
- 239000003429 antifungal agent Substances 0.000 title 1
- OGGVRVMISBQNMQ-UHFFFAOYSA-N sordarin Natural products OC1C(O)C(OC)C(C)OC1OCC1(C2(C(C(C)C)=C3)C(O)=O)C3CC2(C=O)C2CCC(C)C2C1 OGGVRVMISBQNMQ-UHFFFAOYSA-N 0.000 title 1
- 125000000446 sulfanediyl group Chemical group *S* 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C317/00—Sulfones; Sulfoxides
- C07C317/44—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
- C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
- C07C323/55—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being unsaturated and containing rings other than six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/04—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2603/00—Systems containing at least three condensed rings
- C07C2603/56—Ring systems containing bridged rings
- C07C2603/86—Ring systems containing bridged rings containing four rings
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Virology (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US23276200P | 2000-09-15 | 2000-09-15 | |
| US60232762 | 2000-09-15 | ||
| PCT/US2001/028604 WO2002022567A1 (en) | 2000-09-15 | 2001-09-14 | Novel thio derivatives of sordarin as antifungal agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2001289063A1 true AU2001289063A1 (en) | 2002-03-26 |
Family
ID=22874466
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2001289063A Abandoned AU2001289063A1 (en) | 2000-09-15 | 2001-09-14 | Novel thio derivatives of sordarin as antifungal agents |
Country Status (3)
| Country | Link |
|---|---|
| US (1) | US6436930B1 (en) |
| AU (1) | AU2001289063A1 (en) |
| WO (1) | WO2002022567A1 (en) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8337481B2 (en) | 2005-01-25 | 2012-12-25 | Patrick Slater | Method for treating otitis externa |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SK88496A3 (en) * | 1994-11-08 | 1997-04-09 | Glaxo Wellcome Sa | Cyclic derivatives, manufacturing process thereof, pharmaceutical compositions containing them and their use antifungal sordaridin derivatives |
| EP0711783A1 (en) * | 1994-11-08 | 1996-05-15 | Glaxo, S.A. | Antifungal Sordarin derivatives |
| US6040463A (en) * | 1996-10-07 | 2000-03-21 | Merck & Co., Inc. | Sordarin derivatives |
| EP0929217B1 (en) * | 1996-10-07 | 2004-03-03 | Merck & Co., Inc. | Sordarin derivatives |
-
2001
- 2001-09-14 WO PCT/US2001/028604 patent/WO2002022567A1/en not_active Ceased
- 2001-09-14 US US09/952,987 patent/US6436930B1/en not_active Expired - Lifetime
- 2001-09-14 AU AU2001289063A patent/AU2001289063A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2002022567A8 (en) | 2002-06-20 |
| WO2002022567A1 (en) | 2002-03-21 |
| US6436930B1 (en) | 2002-08-20 |
| US20020035073A1 (en) | 2002-03-21 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| AU2002363005A1 (en) | Derivatives of uk-2a | |
| AU2001280099A1 (en) | 4-acylaminopyrazole derivatives | |
| AU2001230584A1 (en) | 1h-imidazopyridine derivatives | |
| AU2001230537A1 (en) | Pyridoxazine derivatives | |
| AU2001281802A1 (en) | 6-phenylpyrrolopyrimidinedione derivatives | |
| AU2001278790A1 (en) | 1h-imidazopyridine derivatives | |
| AU2000223275A1 (en) | Novel triazole derivatives | |
| AU2002213978A1 (en) | Substituted C-cyclohexylmethylamine derivatives | |
| AU5682901A (en) | Fungicidal composition containing n-(alpha-cyano-2-thenyl)-4-ethyl-2-(ethylamino)-5-thiazoleca boxamide | |
| AU2002212301A1 (en) | Diazacycloalkanedione derivatives | |
| AU2002331707A1 (en) | Tetrahydroquinoline derivatives as antithrombotic agents | |
| AU2002212959A1 (en) | Cycloalkylfluorosulfonamide derivatives | |
| AU2001258841A1 (en) | Heterocyclic compounds | |
| AU2002215212A1 (en) | 1-methylcarbapenem derivatives | |
| AU2001254661A1 (en) | Aminosulfonylbiphenyl derivatives | |
| AU2001292122A1 (en) | Heterocyclic derivatives useful as pharmaceutical agents | |
| AU2001289937A1 (en) | Substituted 1-aminobutan-3-ol derivatives | |
| AU2002214024A1 (en) | Novel diaminopyrazole derivatives and dyes containing said compounds | |
| AU2002218215A1 (en) | Novel pleuromutilin derivatives | |
| AU2001230565A1 (en) | Perfluoroisopropylbenzene derivatives | |
| AU2001231173A1 (en) | Laulimalide compounds as microtubule stabilizing agents | |
| AU2001234313A1 (en) | Novel phenylheteroalkylamine derivatives | |
| AU2001282865A1 (en) | Heterocyclic sulfonamide derivatives | |
| AU2001280470A1 (en) | Heterocyclic sulfonamide derivatives | |
| AU2002363600A1 (en) | Novel phenyl-propargylether derivatives |